Compile Data Set for Download or QSAR
Report error Found 63 of ic50 data for polymerid = 2445,50000355,50002089
TargetCytosol aminopeptidase(Bovine)
Enscmu

LigandPNGBDBM23971(CHEMBL29292 | (2S)-2-[(2S,3R)-3-amino-2-hydroxy-4-...)
Affinity DataIC50: 0.5nMpH: 8.0 T: 2°CAssay Description:Spectrophotometric assays were performed by monitoring hydrolysis of chromogenic substrate. The release of para-nitroaniline at 405 nm was measured t...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCytosol aminopeptidase(Bovine)
Enscmu

LigandPNGBDBM23971(CHEMBL29292 | (2S)-2-[(2S,3R)-3-amino-2-hydroxy-4-...)
Affinity DataIC50: 0.5nMAssay Description:Inhibition of bovine lens cytosolic leucine aminopeptidase by Dixon plot analysisMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCytosol aminopeptidase(Human)
Pharmacia and Upjohn

Curated by ChEMBL
LigandPNGBDBM50078391((S)-1-[(R)-3-((2S,3R)-3-Amino-2-hydroxy-4-phenyl-b...)
Affinity DataIC50: 180nMAssay Description:Inhibition against Leucyl aminopeptidase from pig kidney.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCytosol aminopeptidase(Human)
Pharmacia and Upjohn

Curated by ChEMBL
LigandPNGBDBM50078393((S)-1-[(S)-1-((2S,3R)-3-Amino-2-hydroxy-4-phenyl-b...)
Affinity DataIC50: 290nMAssay Description:Inhibition against Leucyl aminopeptidase from pig kidney.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCytosol aminopeptidase(Human)
Pharmacia and Upjohn

Curated by ChEMBL
LigandPNGBDBM50078401((S)-1-[(S)-1-((2S,3R)-3-Amino-2-hydroxy-4-phenyl-b...)
Affinity DataIC50: 300nMAssay Description:Inhibition against Leucyl aminopeptidase from pig kidney.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCytosol aminopeptidase(Human)
Pharmacia and Upjohn

Curated by ChEMBL
LigandPNGBDBM50078400(1-[1-(3-Amino-2-hydroxy-4-phenyl-butyryl)-4-hydrox...)
Affinity DataIC50: 1.60E+3nMAssay Description:Inhibition against Leucyl aminopeptidase from pig kidney.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCytosol aminopeptidase(Human)
Pharmacia and Upjohn

Curated by ChEMBL
LigandPNGBDBM50078394((S)-1-[(S)-1-((2S,3R)-3-Amino-2-hydroxy-4-phenyl-b...)
Affinity DataIC50: 2.50E+3nMAssay Description:Inhibition against Leucyl aminopeptidase from pig kidney.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCytosol aminopeptidase(Pig)
National Institute of Public Health-National Institute of Hygiene

Curated by ChEMBL
LigandPNGBDBM23971(CHEMBL29292 | (2S)-2-[(2S,3R)-3-amino-2-hydroxy-4-...)
Affinity DataIC50: 5.20E+3nMAssay Description:Inhibition of porcine kidney microsomal LAP using l-leucine-7-amido-4-methylcoumarin as substrate incubated for 60 mins measured every 3 mins by fluo...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCytosol aminopeptidase(Human)
Pharmacia and Upjohn

Curated by ChEMBL
LigandPNGBDBM50078402((S)-1-((R)-3-Amino-2-hydroxy-5-methyl-hexanoyl)-py...)
Affinity DataIC50: 7.80E+3nMAssay Description:Inhibition against Leucyl aminopeptidase from pig kidney.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCytosol aminopeptidase(Pig)
National Institute of Public Health-National Institute of Hygiene

Curated by ChEMBL
LigandPNGBDBM23971(CHEMBL29292 | (2S)-2-[(2S,3R)-3-amino-2-hydroxy-4-...)
Affinity DataIC50: 1.12E+4nMAssay Description:Inhibition of porcine kidney microsomal LAP using l-leucine-7-amido-4-methylcoumarin as substrate incubated for 10 hrs measured every 6 mins by fluor...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCytosol aminopeptidase(Human)
Pharmacia and Upjohn

