Report error Found 52 of ic50 data for polymerid = 4840,50007698
TargetShort transient receptor potential channel 4(Human)
University of Nebraska Medical Center
Curated by ChEMBL
University of Nebraska Medical Center
Curated by ChEMBL
Affinity DataIC50: 0.0120nMAssay Description:Inhibition of human TRPC4 expressed in HEK293 cells assessed as reduction in sphingosine-1-phosphate-induced current at -100 mV by patch clamp assayMore data for this Ligand-Target Pair
TargetShort transient receptor potential channel 4(Human)
University of Nebraska Medical Center
Curated by ChEMBL
University of Nebraska Medical Center
Curated by ChEMBL
Affinity DataIC50: 0.0300nMAssay Description:Inhibition of human TRPC4 expressed in HEK293 cells assessed as reduction in sphingosine-1-phosphate-induced current at +100 mV by patch clamp assayMore data for this Ligand-Target Pair
TargetShort transient receptor potential channel 4(Human)
University of Nebraska Medical Center
Curated by ChEMBL
University of Nebraska Medical Center
Curated by ChEMBL
Affinity DataIC50: 0.340nMAssay Description:Inhibition of human TRPC4 expressed in HEK293 cells assessed as reduction in englerin A-induced calcium entry incubated for 30 mins by Fluo-4AM dye b...More data for this Ligand-Target Pair
TargetShort transient receptor potential channel 4(Human)
University of Nebraska Medical Center
Curated by ChEMBL
University of Nebraska Medical Center
Curated by ChEMBL
Affinity DataIC50: 46nMAssay Description:Inhibition of human TRPC4 expressed in human T-REx-293 cells coexpressing M1 receptor assessed as reduction in calcium influx by Fluo-4AM dye based a...More data for this Ligand-Target Pair
TargetShort transient receptor potential channel 4(Human)
University of Nebraska Medical Center
Curated by ChEMBL
University of Nebraska Medical Center
Curated by ChEMBL
Affinity DataIC50: 65nMAssay Description:Inhibition of TRPC4 channel (unknown origin) expressed in HEK293 cells assessed as inhibition of EA-evoked Ca2+ entry by measuring reduction in intra...More data for this Ligand-Target Pair
TargetShort transient receptor potential channel 4(Human)
University of Nebraska Medical Center
Curated by ChEMBL
University of Nebraska Medical Center
Curated by ChEMBL
Affinity DataIC50: 290nMAssay Description:Inhibition of Englerin-activated human TRPC4 channel expressed in HEK293 cells by Q-patch clamp assayMore data for this Ligand-Target Pair
TargetShort transient receptor potential channel 4(Mouse)
Johns Hopkins Ion Channel Center
Curated by PubChem BioAssay
Johns Hopkins Ion Channel Center
Curated by PubChem BioAssay
Affinity DataIC50: 900nMAssay Description:The inhibitory effects of test compounds on TRPC4 channels were evaluated in electrophysiological assays using a QPatch16 automated electrophysiology...More data for this Ligand-Target Pair
TargetShort transient receptor potential channel 4(Mouse)
Johns Hopkins Ion Channel Center
Curated by PubChem BioAssay
Johns Hopkins Ion Channel Center
Curated by PubChem BioAssay
Affinity DataIC50: 960nMAssay Description:Inhibition of mouse TRPC4 beta expressed in HEK293 cells co-expressing mu-opioid receptor assessed as reduction in DAMGO-induced intracellular calciu...More data for this Ligand-Target Pair
TargetShort transient receptor potential channel 4(Mouse)
Johns Hopkins Ion Channel Center
Curated by PubChem BioAssay
Johns Hopkins Ion Channel Center
Curated by PubChem BioAssay
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibition of mouse TRPC4 expressed in HEK293 cells coexpressing M5 receptor assessed as reduction in TRPC4-mediated calcium influx by fluorescence m...More data for this Ligand-Target Pair
TargetShort transient receptor potential channel 4(Mouse)
Johns Hopkins Ion Channel Center
Curated by PubChem BioAssay
Johns Hopkins Ion Channel Center
Curated by PubChem BioAssay
Affinity DataIC50: 1.63E+3nMAssay Description:The inhibitory effects of test compounds on TRPC4 channels were evaluated in electrophysiological assays using a QPatch16 automated electrophysiology...More data for this Ligand-Target Pair
