Compile Data Set for Download or QSAR
Report error Found 78 of ic50 data for polymerid = 49000301,49000813
TargetNeuromedin-B receptor(Human)
Cambridge University Forvie Site

Curated by ChEMBL
LigandPNGBDBM50071739((S)-3-(1H-Indol-3-yl)-N-[1-(5-methoxy-pyridin-2-yl...)
Affinity DataIC50: 0.660nMAssay Description:Antagonistic activity against labelled Bombesin receptor bb1 binding sites in rat olfactory bulb by using [125I]- [Tyr] bombesin in presence of [D-Ph...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetNeuromedin-B receptor(Human)
Cambridge University Forvie Site

Curated by ChEMBL
LigandPNGBDBM50158699([(N4-Bzdig)0]BB(7-14) | CHEMBL414307)
Affinity DataIC50: 0.900nMAssay Description:Inhibition of tachykinin receptor 3 expressed in human ileal carcinoid cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetNeuromedin-B receptor(Human)
Cambridge University Forvie Site

Curated by ChEMBL
LigandPNGBDBM50158702(Universal ligand | CHEMBL413893)
Affinity DataIC50: 0.960nMAssay Description:Inhibition of tachykinin receptor 3 expressed in human ileal carcinoid cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetNeuromedin-B receptor(Human)
Cambridge University Forvie Site

Curated by ChEMBL
LigandPNGBDBM50158698([N40,Pro1,Tyr4]BB | CHEMBL266078)
Affinity DataIC50: 1.60nMAssay Description:Inhibition of tachykinin receptor 3 expressed in human ileal carcinoid cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetNeuromedin-B receptor(Human)
Cambridge University Forvie Site

Curated by ChEMBL
LigandPNGBDBM50158700([(N4-Bzdig)0,Nle14]BB(7-14) | CHEMBL266079)
Affinity DataIC50: 2nMAssay Description:Inhibition of tachykinin receptor 3 expressed in human ileal carcinoid cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetNeuromedin-B receptor(Human)
Cambridge University Forvie Site

Curated by ChEMBL
LigandPNGBDBM50158697([N40,Pro1,Tyr4,Nle 14]BB | CHEMBL268222)
Affinity DataIC50: 11.2nMAssay Description:Inhibition of tachykinin receptor 3 expressed in human ileal carcinoid cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetNeuromedin-B receptor(Human)
Cambridge University Forvie Site

Curated by ChEMBL
LigandPNGBDBM50147019(3-[3-(2,6-Diisopropyl-phenyl)-ureido]-5-methoxy-2,...)
Affinity DataIC50: 29nMAssay Description:Affinity of [125I][D-Tyr0]-NMB to human Neuromedin B receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetNeuromedin-B receptor(Human)
Cambridge University Forvie Site

Curated by ChEMBL
LigandPNGBDBM50147019(3-[3-(2,6-Diisopropyl-phenyl)-ureido]-5-methoxy-2,...)
Affinity DataIC50: 29nMAssay Description:Affinity of [125I][D-Tyr0]-NMB to human Neuromedin B receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetNeuromedin-B receptor(Human)
Cambridge University Forvie Site

Curated by ChEMBL
LigandPNGBDBM50295231((-)-8'-methyl-11'-(2-(trifluoromethyl)phenyl)-4',5...)
Affinity DataIC50: 96nMAssay Description:Displacement of [125I]-(D-Tyr0)NMB from human neuromedin B receptor transfected in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetNeuromedin-B receptor(Human)
Cambridge University Forvie Site

Curated by ChEMBL
LigandPNGBDBM50295231((-)-8'-methyl-11'-(2-(trifluoromethyl)phenyl)-4',5...)
Affinity DataIC50: 96nMAssay Description:Displacement of [125I]-(D-Tyr0)NMB from human neuromedin B receptor transfected in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetNeuromedin-B receptor(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50071754(Xenopus NMB | CHEMBL86828 | NMB | (S)-2-[3-(2,6-Di...)
Affinity DataIC50: 150nMAssay Description:Binding affinity against NMB receptor in rat olfactory bulb was determined using [125I]-[Tyr4] bombesin.More data for this Ligand-Target Pair
In DepthDetails Article