Curated by ChEMBL
LigandPNGBDBM23971(CHEMBL29292 | (2S)-2-[(2S,3R)-3-amino-2-hydroxy-4-...)
Affinity DataIC50: 1.12E+4nMAssay Description:Inhibitory concentration against adipocyte-derived leucine aminopeptidaseMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCytosol aminopeptidase(Human)
Pharmacia and Upjohn

Curated by ChEMBL
LigandPNGBDBM50078397(1-(3-Amino-2-hydroxy-5-methyl-hexanoyl)-pyrrolidin...)
Affinity DataIC50: 1.20E+4nMAssay Description:Inhibition against Leucyl aminopeptidase from pig kidney.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCytosol aminopeptidase(Pig)
National Institute of Public Health-National Institute of Hygiene

Curated by ChEMBL
LigandPNGBDBM50534075(CHEMBL4483393)
Affinity DataIC50: 1.65E+4nMAssay Description:Inhibition of porcine kidney microsomal LAP using l-leucine-7-amido-4-methylcoumarin as substrate incubated for 60 mins measured every 3 mins by fluo...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetCytosol aminopeptidase(Pig)
National Institute of Public Health-National Institute of Hygiene

Curated by ChEMBL
LigandPNGBDBM50534075(CHEMBL4483393)
Affinity DataIC50: 3.36E+4nMAssay Description:Inhibition of porcine kidney microsomal LAP using l-leucine-7-amido-4-methylcoumarin as substrate incubated for 10 hrs measured every 6 mins by fluor...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetCytosol aminopeptidase(Human)
Pharmacia and Upjohn

Curated by ChEMBL
LigandPNGBDBM50046316(2-Amino-3-(4-benzyloxy-phenyl)-propane-1-thiol | C...)
Affinity DataIC50: 5.00E+4nMAssay Description:Inhibitory concentration against cytosolic leucine aminopeptidaseMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCytosol aminopeptidase(Human)
Pharmacia and Upjohn

Curated by ChEMBL
LigandPNGBDBM50046329(3-Amino-4-(4-benzyloxy-phenyl)-2-oxo-butyric acid ...)
Affinity DataIC50: 5.00E+4nMAssay Description:Inhibitory concentration against cytosolic leucine aminopeptidaseMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCytosol aminopeptidase(Pig)
National Institute of Public Health-National Institute of Hygiene

Curated by ChEMBL
LigandPNGBDBM50534077(CHEMBL4464704)
Affinity DataIC50: 6.36E+4nMAssay Description:Inhibition of porcine kidney microsomal LAP using l-leucine-7-amido-4-methylcoumarin as substrate incubated for 60 mins measured every 3 mins by fluo...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetCytosol aminopeptidase(Pig)
National Institute of Public Health-National Institute of Hygiene

Curated by ChEMBL
LigandPNGBDBM50534070(CHEMBL4454667)
Affinity DataIC50: 6.83E+4nMAssay Description:Inhibition of porcine kidney microsomal LAP using l-leucine-7-amido-4-methylcoumarin as substrate incubated for 60 mins measured every 3 mins by fluo...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetCytosol aminopeptidase(Pig)
National Institute of Public Health-National Institute of Hygiene

Curated by ChEMBL
LigandPNGBDBM50534074(CHEMBL4468968)
Affinity DataIC50: 6.93E+4nMAssay Description:Inhibition of porcine kidney microsomal LAP using l-leucine-7-amido-4-methylcoumarin as substrate incubated for 60 mins measured every 3 mins by fluo...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetCytosol aminopeptidase(Pig)
National Institute of Public Health-National Institute of Hygiene

Curated by ChEMBL
LigandPNGBDBM50534069(CHEMBL4473220)
Affinity DataIC50: 7.68E+4nMAssay Description:Inhibition of porcine kidney microsomal LAP using l-leucine-7-amido-4-methylcoumarin as substrate incubated for 60 mins measured every 3 mins by fluo...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetCytosol aminopeptidase(Human)
Pharmacia and Upjohn