TargetShort transient receptor potential channel 4(Mouse)
Johns Hopkins Ion Channel Center
Curated by PubChem BioAssay
Johns Hopkins Ion Channel Center
Curated by PubChem BioAssay
Affinity DataIC50: 1.96E+3nMAssay Description:The inhibitory effects of test compounds on TRPC4 channels were evaluated in electrophysiological assays using a QPatch16 automated electrophysiology...More data for this Ligand-Target Pair
TargetShort transient receptor potential channel 4(Mouse)
Johns Hopkins Ion Channel Center
Curated by PubChem BioAssay
Johns Hopkins Ion Channel Center
Curated by PubChem BioAssay
Affinity DataIC50: 2.05E+3nMAssay Description:Data Source: Johns Hopkins Ion Channel Center BioAssay Type: Confirmatory, Concentration-Response Relationship Observed Source (MLPCN Center Name): ...More data for this Ligand-Target Pair
TargetShort transient receptor potential channel 4(Human)
University of Nebraska Medical Center
Curated by ChEMBL
University of Nebraska Medical Center
Curated by ChEMBL
Affinity DataIC50: 2.06E+3nMAssay Description:Inhibition of human TRPC4 channel expressed in HEK293 cells assessed as inhibition of EA-evoked Calcium influx by measuring reduction in intracellula...More data for this Ligand-Target Pair
TargetShort transient receptor potential channel 4(Mouse)
Johns Hopkins Ion Channel Center
Curated by PubChem BioAssay
Johns Hopkins Ion Channel Center
Curated by PubChem BioAssay
Affinity DataIC50: 2.38E+3nMAssay Description:Data Source: Johns Hopkins Ion Channel Center BioAssay Type: Confirmatory, Concentration-Response Relationship Observed Source (MLPCN Center Name): ...More data for this Ligand-Target Pair
TargetShort transient receptor potential channel 4(Mouse)
Johns Hopkins Ion Channel Center
Curated by PubChem BioAssay
Johns Hopkins Ion Channel Center
Curated by PubChem BioAssay
Affinity DataIC50: 2.60E+3nMAssay Description:Inhibition of mouse TRPC4 beta expressed in HEK293 cells co-expressing mu-opioid receptor assessed as reduction in DAMGO-induced current by QPatch cl...More data for this Ligand-Target Pair
TargetShort transient receptor potential channel 4(Mouse)
Johns Hopkins Ion Channel Center
Curated by PubChem BioAssay
Johns Hopkins Ion Channel Center
Curated by PubChem BioAssay
Affinity DataIC50: 2.63E+3nMAssay Description:Data Source: Johns Hopkins Ion Channel Center BioAssay Type: Confirmatory, Concentration-Response Relationship Observed Source (MLPCN Center Name): ...More data for this Ligand-Target Pair
TargetShort transient receptor potential channel 4(Mouse)
Johns Hopkins Ion Channel Center
Curated by PubChem BioAssay
Johns Hopkins Ion Channel Center
Curated by PubChem BioAssay
Affinity DataIC50: 3.14E+3nMAssay Description:Data Source: Johns Hopkins Ion Channel Center BioAssay Type: Confirmatory, Concentration-Response Relationship Observed Source (MLPCN Center Name): ...More data for this Ligand-Target Pair
TargetShort transient receptor potential channel 4(Mouse)
Johns Hopkins Ion Channel Center
Curated by PubChem BioAssay
Johns Hopkins Ion Channel Center
Curated by PubChem BioAssay
Affinity DataIC50: 3.30E+3nMAssay Description:The inhibitory effects of test compounds on TRPC4 channels were evaluated in electrophysiological assays using a QPatch16 automated electrophysiology...More data for this Ligand-Target Pair
TargetShort transient receptor potential channel 4(Mouse)
Johns Hopkins Ion Channel Center
Curated by PubChem BioAssay
Johns Hopkins Ion Channel Center
Curated by PubChem BioAssay
Affinity DataIC50: 3.59E+3nMAssay Description:Data Source: Johns Hopkins Ion Channel Center BioAssay Type: Confirmatory, Concentration-Response Relationship Observed Source (MLPCN Center Name): ...More data for this Ligand-Target Pair
TargetShort transient receptor potential channel 4(Mouse)
Johns Hopkins Ion Channel Center
Curated by PubChem BioAssay
Johns Hopkins Ion Channel Center
Curated by PubChem BioAssay
Affinity DataIC50: 3.70E+3nMAssay Description:Inhibition of mouse TRPC4 beta expressed in HEK293 cells co-expressing mu-opioid receptor assessed as reduction in DAMGO-induced intracellular calciu...More data for this Ligand-Target Pair