TargetNeuromedin-B receptor(Human)
Cambridge University Forvie Site

Curated by ChEMBL
LigandPNGBDBM50295222(10-butyl-11-(2-chloro-6-fluorophenyl)-3,3,8-trimet...)
Affinity DataIC50: 150nMAssay Description:Displacement of [125I]-(D-Tyr0)NMB from human neuromedin B receptor transfected in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetNeuromedin-B receptor(Human)
Cambridge University Forvie Site

Curated by ChEMBL
LigandPNGBDBM50295254(11-(2-chloro-6-fluorophenyl)-3,3,8,10-tetramethyl-...)
Affinity DataIC50: 170nMAssay Description:Displacement of [125I]-(D-Tyr0)NMB from human neuromedin B receptor transfected in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetNeuromedin-B receptor(Human)
Cambridge University Forvie Site

Curated by ChEMBL
LigandPNGBDBM50295221(11-(2-chloro-6-fluorophenyl)-10-ethyl-3,3,8-trimet...)
Affinity DataIC50: 180nMAssay Description:Displacement of [125I]-(D-Tyr0)NMB from human neuromedin B receptor transfected in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetNeuromedin-B receptor(Human)
Cambridge University Forvie Site

Curated by ChEMBL
LigandPNGBDBM50295245(3,3,8-trimethyl-11-(2-(methylthio)phenyl)-2,3,4,5,...)
Affinity DataIC50: 200nMAssay Description:Displacement of [125I]-(D-Tyr0)NMB from human neuromedin B receptor transfected in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetNeuromedin-B receptor(Human)
Cambridge University Forvie Site

Curated by ChEMBL
LigandPNGBDBM50295232(11'-(2-chlorophenyl)-8'-methyl-4',5',10',11'-tetra...)
Affinity DataIC50: 240nMAssay Description:Displacement of [125I]-(D-Tyr0)NMB from human neuromedin B receptor transfected in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetNeuromedin-B receptor(Human)
Cambridge University Forvie Site

Curated by ChEMBL
LigandPNGBDBM50295233(8'-methyl-11'-(2-(methylthio)phenyl)-4',5',10',11'...)
Affinity DataIC50: 250nMAssay Description:Displacement of [125I]-(D-Tyr0)NMB from human neuromedin B receptor transfected in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetNeuromedin-B receptor(Human)
Cambridge University Forvie Site

Curated by ChEMBL
LigandPNGBDBM50295246(3,3,8-trimethyl-11-(2-(trifluoromethyl)phenyl)-2,3...)
Affinity DataIC50: 250nMAssay Description:Displacement of [125I]-(D-Tyr0)NMB from human neuromedin B receptor transfected in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetNeuromedin-B receptor(Human)
Cambridge University Forvie Site

Curated by ChEMBL
LigandPNGBDBM50295223(11'-(2-chloro-6-fluorophenyl)-8'-methyl-4',5',10',...)
Affinity DataIC50: 280nMAssay Description:Displacement of [125I]-(D-Tyr0)NMB from human neuromedin B receptor transfected in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetNeuromedin-B receptor(Human)
Cambridge University Forvie Site

Curated by ChEMBL
LigandPNGBDBM50295247(11-(2-chlorophenyl)-3,3,8-trimethyl-2,3,4,5,10,11-...)
Affinity DataIC50: 280nMAssay Description:Displacement of [125I]-(D-Tyr0)NMB from human neuromedin B receptor transfected in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetNeuromedin-B receptor(Human)
Cambridge University Forvie Site

Curated by ChEMBL
LigandPNGBDBM50295236(11-(2-chloro-6-fluorophenyl)-3,3,8-trimethyl-2,3,4...)
Affinity DataIC50: 300nMAssay Description:Displacement of [125I]-(D-Tyr0)NMB from human neuromedin B receptor transfected in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetNeuromedin-B receptor(Human)
Cambridge University Forvie Site

Curated by ChEMBL
LigandPNGBDBM50147021(3-[3-(2,6-Diisopropyl-phenyl)-ureido]-2,3,4,9-tetr...)
Affinity DataIC50: 320nMAssay Description:Affinity of [125I][D-Tyr0]-NMB to human Neuromedin B receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetNeuromedin-B receptor(Human)
Cambridge University Forvie Site

Curated by ChEMBL
LigandPNGBDBM50071754(Xenopus NMB | CHEMBL86828 | NMB | (S)-2-[3-(2,6-Di...)
Affinity DataIC50: 350nMAssay Description:Agonistic activity was determined against human Neuromedin B receptor transfected in HEK293 cells as accumulation levels of inositol phosphateMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetNeuromedin-B receptor(Human)
Cambridge University Forvie Site

Curated by ChEMBL
LigandPNGBDBM50295237(11-(2-chloro-6-fluorophenyl)-3,3-dimethyl-8-(trifl...)
Affinity DataIC50: 370nMAssay Description:Displacement of [125I]-(D-Tyr0)NMB from human neuromedin B receptor transfected in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetNeuromedin-B receptor(Human)
Cambridge University Forvie Site

Curated by ChEMBL
LigandPNGBDBM50295224(11-(2-chloro-6-fluorophenyl)-3,8-dimethyl-2,3,4,5,...)
Affinity DataIC50: 450nMAssay Description:Displacement of [125I]-(D-Tyr0)NMB from human neuromedin B receptor transfected in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetNeuromedin-B receptor(Human)
Cambridge University Forvie Site

Curated by ChEMBL
LigandPNGBDBM50295234(11'-(2-fluoro-6-(trifluoromethyl)phenyl)-8'-methyl...)
Affinity DataIC50: 540nMAssay Description:Displacement of [125I]-(D-Tyr0)NMB from human neuromedin B receptor transfected in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetNeuromedin-B receptor(Human)
Cambridge University Forvie Site

Curated by ChEMBL
LigandPNGBDBM50295248(3,3,8-trimethyl-11-(2-nitrophenyl)-2,3,4,5,10,11-h...)
Affinity DataIC50: 550nMAssay Description:Displacement of [125I]-(D-Tyr0)NMB from human neuromedin B receptor transfected in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetNeuromedin-B receptor(Human)
Cambridge University Forvie Site

Curated by ChEMBL
LigandPNGBDBM50295231((-)-8'-methyl-11'-(2-(trifluoromethyl)phenyl)-4',5...)
Affinity DataIC50: 580nMAssay Description:Antagonist activity at human neuromedin B receptor transfected in HEK293 cells assessed as inhibition of 1 nM neuromedin B-induced myo-[3H]inositol p...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetNeuromedin-B receptor(Human)
Cambridge University Forvie Site

Curated by ChEMBL
LigandPNGBDBM50147035(3-[3-(2-Methyl-4-nitro-phenyl)-ureido]-2,3,4,9-tet...)
Affinity DataIC50: 620nMAssay Description:Agonistic activity was determined against human Neuromedin B receptor transfected in HEK293 cells as accumulation levels of inositol phosphateMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetNeuromedin-B receptor(Human)
Cambridge University Forvie Site

Curated by ChEMBL
LigandPNGBDBM50295235(8'-methyl-11'-(2-(trifluoromethylthio)phenyl)-4',5...)
Affinity DataIC50: 640nMAssay Description:Displacement of [125I]-(D-Tyr0)NMB from human neuromedin B receptor transfected in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetNeuromedin-B receptor(Human)
Cambridge University Forvie Site

Curated by ChEMBL
LigandPNGBDBM50147043(3-[3-(2,6-Diisopropyl-phenyl)-ureido]-5-methyl-2,3...)
Affinity DataIC50: 660nMAssay Description:Agonistic activity was determined against human Neuromedin B receptor transfected in HEK293 cells as accumulation levels of inositol phosphateMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetNeuromedin-B receptor(Human)
Cambridge University Forvie Site

Curated by ChEMBL
LigandPNGBDBM50147036(3-[3-(2,6-Diisopropyl-phenyl)-ureido]-4,6-dimethyl...)
Affinity DataIC50: 700nMAssay Description:Affinity of [125I][D-Tyr0]-NMB to human Neuromedin B receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetNeuromedin-B receptor(Human)
Cambridge University Forvie Site

Curated by ChEMBL
LigandPNGBDBM50147036(3-[3-(2,6-Diisopropyl-phenyl)-ureido]-4,6-dimethyl...)
Affinity DataIC50: 700nMAssay Description:Agonistic activity was determined against human Neuromedin B receptor transfected in HEK293 cells as accumulation levels of inositol phosphateMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetNeuromedin-B receptor(Human)
Cambridge University Forvie Site

Curated by ChEMBL
LigandPNGBDBM50147031(3-[3-(4-Nitro-phenyl)-ureido]-2,3,4,9-tetrahydro-1...)
Affinity DataIC50: 800nMAssay Description:Agonistic activity was determined against human Neuromedin B receptor transfected in HEK293 cells as accumulation levels of inositol phosphateMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetNeuromedin-B receptor(Human)
Cambridge University Forvie Site

Curated by ChEMBL
LigandPNGBDBM50295225(11-(2-chloro-6-fluorophenyl)-3-isopropyl-8-methyl-...)
Affinity DataIC50: 810nMAssay Description:Displacement of [125I]-(D-Tyr0)NMB from human neuromedin B receptor transfected in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetNeuromedin-B receptor(Human)
Cambridge University Forvie Site

Curated by ChEMBL
LigandPNGBDBM50295238(8-chloro-11-(2-chloro-6-fluorophenyl)-3,3-dimethyl...)
Affinity DataIC50: 860nMAssay Description:Displacement of [125I]-(D-Tyr0)NMB from human neuromedin B receptor transfected in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetNeuromedin-B receptor(Human)
Cambridge University Forvie Site

Curated by ChEMBL
LigandPNGBDBM50147023(3-[3-(2,6-Diisopropyl-phenyl)-ureido]-4,7-difluoro...)
Affinity DataIC50: 1.01E+3nMAssay Description:Agonistic activity was determined against human Neuromedin B receptor transfected in HEK293 cells as accumulation levels of inositol phosphateMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetNeuromedin-B receptor(Human)
Cambridge University Forvie Site

Curated by ChEMBL
LigandPNGBDBM50295249(11-(2-methoxyphenyl)-3,3,8-trimethyl-2,3,4,5,10,11...)
Affinity DataIC50: 1.10E+3nMAssay Description:Displacement of [125I]-(D-Tyr0)NMB from human neuromedin B receptor transfected in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetNeuromedin-B receptor(Human)
Cambridge University Forvie Site

Curated by ChEMBL
LigandPNGBDBM50147041(3-[3-(4-Trifluoromethyl-phenyl)-ureido]-2,3,4,9-te...)
Affinity DataIC50: 1.11E+3nMAssay Description:Agonistic activity was determined against human Neuromedin B receptor transfected in HEK293 cells as accumulation levels of inositol phosphateMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetNeuromedin-B receptor(Human)
Cambridge University Forvie Site

Curated by ChEMBL
LigandPNGBDBM50295239(11-(2-chloro-6-fluorophenyl)-3,3-dimethyl-8-(trifl...)
Affinity DataIC50: 1.30E+3nMAssay Description:Displacement of [125I]-(D-Tyr0)NMB from human neuromedin B receptor transfected in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetNeuromedin-B receptor(Human)
Cambridge University Forvie Site

Curated by ChEMBL
LigandPNGBDBM50295250(11-(2-fluorophenyl)-3,3,8-trimethyl-2,3,4,5,10,11-...)
Affinity DataIC50: 1.30E+3nMAssay Description:Displacement of [125I]-(D-Tyr0)NMB from human neuromedin B receptor transfected in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetNeuromedin-B receptor(Human)
Cambridge University Forvie Site

Curated by ChEMBL
LigandPNGBDBM50295240(11-(2-chloro-6-fluorophenyl)-3,3-dimethyl-1-oxo-2,...)
Affinity DataIC50: 1.30E+3nMAssay Description:Displacement of [125I]-(D-Tyr0)NMB from human neuromedin B receptor transfected in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetNeuromedin-B receptor(Human)
Cambridge University Forvie Site

Curated by ChEMBL
LigandPNGBDBM50295226(11-(2-chloro-6-fluorophenyl)-8-methyl-2,3,4,5,10,1...)
Affinity DataIC50: 1.40E+3nMAssay Description:Displacement of [125I]-(D-Tyr0)NMB from human neuromedin B receptor transfected in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetNeuromedin-B receptor(Human)
Cambridge University Forvie Site

Curated by ChEMBL
LigandPNGBDBM50147029(5-(3-{3-[(1-Pyridin-2-yl-cyclohexylmethyl)-carbamo...)
Affinity DataIC50: 1.85E+3nMAssay Description:Agonistic activity was determined against human Neuromedin B receptor transfected in HEK293 cells as accumulation levels of inositol phosphateMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetNeuromedin-B receptor(Human)
Cambridge University Forvie Site

Curated by ChEMBL
LigandPNGBDBM50147040(3-[3-(2,6-Diisopropyl-phenyl)-ureido]-5-trifluorom...)
Affinity DataIC50: 1.89E+3nMAssay Description:Agonistic activity was determined against human Neuromedin B receptor transfected in HEK293 cells as accumulation levels of inositol phosphateMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetNeuromedin-B receptor(Human)
Cambridge University Forvie Site

Curated by ChEMBL
LigandPNGBDBM50295227(11-(2-chloro-6-fluorophenyl)-3-(4-methoxyphenyl)-8...)
Affinity DataIC50: 2.00E+3nMAssay Description:Displacement of [125I]-(D-Tyr0)NMB from human neuromedin B receptor transfected in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetNeuromedin-B receptor(Human)
Cambridge University Forvie Site

Curated by ChEMBL
LigandPNGBDBM50147028(7-Bromo-3-[3-(2,6-diisopropyl-phenyl)-ureido]-2,3,...)
Affinity DataIC50: 2.14E+3nMAssay Description:Agonistic activity was determined against human Neuromedin B receptor transfected in HEK293 cells as accumulation levels of inositol phosphateMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetNeuromedin-B receptor(Human)
Cambridge University Forvie Site

Curated by ChEMBL
LigandPNGBDBM50295241(11-(2-chloro-6-fluorophenyl)-8-methoxy-3,3-dimethy...)
Affinity DataIC50: 2.20E+3nMAssay Description:Displacement of [125I]-(D-Tyr0)NMB from human neuromedin B receptor transfected in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetNeuromedin-B receptor(Human)
Cambridge University Forvie Site

Curated by ChEMBL
LigandPNGBDBM50147020(3-[3-(3-Acetyl-phenyl)-ureido]-2,3,4,9-tetrahydro-...)
Affinity DataIC50: 2.27E+3nMAssay Description:Agonistic activity was determined against human Neuromedin B receptor transfected in HEK293 cells as accumulation levels of inositol phosphateMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetNeuromedin-B receptor(Human)
Cambridge University Forvie Site

Curated by ChEMBL
LigandPNGBDBM50295251(11-(2,6-difluorophenyl)-3,3,8-trimethyl-2,3,4,5,10...)
Affinity DataIC50: 2.50E+3nMAssay Description:Displacement of [125I]-(D-Tyr0)NMB from human neuromedin B receptor transfected in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
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