Curated by ChEMBL
LigandPNGBDBM50046321(3-Amino-4-(4-benzyloxy-phenyl)-2-hydroxy-butyric a...)
Affinity DataIC50: 8.00E+4nMAssay Description:Inhibitory concentration against cytosolic leucine aminopeptidaseMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCytosol aminopeptidase(Human)
Pharmacia and Upjohn

Curated by ChEMBL
LigandPNGBDBM50051495((S)-2-[(S)-2-(2-Hydroxy-acetyl)-pyrrolidine-1-carb...)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of proline iminopeptidase)More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCytosol aminopeptidase(Bovine)
Enscmu

LigandPNGBDBM50336496(2-aminocycloheptanone hydrochloride | CHEMBL166862...)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of bovine lens cytosolic leucine aminopeptidase by Dixon plot analysisMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCytosol aminopeptidase(Bovine)
Enscmu

LigandPNGBDBM23977((3Z)-3-[(2-phenylethoxy)imino]-1,2,3,4-tetrahydron...)
Affinity DataIC50: 1.00E+5nMpH: 8.0 T: 2°CAssay Description:Spectrophotometric assays were performed by monitoring hydrolysis of chromogenic substrate. The release of para-nitroaniline at 405 nm was measured t...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetCytosol aminopeptidase(Human)
Pharmacia and Upjohn

Curated by ChEMBL
LigandPNGBDBM50046314(3-Amino-4-(4-benzyloxy-phenyl)-2-oxo-butyric acid ...)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibitory concentration against cytosolic leucine aminopeptidaseMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCytosol aminopeptidase(Bovine)
Enscmu

LigandPNGBDBM23980((3Z)-3-{[(5-phenylpentyl)oxy]imino}-1,2,3,4-tetrah...)
Affinity DataIC50: 1.00E+5nMpH: 8.0 T: 2°CAssay Description:Spectrophotometric assays were performed by monitoring hydrolysis of chromogenic substrate. The release of para-nitroaniline at 405 nm was measured t...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetCytosol aminopeptidase(Bovine)
Enscmu

LigandPNGBDBM23979((3Z)-3-[(4-phenylbutoxy)imino]-1,2,3,4-tetrahydron...)
Affinity DataIC50: 1.00E+5nMpH: 8.0 T: 2°CAssay Description:Spectrophotometric assays were performed by monitoring hydrolysis of chromogenic substrate. The release of para-nitroaniline at 405 nm was measured t...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetCytosol aminopeptidase(Pig)
National Institute of Public Health-National Institute of Hygiene

Curated by ChEMBL
LigandPNGBDBM50534072(CHEMBL4455383)
Affinity DataIC50: 1.11E+5nMAssay Description:Inhibition of porcine kidney microsomal LAP using l-leucine-7-amido-4-methylcoumarin as substrate incubated for 60 mins measured every 3 mins by fluo...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetCytosol aminopeptidase(Bovine)
Enscmu

LigandPNGBDBM23973(3-amino-1,2,3,4-tetrahydronaphthalen-2-one hydroch...)
Affinity DataIC50: 1.20E+5nMpH: 8.0 T: 2°CAssay Description:Spectrophotometric assays were performed by monitoring hydrolysis of chromogenic substrate. The release of para-nitroaniline at 405 nm was measured t...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetCytosol aminopeptidase(Bovine)
Enscmu

LigandPNGBDBM23973(3-amino-1,2,3,4-tetrahydronaphthalen-2-one hydroch...)
Affinity DataIC50: 1.20E+5nMAssay Description:Inhibition of bovine lens cytosolic leucine aminopeptidase by Dixon plot analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetCytosol aminopeptidase(Pig)
National Institute of Public Health-National Institute of Hygiene

