Compile Data Set for Download or QSAR
Report error Found 137 of ic50 data for polymerid = 49000302,49000604,49000605,50007223
TargetGastrin-releasing peptide receptor(Mouse)
Burroughs Wellcome

Curated by ChEMBL
LigandPNGBDBM50040307(1-naphthyl(CO)His-Trp-Ala-Val-DAla-His-DPro(psi)Ph...)
Affinity DataIC50: 0.00100nMAssay Description:The ability of the peptide to inhibit the binding of 50 pM [125I]gastrin releasing peptide to intact S-3T3 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetGastrin-releasing peptide receptor(Mouse)
Burroughs Wellcome

Curated by ChEMBL
LigandPNGBDBM50040317(PhCH2CH2(CO)His-Trp-Ala-Val-DAla-His-DPro(psi)Phe-...)
Affinity DataIC50: 0.00100nMAssay Description:The ability of the peptide to inhibit the binding of 50 pM [125I]gastrin releasing peptide to intact S-3T3 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetGastrin-releasing peptide receptor(Mouse)
Burroughs Wellcome

Curated by ChEMBL
LigandPNGBDBM50040299(cyclopropylbenzene(CO)His-Trp-Ala-Val-DAla-His-DPr...)
Affinity DataIC50: 0.0300nMAssay Description:The ability of the peptide to inhibit the binding of 50 pM [125I]gastrin releasing peptide to intact S-3T3 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetGastrin-releasing peptide receptor(Mouse)
Burroughs Wellcome

Curated by ChEMBL
LigandPNGBDBM50040325(PhCH2CH2(CO)His-Trp-Ala-Val-DAla-His-DPro(psi)DPhe...)
Affinity DataIC50: 0.0380nMAssay Description:Ability of peptide to inhibit binding of 10 pM [125I]gastrin releasing peptide to S-3T3 cell membrane.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetGastrin-releasing peptide receptor(Mouse)
Burroughs Wellcome

Curated by ChEMBL
LigandPNGBDBM50040299(cyclopropylbenzene(CO)His-Trp-Ala-Val-DAla-His-DPr...)
Affinity DataIC50: 0.0490nMAssay Description:Ability of peptide to inhibit binding of 10 pM [125I]gastrin releasing peptide to S-3T3 cell membrane.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetGastrin-releasing peptide receptor(Mouse)
Burroughs Wellcome

Curated by ChEMBL
LigandPNGBDBM50040307(1-naphthyl(CO)His-Trp-Ala-Val-DAla-His-DPro(psi)Ph...)
Affinity DataIC50: 0.0500nMAssay Description:Ability of peptide to inhibit binding of 10 pM [125I]gastrin releasing peptide to S-3T3 cell membrane.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetGastrin-releasing peptide receptor(Mouse)
Burroughs Wellcome

Curated by ChEMBL
LigandPNGBDBM50040301(4-OHPhCH2CH2(CO)His-Trp-Ala-Val-DAla-His-DPro(psi)...)
Affinity DataIC50: 0.0500nMAssay Description:The ability of the peptide to inhibit the binding of 50 pM [125I]gastrin releasing peptide to intact S-3T3 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetGastrin-releasing peptide receptor(Human)
National Center For Scientific Research Demokritos

Curated by ChEMBL
LigandPNGBDBM50158698([N40,Pro1,Tyr4]BB | CHEMBL266078)
Affinity DataIC50: 0.0600nMAssay Description:Displacement of [125 I-Tyr4]BB from human gastrin releasing peptide receptor expressed in PC-3 cell membranesMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetGastrin-releasing peptide receptor(Mouse)
Burroughs Wellcome

Curated by ChEMBL
LigandPNGBDBM50040312(2-tetrahydronaphthyl(CO)His-Trp-Ala-Val-DAla-His-D...)
Affinity DataIC50: 0.0790nMAssay Description:Ability of peptide to inhibit binding of 10 pM [125I]gastrin releasing peptide to S-3T3 cell membrane.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetGastrin-releasing peptide receptor(Human)
National Center For Scientific Research Demokritos