TargetShort transient receptor potential channel 4(Mouse)
Johns Hopkins Ion Channel Center
Curated by PubChem BioAssay
Johns Hopkins Ion Channel Center
Curated by PubChem BioAssay
Affinity DataIC50: 3.71E+3nMAssay Description:Data Source: Johns Hopkins Ion Channel Center BioAssay Type: Confirmatory, Concentration-Response Relationship Observed Source (MLPCN Center Name): ...More data for this Ligand-Target Pair
TargetShort transient receptor potential channel 4(Mouse)
Johns Hopkins Ion Channel Center
Curated by PubChem BioAssay
Johns Hopkins Ion Channel Center
Curated by PubChem BioAssay
Affinity DataIC50: 3.73E+3nMAssay Description:The inhibitory effects of test compounds on TRPC4 channels were evaluated in electrophysiological assays using a QPatch16 automated electrophysiology...More data for this Ligand-Target Pair
TargetShort transient receptor potential channel 4(Mouse)
Johns Hopkins Ion Channel Center
Curated by PubChem BioAssay
Johns Hopkins Ion Channel Center
Curated by PubChem BioAssay
Affinity DataIC50: 3.94E+3nMAssay Description:The inhibitory effects of test compounds on TRPC4 channels were evaluated in electrophysiological assays using a QPatch16 automated electrophysiology...More data for this Ligand-Target Pair
TargetShort transient receptor potential channel 4(Mouse)
Johns Hopkins Ion Channel Center
Curated by PubChem BioAssay
Johns Hopkins Ion Channel Center
Curated by PubChem BioAssay
Affinity DataIC50: 4.10E+3nMAssay Description:Inhibition of mouse TRPC4 beta expressed in HEK293 cells co-expressing mu-opioid receptor assessed as reduction in DAMGO-induced membrane potential b...More data for this Ligand-Target Pair
TargetShort transient receptor potential channel 4(Mouse)
Johns Hopkins Ion Channel Center
Curated by PubChem BioAssay
Johns Hopkins Ion Channel Center
Curated by PubChem BioAssay
Affinity DataIC50: 4.26E+3nMAssay Description:Data Source: Johns Hopkins Ion Channel Center BioAssay Type: Confirmatory, Concentration-Response Relationship Observed Source (MLPCN Center Name): ...More data for this Ligand-Target Pair
TargetShort transient receptor potential channel 4(Mouse)
Johns Hopkins Ion Channel Center
Curated by PubChem BioAssay
Johns Hopkins Ion Channel Center
Curated by PubChem BioAssay
Affinity DataIC50: 4.28E+3nMAssay Description:Data Source: Johns Hopkins Ion Channel Center BioAssay Type: Confirmatory, Concentration-Response Relationship Observed Source (MLPCN Center Name): ...More data for this Ligand-Target Pair
TargetShort transient receptor potential channel 4(Mouse)
Johns Hopkins Ion Channel Center
Curated by PubChem BioAssay
Johns Hopkins Ion Channel Center
Curated by PubChem BioAssay
Affinity DataIC50: 4.30E+3nMAssay Description:Inhibition of mouse TRPC4 beta expressed in HEK293 cells co-expressing mu-opioid receptor assessed as reduction in DAMGO-induced membrane potential b...More data for this Ligand-Target Pair
TargetShort transient receptor potential channel 4(Mouse)
Johns Hopkins Ion Channel Center
Curated by PubChem BioAssay
Johns Hopkins Ion Channel Center
Curated by PubChem BioAssay
Affinity DataIC50: 4.56E+3nMAssay Description:Data Source: Johns Hopkins Ion Channel Center BioAssay Type: Confirmatory, Concentration-Response Relationship Observed Source (MLPCN Center Name): ...More data for this Ligand-Target Pair
TargetShort transient receptor potential channel 4(Mouse)
Johns Hopkins Ion Channel Center
Curated by PubChem BioAssay
Johns Hopkins Ion Channel Center
Curated by PubChem BioAssay
Affinity DataIC50: 5.20E+3nMAssay Description:Inhibition of mouse TRPC4 beta expressed in HEK293 cells co-expressing mu-opioid receptor assessed as reduction in DAMGO-induced membrane potential b...More data for this Ligand-Target Pair
TargetShort transient receptor potential channel 4(Mouse)
Johns Hopkins Ion Channel Center
Curated by PubChem BioAssay
Johns Hopkins Ion Channel Center
Curated by PubChem BioAssay
Affinity DataIC50: 5.49E+3nMAssay Description:Data Source: Johns Hopkins Ion Channel Center BioAssay Type: Confirmatory, Concentration-Response Relationship Observed Source (MLPCN Center Name): ...More data for this Ligand-Target Pair