Curated by ChEMBL
LigandPNGBDBM50534078(CHEMBL4557950)
Affinity DataIC50: 1.38E+5nMAssay Description:Inhibition of porcine kidney microsomal LAP using l-leucine-7-amido-4-methylcoumarin as substrate incubated for 60 mins measured every 3 mins by fluo...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetCytosol aminopeptidase(Pig)
National Institute of Public Health-National Institute of Hygiene

Curated by ChEMBL
LigandPNGBDBM50534081(CHEMBL4460083)
Affinity DataIC50: 1.63E+5nMAssay Description:Inhibition of porcine kidney microsomal LAP using l-leucine-7-amido-4-methylcoumarin as substrate incubated for 60 mins measured every 3 mins by fluo...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetCytosol aminopeptidase(Human)
Pharmacia and Upjohn

Curated by ChEMBL
LigandPNGBDBM50078395((S)-1-(2-Hydroxycarbamoyl-cyclohexanecarbonyl)-pyr...)
Affinity DataIC50: 2.20E+5nMAssay Description:Inhibition against Leucyl aminopeptidase from pig kidney.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCytosol aminopeptidase(Human)
Pharmacia and Upjohn

Curated by ChEMBL
LigandPNGBDBM50078395((S)-1-(2-Hydroxycarbamoyl-cyclohexanecarbonyl)-pyr...)
Affinity DataIC50: 2.20E+5nMAssay Description:Inhibition against Leucyl aminopeptidase from pig kidney.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCytosol aminopeptidase(Pig)
National Institute of Public Health-National Institute of Hygiene

Curated by ChEMBL
LigandPNGBDBM50534071(CHEMBL4563759)
Affinity DataIC50: 3.79E+5nMAssay Description:Inhibition of porcine kidney microsomal LAP using l-leucine-7-amido-4-methylcoumarin as substrate incubated for 60 mins measured every 3 mins by fluo...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetCytosol aminopeptidase(Pig)
National Institute of Public Health-National Institute of Hygiene

Curated by ChEMBL
LigandPNGBDBM50534080(CHEMBL4576374)
Affinity DataIC50: 4.09E+5nMAssay Description:Inhibition of porcine kidney microsomal LAP using l-leucine-7-amido-4-methylcoumarin as substrate incubated for 60 mins measured every 3 mins by fluo...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetCytosol aminopeptidase(Human)
Pharmacia and Upjohn

Curated by ChEMBL
LigandPNGBDBM50078390((S)-1-((2S,3S)-3-Amino-2-hydroxy-5-methyl-hexanoyl...)
Affinity DataIC50: 4.50E+5nMAssay Description:Inhibition against Leucyl aminopeptidase from pig kidney.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCytosol aminopeptidase(Pig)
National Institute of Public Health-National Institute of Hygiene

Curated by ChEMBL
LigandPNGBDBM50534073(CHEMBL4537106)
Affinity DataIC50: 7.81E+5nMAssay Description:Inhibition of porcine kidney microsomal LAP using l-leucine-7-amido-4-methylcoumarin as substrate incubated for 60 mins measured every 3 mins by fluo...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetCytosol aminopeptidase(Human)
Pharmacia and Upjohn

Curated by ChEMBL
LigandPNGBDBM50078399((S)-1-((3R,4S)-4-Amino-3-hydroxy-6-methyl-heptanoy...)
Affinity DataIC50: 8.00E+5nMAssay Description:Inhibition against Leucyl aminopeptidase from pig kidney.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCytosol aminopeptidase(Bovine)
Enscmu

LigandPNGBDBM23984(3-amino-1,2,3,4-tetrahydronaphthalene-2-phosphonic...)
Affinity DataIC50: 1.00E+6nMpH: 8.0 T: 2°CAssay Description:Spectrophotometric assays were performed by monitoring hydrolysis of chromogenic substrate. The release of para-nitroaniline at 405 nm was measured t...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetCytosol aminopeptidase(Bovine)
Enscmu