Curated by ChEMBL
LigandPNGBDBM50158699([(N4-Bzdig)0]BB(7-14) | CHEMBL414307)
Affinity DataIC50: 0.0800nMAssay Description:Displacement of [125 I-Tyr4]BB from human gastrin releasing peptide receptor expressed in PC-3 cell membranesMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetGastrin-releasing peptide receptor(Mouse)
Burroughs Wellcome

Curated by ChEMBL
LigandPNGBDBM50040308(2-aminoPhCH2(CO)His-Trp-Ala-Val-DAla-His-DPro(psi)...)
Affinity DataIC50: 0.100nMAssay Description:The ability of the peptide to inhibit the binding of 50 pM [125I]gastrin releasing peptide to intact S-3T3 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetGastrin-releasing peptide receptor(Human)
National Center For Scientific Research Demokritos

Curated by ChEMBL
LigandPNGBDBM50158697([N40,Pro1,Tyr4,Nle 14]BB | CHEMBL268222)
Affinity DataIC50: 0.150nMAssay Description:Displacement of [125 I-Tyr4]BB from human gastrin releasing peptide receptor expressed in PC-3 cell membranesMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetGastrin-releasing peptide receptor(Mouse)
Burroughs Wellcome

Curated by ChEMBL
LigandPNGBDBM50040310(3-CF3PhCH2CH2(CO)His-Trp-Ala-Val-DAla-His-DPro(psi...)
Affinity DataIC50: 0.160nMAssay Description:Ability of peptide to inhibit binding of 10 pM [125I]gastrin releasing peptide to S-3T3 cell membrane.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetGastrin-releasing peptide receptor(Mouse)
Burroughs Wellcome

Curated by ChEMBL
LigandPNGBDBM50040315((CH3)2PhC(CO)His-Trp-Ala-Val-DAla-His-DPro(psi)Phe...)
Affinity DataIC50: 0.180nMAssay Description:Ability of peptide to inhibit binding of 10 pM [125I]gastrin releasing peptide to S-3T3 cell membrane.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetGastrin-releasing peptide receptor(Mouse)
Burroughs Wellcome

Curated by ChEMBL
LigandPNGBDBM50040315((CH3)2PhC(CO)His-Trp-Ala-Val-DAla-His-DPro(psi)Phe...)
Affinity DataIC50: 0.180nMAssay Description:Ability of peptide to inhibit binding of 10 pM [125I]gastrin releasing peptide to S-3T3 cell membrane.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetGastrin-releasing peptide receptor(Mouse)
Burroughs Wellcome

Curated by ChEMBL
LigandPNGBDBM50040317(PhCH2CH2(CO)His-Trp-Ala-Val-DAla-His-DPro(psi)Phe-...)
Affinity DataIC50: 0.220nMAssay Description:Ability of peptide to inhibit binding of 10 pM [125I]gastrin releasing peptide to S-3T3 cell membrane.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetGastrin-releasing peptide receptor(Mouse)
Burroughs Wellcome

Curated by ChEMBL
LigandPNGBDBM50040301(4-OHPhCH2CH2(CO)His-Trp-Ala-Val-DAla-His-DPro(psi)...)
Affinity DataIC50: 0.230nMAssay Description:Ability of peptide to inhibit binding of 10 pM [125I]gastrin releasing peptide to S-3T3 cell membrane.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetGastrin-releasing peptide receptor(Mouse)
Burroughs Wellcome

Curated by ChEMBL
LigandPNGBDBM50040312(2-tetrahydronaphthyl(CO)His-Trp-Ala-Val-DAla-His-D...)
Affinity DataIC50: 0.300nMAssay Description:The ability of the peptide to inhibit the binding of 50 pM [125I]gastrin releasing peptide to intact S-3T3 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetGastrin-releasing peptide receptor(Mouse)
Burroughs Wellcome

Curated by ChEMBL
LigandPNGBDBM50040320(PhCH2CH2(CO)His-Trp-Ala-Val-DAla-His-DPro(psi)Tyr-...)
Affinity DataIC50: 0.330nMAssay Description:Ability of peptide to inhibit binding of 10 pM [125I]gastrin releasing peptide to S-3T3 cell membrane.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetGastrin-releasing peptide receptor(Human)
National Center For Scientific Research Demokritos