TargetShort transient receptor potential channel 4(Mouse)
Johns Hopkins Ion Channel Center
Curated by PubChem BioAssay
Johns Hopkins Ion Channel Center
Curated by PubChem BioAssay
Affinity DataIC50: 5.50E+3nMAssay Description:Inhibition of mouse TRPC4 beta expressed in HEK293 cells co-expressing mu-opioid receptor assessed as reduction in DAMGO-induced membrane potential b...More data for this Ligand-Target Pair
TargetShort transient receptor potential channel 4(Mouse)
Johns Hopkins Ion Channel Center
Curated by PubChem BioAssay
Johns Hopkins Ion Channel Center
Curated by PubChem BioAssay
Affinity DataIC50: 6.18E+3nMAssay Description:Data Source: Johns Hopkins Ion Channel Center BioAssay Type: Confirmatory, Concentration-Response Relationship Observed Source (MLPCN Center Name): ...More data for this Ligand-Target Pair
TargetShort transient receptor potential channel 4(Mouse)
Johns Hopkins Ion Channel Center
Curated by PubChem BioAssay
Johns Hopkins Ion Channel Center
Curated by PubChem BioAssay
Affinity DataIC50: 6.40E+3nMAssay Description:Inhibition of YFP-tagged mouse TRPC4 beta expressed in thapsigargin treated HEK293 cells co-expressing M3 receptor assessed as reduction in carbachol...More data for this Ligand-Target Pair
TargetShort transient receptor potential channel 4(Mouse)
Johns Hopkins Ion Channel Center
Curated by PubChem BioAssay
Johns Hopkins Ion Channel Center
Curated by PubChem BioAssay
Affinity DataIC50: 7.54E+3nMAssay Description:The inhibitory effects of test compounds on TRPC4 channels were evaluated in electrophysiological assays using a QPatch16 automated electrophysiology...More data for this Ligand-Target Pair
TargetShort transient receptor potential channel 4(Mouse)
Johns Hopkins Ion Channel Center
Curated by PubChem BioAssay
Johns Hopkins Ion Channel Center
Curated by PubChem BioAssay
Affinity DataIC50: 8.18E+3nMAssay Description:Data Source: Johns Hopkins Ion Channel Center BioAssay Type: Confirmatory, Concentration-Response Relationship Observed Source (MLPCN Center Name): ...More data for this Ligand-Target Pair
TargetShort transient receptor potential channel 4(Mouse)
Johns Hopkins Ion Channel Center
Curated by PubChem BioAssay
Johns Hopkins Ion Channel Center
Curated by PubChem BioAssay
Affinity DataIC50: 8.40E+3nMAssay Description:Inhibition of mouse TRPC4 expressed in HEK293 cells coexpressing M5 receptor assessed as reduction in TRPC4-mediated calcium influx by fluorescence m...More data for this Ligand-Target Pair
TargetShort transient receptor potential channel 4(Mouse)
Johns Hopkins Ion Channel Center
Curated by PubChem BioAssay
Johns Hopkins Ion Channel Center
Curated by PubChem BioAssay
Affinity DataIC50: 8.90E+3nMAssay Description:The inhibitory effects of test compounds on TRPC4 channels were evaluated in electrophysiological assays using a QPatch16 automated electrophysiology...More data for this Ligand-Target Pair
TargetShort transient receptor potential channel 4(Mouse)
Johns Hopkins Ion Channel Center
Curated by PubChem BioAssay
Johns Hopkins Ion Channel Center
Curated by PubChem BioAssay
Affinity DataIC50: 9.40E+3nMAssay Description:The inhibitory effects of test compounds on TRPC4 channels were evaluated in electrophysiological assays using a QPatch16 automated electrophysiology...More data for this Ligand-Target Pair
TargetShort transient receptor potential channel 4(Mouse)
Johns Hopkins Ion Channel Center
Curated by PubChem BioAssay
Johns Hopkins Ion Channel Center
Curated by PubChem BioAssay
Affinity DataIC50: 9.89E+3nMAssay Description:The inhibitory effects of test compounds on TRPC4 channels were evaluated in electrophysiological assays using a QPatch16 automated electrophysiology...More data for this Ligand-Target Pair
TargetShort transient receptor potential channel 4(Mouse)
Johns Hopkins Ion Channel Center
Curated by PubChem BioAssay
Johns Hopkins Ion Channel Center
Curated by PubChem BioAssay
Affinity DataIC50: 9.96E+3nMAssay Description:The inhibitory effects of test compounds on TRPC4 channels were evaluated in electrophysiological assays using a QPatch16 automated electrophysiology...More data for this Ligand-Target Pair
TargetShort transient receptor potential channel 4(Mouse)
Johns Hopkins Ion Channel Center
Curated by PubChem BioAssay
Johns Hopkins Ion Channel Center
Curated by PubChem BioAssay
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of mouse TRPC4 by FLIPR assayMore data for this Ligand-Target Pair
TargetShort transient receptor potential channel 4(Human)
University of Nebraska Medical Center
Curated by ChEMBL
University of Nebraska Medical Center
Curated by ChEMBL
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of TRPC4 (unknown origin)More data for this Ligand-Target Pair
TargetShort transient receptor potential channel 4(Mouse)
Johns Hopkins Ion Channel Center
Curated by PubChem BioAssay
Johns Hopkins Ion Channel Center
Curated by PubChem BioAssay
Affinity DataIC50: 1.00E+4nMAssay Description:Antagonist activity at mouse TRPC4beta expressed in HEK293 cells co-expressing MOR decrease in DAMGO-evoked intracellular calcium level by Fluo-8-AM ...More data for this Ligand-Target Pair
TargetShort transient receptor potential channel 4(Mouse)
Johns Hopkins Ion Channel Center
Curated by PubChem BioAssay
Johns Hopkins Ion Channel Center
Curated by PubChem BioAssay
Affinity DataIC50: 1.02E+4nMAssay Description:Inhibition of mouse TRPC4 beta expressed in HEK293 cells co-expressing mu-opioid receptor assessed as reduction in DAMGO-induced membrane potential b...More data for this Ligand-Target Pair
TargetShort transient receptor potential channel 4(Mouse)
Johns Hopkins Ion Channel Center
Curated by PubChem BioAssay
Johns Hopkins Ion Channel Center
Curated by PubChem BioAssay
Affinity DataIC50: 1.03E+4nMAssay Description:Inhibition of mouse TRPC4 beta expressed in HEK293 cells co-expressing mu-opioid receptor assessed as reduction in DAMGO-induced membrane potential b...More data for this Ligand-Target Pair
TargetShort transient receptor potential channel 4(Mouse)
Johns Hopkins Ion Channel Center
Curated by PubChem BioAssay
Johns Hopkins Ion Channel Center
Curated by PubChem BioAssay
Affinity DataIC50: 1.10E+4nMAssay Description:Inhibition of mouse TRPC4 beta expressed in HEK293 cells co-expressing mu-opioid receptor assessed as reduction in DAMGO-induced membrane potential b...More data for this Ligand-Target Pair
TargetShort transient receptor potential channel 4(Mouse)
Johns Hopkins Ion Channel Center
Curated by PubChem BioAssay
Johns Hopkins Ion Channel Center
Curated by PubChem BioAssay
Affinity DataIC50: 1.19E+4nMAssay Description:The inhibitory effects of test compounds on TRPC4 channels were evaluated in electrophysiological assays using a QPatch16 automated electrophysiology...More data for this Ligand-Target Pair
TargetShort transient receptor potential channel 4(Mouse)
Johns Hopkins Ion Channel Center
Curated by PubChem BioAssay
Johns Hopkins Ion Channel Center
Curated by PubChem BioAssay
Affinity DataIC50: 2.45E+4nMAssay Description:The inhibitory effects of test compounds on TRPC4 channels were evaluated in electrophysiological assays using a QPatch16 automated electrophysiology...More data for this Ligand-Target Pair
TargetShort transient receptor potential channel 4(Mouse)
Johns Hopkins Ion Channel Center
Curated by PubChem BioAssay
Johns Hopkins Ion Channel Center
Curated by PubChem BioAssay
Affinity DataIC50: 3.50E+4nMAssay Description:Antagonist activity at mouse TRPC4beta expressed in HEK293 cells co-expressing MOR decrease in DAMGO-evoked intracellular calcium level by Fluo-8-AM ...More data for this Ligand-Target Pair
TargetShort transient receptor potential channel 4(Mouse)
Johns Hopkins Ion Channel Center
Curated by PubChem BioAssay
Johns Hopkins Ion Channel Center
Curated by PubChem BioAssay
Affinity DataIC50: 3.87E+4nMAssay Description:Data Source: Johns Hopkins Ion Channel Center BioAssay Type: Confirmatory, Concentration-Response Relationship Observed Source (MLPCN Center Name): ...More data for this Ligand-Target Pair