LigandPNGBDBM23987(2-hydroxy-1,2,3,4-tetrahydroisoquinolin-3-one | CH...)
Affinity DataIC50: 1.00E+6nMpH: 8.0 T: 2°CAssay Description:Spectrophotometric assays were performed by monitoring hydrolysis of chromogenic substrate. The release of para-nitroaniline at 405 nm was measured t...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCytosol aminopeptidase(Bovine)
Enscmu

LigandPNGBDBM23982(1-(3-amino-1,2,3,4-tetrahydronaphthalen-2-yl)ethan...)
Affinity DataIC50: 1.00E+6nMpH: 8.0 T: 2°CAssay Description:Spectrophotometric assays were performed by monitoring hydrolysis of chromogenic substrate. The release of para-nitroaniline at 405 nm was measured t...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetCytosol aminopeptidase(Bovine)
Enscmu

LigandPNGBDBM23981((2S)-1,2,3,4-Tetrahydro-naphthalen-2-ylamine | 1,2...)
Affinity DataIC50: 1.00E+6nMpH: 8.0 T: 2°CAssay Description:Spectrophotometric assays were performed by monitoring hydrolysis of chromogenic substrate. The release of para-nitroaniline at 405 nm was measured t...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCytosol aminopeptidase(Bovine)
Enscmu

LigandPNGBDBM23978((3Z)-3-[(3-phenylpropoxy)imino]-1,2,3,4-tetrahydro...)
Affinity DataIC50: 1.00E+6nMpH: 8.0 T: 2°CAssay Description:Spectrophotometric assays were performed by monitoring hydrolysis of chromogenic substrate. The release of para-nitroaniline at 405 nm was measured t...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetCytosol aminopeptidase(Bovine)
Enscmu

LigandPNGBDBM23976((3Z)-3-[(benzyloxy)imino]-1,2,3,4-tetrahydronaphth...)
Affinity DataIC50: 1.00E+6nMpH: 8.0 T: 2°CAssay Description:Spectrophotometric assays were performed by monitoring hydrolysis of chromogenic substrate. The release of para-nitroaniline at 405 nm was measured t...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetCytosol aminopeptidase(Pig)
National Institute of Public Health-National Institute of Hygiene

Curated by ChEMBL
LigandPNGBDBM50534076(CHEMBL4435767)
Affinity DataIC50: 1.05E+6nMAssay Description:Inhibition of porcine kidney microsomal LAP using l-leucine-7-amido-4-methylcoumarin as substrate incubated for 60 mins measured every 3 mins by fluo...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetCytosol aminopeptidase(Bovine)
Enscmu

LigandPNGBDBM23975((3Z)-3-(methoxyimino)-1,2,3,4-tetrahydronaphthalen...)
Affinity DataIC50: 1.00E+6nMpH: 8.0 T: 2°CAssay Description:Spectrophotometric assays were performed by monitoring hydrolysis of chromogenic substrate. The release of para-nitroaniline at 405 nm was measured t...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetCytosol aminopeptidase(Bovine)
Enscmu

LigandPNGBDBM23974((3Z)-3-(hydroxyimino)-1,2,3,4-tetrahydronaphthalen...)
Affinity DataIC50: 1.00E+6nMpH: 8.0 T: 2°CAssay Description:Spectrophotometric assays were performed by monitoring hydrolysis of chromogenic substrate. The release of para-nitroaniline at 405 nm was measured t...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetCytosol aminopeptidase(Pig)
National Institute of Public Health-National Institute of Hygiene

Curated by ChEMBL
LigandPNGBDBM50534079(CHEMBL4456116)
Affinity DataIC50: 1.11E+6nMAssay Description:Inhibition of porcine kidney microsomal LAP using l-leucine-7-amido-4-methylcoumarin as substrate incubated for 60 mins measured every 3 mins by fluo...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetCytosol aminopeptidase(Bovine)
Enscmu

LigandPNGBDBM23985(3,4-dihydro-1H-2-benzopyran-3-one | isochromanone,...)
Affinity DataIC50: 1.00E+6nMpH: 8.0 T: 2°CAssay Description:Spectrophotometric assays were performed by monitoring hydrolysis of chromogenic substrate. The release of para-nitroaniline at 405 nm was measured t...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
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