Curated by ChEMBL
LigandPNGBDBM50158698([N40,Pro1,Tyr4]BB | CHEMBL266078)
Affinity DataIC50: 0.470nMAssay Description:Inhibition of gastrin releasing peptide receptor expressed in human prostate cancer cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetGastrin-releasing peptide receptor(Mouse)
Burroughs Wellcome

Curated by ChEMBL
LigandPNGBDBM50407275(CHEMBL2112786)
Affinity DataIC50: 0.490nMAssay Description:Ability of peptide to inhibit binding of 10 pM [125I]gastrin releasing peptide to S-3T3 cell membrane.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetGastrin-releasing peptide receptor(Mouse)
Burroughs Wellcome

Curated by ChEMBL
LigandPNGBDBM50040316(3-isoquinolyl(CO)His-Trp-Ala-Val-DAla-His-DPro(psi...)
Affinity DataIC50: 0.570nMAssay Description:Ability of peptide to inhibit binding of 10 pM [125I]gastrin releasing peptide to S-3T3 cell membrane.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetGastrin-releasing peptide receptor(Human)
National Center For Scientific Research Demokritos

Curated by ChEMBL
LigandPNGBDBM50279041((2S)-N1-((5S,8S,11S,17S,20S,23S,26S,29S,35S,38S)-1...)
Affinity DataIC50: 0.590nMAssay Description:Displacement of [125I-Tyr4]BN form BB2 receptor in human PC3 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetGastrin-releasing peptide receptor(Mouse)
Burroughs Wellcome

Curated by ChEMBL
LigandPNGBDBM50012304(2-{2-[2-[2-(2,2-Dimethyl-propionylamino)-3-(3H-imi...)
Affinity DataIC50: 0.600nMAssay Description:Compound was evaluated for mitogenic inhibition against Swiss 3T3 murine fibroblast cells.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetGastrin-releasing peptide receptor(Human)
National Center For Scientific Research Demokritos

Curated by ChEMBL
LigandPNGBDBM50158700([(N4-Bzdig)0,Nle14]BB(7-14) | CHEMBL266079)
Affinity DataIC50: 0.600nMAssay Description:Displacement of [125 I-Tyr4]BB from human gastrin releasing peptide receptor expressed in PC-3 cell membranesMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetGastrin-releasing peptide receptor(Human)
National Center For Scientific Research Demokritos

Curated by ChEMBL
LigandPNGBDBM50066009(CHEMBL3401466)
Affinity DataIC50: 0.600nMAssay Description:Displacement of [125I-Tyr4]bombesin from GRPR (unknown origin) expressed in human PC3 cells after 45 mins by gamma counting analysisMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetGastrin-releasing peptide receptor(Human)
National Center For Scientific Research Demokritos

Curated by ChEMBL
LigandPNGBDBM50158699([(N4-Bzdig)0]BB(7-14) | CHEMBL414307)
Affinity DataIC50: 0.650nMAssay Description:Inhibition of gastrin releasing peptide receptor expressed in human prostate cancer cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetGastrin-releasing peptide receptor(Human)
National Center For Scientific Research Demokritos

Curated by ChEMBL
LigandPNGBDBM50158702(Universal ligand | CHEMBL413893)
Affinity DataIC50: 0.720nMAssay Description:Inhibition of gastrin releasing peptide receptor expressed in human prostate cancer cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetGastrin-releasing peptide receptor(Mouse)
Burroughs Wellcome

Curated by ChEMBL
LigandPNGBDBM50040324(PhCH2CH2(CO)His-(BzthAla)-Ala-Val-DAla-His-Pro(psi...)
Affinity DataIC50: 0.75nMAssay Description:Ability of peptide to inhibit binding of 10 pM [125I]gastrin releasing peptide to S-3T3 cell membrane.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetGastrin-releasing peptide receptor(Human)
National Center For Scientific Research Demokritos

Curated by ChEMBL
LigandPNGBDBM50158701([Tyr4]Bombesin | CHEMBL407101)
Affinity DataIC50: 0.850nMAssay Description:Displacement of [125 I-Tyr4]BB from human gastrin releasing peptide receptor expressed in PC-3 cell membranesMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetGastrin-releasing peptide receptor(Mouse)
Burroughs Wellcome

Curated by ChEMBL
LigandPNGBDBM50407276(CHEMBL2111952)
Affinity DataIC50: 1nMAssay Description:The ability of the peptide to inhibit the binding of 50 pM [125I]gastrin releasing peptide to intact S-3T3 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetGastrin-releasing peptide receptor(Mouse)
Burroughs Wellcome

Curated by ChEMBL
LigandPNGBDBM50407273(CHEMBL2111953)
Affinity DataIC50: 1nMAssay Description:The ability of the peptide to inhibit the binding of 50 pM [125I]gastrin releasing peptide to intact S-3T3 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetGastrin-releasing peptide receptor(Mouse)
Burroughs Wellcome

Curated by ChEMBL
LigandPNGBDBM50040310(3-CF3PhCH2CH2(CO)His-Trp-Ala-Val-DAla-His-DPro(psi...)
Affinity DataIC50: 1nMAssay Description:The ability of the peptide to inhibit the binding of 50 pM [125I]gastrin releasing peptide to intact S-3T3 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetGastrin-releasing peptide receptor(Mouse)
Burroughs Wellcome

Curated by ChEMBL
LigandPNGBDBM50407276(CHEMBL2111952)
Affinity DataIC50: 1nMAssay Description:The ability of the peptide to inhibit the binding of 50 pM [125I]gastrin releasing peptide to intact S-3T3 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetGastrin-releasing peptide receptor(Rat)
Washington University

Curated by ChEMBL
LigandPNGBDBM50112639(pQ-Q-R-Y-G-N-Q-W-A-V-G-H-L-M-NH2 | CHEMBL402688)
Affinity DataIC50: 1.10nMAssay Description:In vitro binding affinity of [111In]DTPA-[Y4]-bombesin to bombesin receptor in the rat pancreatic acinar cell line, AR42JMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetGastrin-releasing peptide receptor(Mouse)
Burroughs Wellcome

Curated by ChEMBL
LigandPNGBDBM50012313(2-{2-[2-[2-Acetylamino-3-(3H-imidazol-4-yl)-propio...)
Affinity DataIC50: 1.20nMAssay Description:Inhibition against Swiss 3T3 murine fibroblast cells.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetGastrin-releasing peptide receptor(Mouse)
Burroughs Wellcome

Curated by ChEMBL
LigandPNGBDBM50040314((CH3)2PhCCH2(CO)His-Trp-Ala-Val-DAla-His-DPro(psi)...)
Affinity DataIC50: 1.20nMAssay Description:Ability of peptide to inhibit binding of 10 pM [125I]gastrin releasing peptide to S-3T3 cell membrane.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetGastrin-releasing peptide receptor(Human)
National Center For Scientific Research Demokritos

Curated by ChEMBL
LigandPNGBDBM50279043((S)-N1-((5S,8S,11S,17S,20S,23S,26S,29S,35S,38S)-11...)
Affinity DataIC50: 1.24nMAssay Description:Displacement of [125I-Tyr4]BN form BB2 receptor in human PC3 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetGastrin-releasing peptide receptor(Human)
National Center For Scientific Research Demokritos

Curated by ChEMBL
LigandPNGBDBM50158700([(N4-Bzdig)0,Nle14]BB(7-14) | CHEMBL266079)
Affinity DataIC50: 1.30nMAssay Description:Inhibition of gastrin releasing peptide receptor expressed in human prostate cancer cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetGastrin-releasing peptide receptor(Mouse)
Burroughs Wellcome

Curated by ChEMBL
LigandPNGBDBM50407273(CHEMBL2111953)
Affinity DataIC50: 1.30nMAssay Description:Ability of peptide to inhibit binding of 10 pM [125I]gastrin releasing peptide to S-3T3 cell membrane.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetGastrin-releasing peptide receptor(Mouse)
Burroughs Wellcome

Curated by ChEMBL
LigandPNGBDBM50012318(2-{2-[2-[2-Acetylamino-3-(3H-imidazol-4-yl)-propio...)
Affinity DataIC50: 1.40nMAssay Description:Inhibition against Swiss 3T3 murine fibroblast cells.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetGastrin-releasing peptide receptor(Human)
National Center For Scientific Research Demokritos

Curated by ChEMBL
LigandPNGBDBM50279042((2S)-N1-((5S,8S,11S,17S,20S,23S)-11-((1H-imidazol-...)
Affinity DataIC50: 1.45nMAssay Description:Displacement of [125I-Tyr4]BN form BB2 receptor in human PC3 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetGastrin-releasing peptide receptor(Mouse)
Burroughs Wellcome

Curated by ChEMBL
LigandPNGBDBM50012306(CHEMBL274874 | Ac-His-Trp-Ala-Val-Gly-His-Leu-Met-...)
Affinity DataIC50: 1.80nMAssay Description:Inhibition against Swiss 3T3 murine fibroblast cells.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetGastrin-releasing peptide receptor(Mouse)
Burroughs Wellcome

Curated by ChEMBL
LigandPNGBDBM50012304(2-{2-[2-[2-(2,2-Dimethyl-propionylamino)-3-(3H-imi...)
Affinity DataIC50: 1.80nMAssay Description:Inhibition against Swiss 3T3 murine fibroblast cells.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetGastrin-releasing peptide receptor(Rat)
Washington University

Curated by ChEMBL
LigandPNGBDBM50112626(Carbocyanine derivative | CHEMBL442514)
Affinity DataIC50: 1.80nMAssay Description:In vitro binding affinity of [111In]DTPA-[Y4]-bombesin to bombesin receptor in the rat pancreatic acinar cell line, AR42JMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetGastrin-releasing peptide receptor(Mouse)
Burroughs Wellcome

Curated by ChEMBL
LigandPNGBDBM50040323(phenothiazoneCH2CH2(CO)His-Trp-Ala-Val-DAla-His-DP...)
Affinity DataIC50: 1.90nMAssay Description:Ability of peptide to inhibit binding of 10 pM [125I]gastrin releasing peptide to S-3T3 cell membrane.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetGastrin-releasing peptide receptor(Human)
National Center For Scientific Research Demokritos

Curated by ChEMBL
LigandPNGBDBM50158697([N40,Pro1,Tyr4,Nle 14]BB | CHEMBL268222)
Affinity DataIC50: 1.94nMAssay Description:Inhibition of gastrin releasing peptide receptor expressed in human prostate cancer cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetGastrin-releasing peptide receptor(Mouse)
Burroughs Wellcome

Curated by ChEMBL
LigandPNGBDBM50012317(2-{2-[2-[2-Acetylamino-3-(3H-imidazol-4-yl)-propio...)
Affinity DataIC50: 2nMAssay Description:Inhibition against Swiss 3T3 murine fibroblast cells.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetGastrin-releasing peptide receptor(Mouse)
Burroughs Wellcome

Curated by ChEMBL
LigandPNGBDBM50040308(2-aminoPhCH2(CO)His-Trp-Ala-Val-DAla-His-DPro(psi)...)
Affinity DataIC50: 2nMAssay Description:Ability of peptide to inhibit binding of 10 pM [125I]gastrin releasing peptide to S-3T3 cell membrane.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetGastrin-releasing peptide receptor(Mouse)
Burroughs Wellcome

Curated by ChEMBL
LigandPNGBDBM50040298(PhCH2CH2(CO)His-Trp-Ala-Val-DAla-His-DPro(psi)D2Na...)
Affinity DataIC50: 2nMAssay Description:Ability of peptide to inhibit binding of 10 pM [125I]gastrin releasing peptide to S-3T3 cell membrane.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
Displayed 1 to 50 (of 137 total ) | Next | Last >>
Jump to: