Report error Found 416 of ic50 data for polymerid = 10032
TargetNAD-dependent protein deacetylase sirtuin-3, mitochondrial(Human)
Sirtris A Gsk
Curated by ChEMBL
Sirtris A Gsk
Curated by ChEMBL
Affinity DataIC50: 3.20nMAssay Description:Inhibition of human His-tagged SIRT3 (102 to 399) expressed in Escherichia coli BL21(DE3) assessed as inhibition of deacetylation of Ac-RHKKAcW-NH2 s...More data for this Ligand-Target Pair
TargetNAD-dependent protein deacetylase sirtuin-3, mitochondrial(Human)
Sirtris A Gsk
Curated by ChEMBL
Sirtris A Gsk
Curated by ChEMBL
Affinity DataIC50: 4nMAssay Description:Inhibition of human His-tagged SIRT3 (102 to 399) expressed in Escherichia coli BL21(DE3) assessed as inhibition of deacetylation of Ac-RHKKAcW-NH2 s...More data for this Ligand-Target Pair
TargetNAD-dependent protein deacetylase sirtuin-3, mitochondrial(Human)
Sirtris A Gsk
Curated by ChEMBL
Sirtris A Gsk
Curated by ChEMBL
Affinity DataIC50: 4.90nMAssay Description:Inhibition of human His-tagged SIRT3 (102 to 399) expressed in Escherichia coli BL21(DE3) assessed as inhibition of deacetylation of Ac-RHKKAcW-NH2 s...More data for this Ligand-Target Pair
TargetNAD-dependent protein deacetylase sirtuin-3, mitochondrial(Human)
Sirtris A Gsk
Curated by ChEMBL
Sirtris A Gsk
Curated by ChEMBL
Affinity DataIC50: 7.20nMAssay Description:Inhibition of human His-tagged SIRT3 (102 to 399) expressed in Escherichia coli BL21(DE3) assessed as inhibition of deacetylation of Ac-RHKKAcW-NH2 s...More data for this Ligand-Target Pair
TargetNAD-dependent protein deacetylase sirtuin-3, mitochondrial(Human)
Sirtris A Gsk
Curated by ChEMBL
Sirtris A Gsk
Curated by ChEMBL
Affinity DataIC50: 7.60nMAssay Description:Inhibition of human His-tagged SIRT3 (102 to 399) expressed in Escherichia coli BL21(DE3) assessed as inhibition of deacetylation of Ac-RHKKAcW-NH2 s...More data for this Ligand-Target Pair
TargetNAD-dependent protein deacetylase sirtuin-3, mitochondrial(Human)
Sirtris A Gsk
Curated by ChEMBL
Sirtris A Gsk
Curated by ChEMBL
Affinity DataIC50: 13nMAssay Description:Inhibition of human His-tagged SIRT3 (102 to 399) expressed in Escherichia coli BL21(DE3) assessed as inhibition of deacetylation of Ac-RHKKAcW-NH2 s...More data for this Ligand-Target Pair
TargetNAD-dependent protein deacetylase sirtuin-3, mitochondrial(Human)
Sirtris A Gsk
Curated by ChEMBL
Sirtris A Gsk
Curated by ChEMBL
Affinity DataIC50: 23nMAssay Description:Inhibition of human His-tagged SIRT3 (102 to 399) expressed in Escherichia coli BL21(DE3) assessed as inhibition of deacetylation of Ac-RHKKAcW-NH2 s...More data for this Ligand-Target Pair
TargetNAD-dependent protein deacetylase sirtuin-3, mitochondrial(Human)
Sirtris A Gsk
Curated by ChEMBL
Sirtris A Gsk
Curated by ChEMBL
Affinity DataIC50: 24nMAssay Description:Inhibition of human His-tagged SIRT3 (102 to 399) expressed in Escherichia coli BL21(DE3) assessed as inhibition of deacetylation of Ac-RHKKAcW-NH2 s...More data for this Ligand-Target Pair
TargetNAD-dependent protein deacetylase sirtuin-3, mitochondrial(Human)
Sirtris A Gsk
Curated by ChEMBL
Sirtris A Gsk
Curated by ChEMBL
Affinity DataIC50: 28nMAssay Description:Inhibition of human His-tagged SIRT3 (102 to 399) expressed in Escherichia coli BL21(DE3) assessed as inhibition of deacetylation of Ac-RHKKAcW-NH2 s...More data for this Ligand-Target Pair
TargetNAD-dependent protein deacetylase sirtuin-3, mitochondrial(Human)
Sirtris A Gsk
Curated by ChEMBL
Sirtris A Gsk
Curated by ChEMBL
Affinity DataIC50: 29nMAssay Description:Inhibition of human His-tagged SIRT3 (102 to 399) expressed in Escherichia coli BL21(DE3) assessed as inhibition of deacetylation of Ac-RHKKAcW-NH2 s...More data for this Ligand-Target Pair
TargetNAD-dependent protein deacetylase sirtuin-3, mitochondrial(Human)
Sirtris A Gsk
Curated by ChEMBL
Sirtris A Gsk
Curated by ChEMBL
Affinity DataIC50: 30nMAssay Description:Inhibition of human His-tagged SIRT3 (102 to 399) expressed in Escherichia coli BL21(DE3) assessed as inhibition of deacetylation of Ac-RHKKAcW-NH2 s...More data for this Ligand-Target Pair
TargetNAD-dependent protein deacetylase sirtuin-3, mitochondrial(Human)
Sirtris A Gsk
Curated by ChEMBL
Sirtris A Gsk
Curated by ChEMBL
Affinity DataIC50: 33nMAssay Description:Inhibition of human His-tagged SIRT3 (102 to 399) expressed in Escherichia coli BL21(DE3) assessed as inhibition of deacetylation of Ac-RHKKAcW-NH2 s...More data for this Ligand-Target Pair
TargetNAD-dependent protein deacetylase sirtuin-3, mitochondrial(Human)
Sirtris A Gsk
Curated by ChEMBL
Sirtris A Gsk
Curated by ChEMBL
Affinity DataIC50: 39nMAssay Description:Inhibition of human His-tagged SIRT3 (102 to 399) expressed in Escherichia coli BL21(DE3) assessed as inhibition of deacetylation of Ac-RHKKAcW-NH2 s...More data for this Ligand-Target Pair
TargetNAD-dependent protein deacetylase sirtuin-3, mitochondrial(Human)
Sirtris A Gsk
Curated by ChEMBL
Sirtris A Gsk
Curated by ChEMBL
Affinity DataIC50: 43nMAssay Description:Inhibition of recombinant His6 tagged human SIRT3 using 0.105 mM H2N-HK-[N(epsilon)-acetyl-lysine]-LM-COOH as substrate measured after 10 mins HPLC a...More data for this Ligand-Target Pair
TargetNAD-dependent protein deacetylase sirtuin-3, mitochondrial(Human)
Sirtris A Gsk
Curated by ChEMBL
Sirtris A Gsk
Curated by ChEMBL
Affinity DataIC50: 46nMAssay Description:Inhibition of recombinant human SIRT3 (118 to 399 residues) defatty-acylase activity expressed in Escherichia coli using SFP3 as substrate measured a...More data for this Ligand-Target Pair
TargetNAD-dependent protein deacetylase sirtuin-3, mitochondrial(Human)
Sirtris A Gsk
Curated by ChEMBL
Sirtris A Gsk
Curated by ChEMBL
Affinity DataIC50: 53nMAssay Description:Inhibition of recombinant His6 tagged human SIRT3 using 0.105 mM H2N-HK-[N(epsilon)-acetyl-lysine]-LM-COOH as substrate measured after 10 mins HPLC a...More data for this Ligand-Target Pair
TargetNAD-dependent protein deacetylase sirtuin-3, mitochondrial(Human)
Sirtris A Gsk
Curated by ChEMBL
Sirtris A Gsk
Curated by ChEMBL
Affinity DataIC50: 55nMAssay Description:Inhibition of recombinant human SIRT3 (118 to 399 residues) defatty-acylase activity expressed in Escherichia coli using SFP3 as substrate measured a...More data for this Ligand-Target Pair
TargetNAD-dependent protein deacetylase sirtuin-3, mitochondrial(Human)
Sirtris A Gsk
Curated by ChEMBL
Sirtris A Gsk
Curated by ChEMBL
Affinity DataIC50: 56nMAssay Description:Inhibition of human His-tagged SIRT3 (102 to 399) expressed in Escherichia coli BL21(DE3) assessed as inhibition of deacetylation of Ac-RHKKAcW-NH2 s...More data for this Ligand-Target Pair
TargetNAD-dependent protein deacetylase sirtuin-3, mitochondrial(Human)
Sirtris A Gsk
Curated by ChEMBL
Sirtris A Gsk
Curated by ChEMBL
Affinity DataIC50: 57nMAssay Description:Inhibition of recombinant His6 tagged human SIRT3 using 0.105 mM H2N-HK-[N(epsilon)-acetyl-lysine]-LM-COOH as substrate measured after 10 mins HPLC a...More data for this Ligand-Target Pair
TargetNAD-dependent protein deacetylase sirtuin-3, mitochondrial(Human)
Sirtris A Gsk
Curated by ChEMBL
Sirtris A Gsk
Curated by ChEMBL
Affinity DataIC50: 61nMAssay Description:Inhibition of human His-tagged SIRT3 (102 to 399) expressed in Escherichia coli BL21(DE3) assessed as inhibition of deacetylation of Ac-RHKKAcW-NH2 s...More data for this Ligand-Target Pair
TargetNAD-dependent protein deacetylase sirtuin-3, mitochondrial(Human)
Sirtris A Gsk
Curated by ChEMBL
Sirtris A Gsk
Curated by ChEMBL
Affinity DataIC50: 67nMAssay Description:Inhibition of human His-tagged SIRT3 (102 to 399) expressed in Escherichia coli BL21(DE3) assessed as inhibition of deacetylation of Ac-RHKKAcW-NH2 s...More data for this Ligand-Target Pair
TargetNAD-dependent protein deacetylase sirtuin-3, mitochondrial(Human)
Sirtris A Gsk
Curated by ChEMBL
Sirtris A Gsk
Curated by ChEMBL
Affinity DataIC50: 71nMAssay Description:Inhibition of recombinant His6 tagged human SIRT3 using 0.105 mM H2N-HK-[N(epsilon)-acetyl-lysine]-LM-COOH as substrate measured after 10 mins HPLC a...More data for this Ligand-Target Pair
TargetNAD-dependent protein deacetylase sirtuin-3, mitochondrial(Human)
Sirtris A Gsk
Curated by ChEMBL
Sirtris A Gsk
Curated by ChEMBL
Affinity DataIC50: 77nMAssay Description:Inhibition of recombinant human SIRT3 (118 to 399 residues) defatty-acylase activity expressed in Escherichia coli using SFP3 as substrate measured a...More data for this Ligand-Target Pair
TargetNAD-dependent protein deacetylase sirtuin-3, mitochondrial(Human)
Sirtris A Gsk
Curated by ChEMBL
Sirtris A Gsk
Curated by ChEMBL
Affinity DataIC50: 83nMAssay Description:Inhibition of recombinant His6 tagged human SIRT3 using 0.105 mM H2N-HK-[N(epsilon)-acetyl-lysine]-LM-COOH as substrate measured after 10 mins HPLC a...More data for this Ligand-Target Pair
TargetNAD-dependent protein deacetylase sirtuin-3, mitochondrial(Human)
Sirtris A Gsk
Curated by ChEMBL
Sirtris A Gsk
Curated by ChEMBL
Affinity DataIC50: 92nMAssay Description:Inhibition of human His-tagged SIRT3 (102 to 399) expressed in Escherichia coli BL21(DE3) assessed as inhibition of deacetylation of Ac-RHKKAcW-NH2 s...More data for this Ligand-Target Pair
TargetNAD-dependent protein deacetylase sirtuin-3, mitochondrial(Human)
Sirtris A Gsk
Curated by ChEMBL
Sirtris A Gsk
Curated by ChEMBL
Affinity DataIC50: 100nMAssay Description:Inhibition of human SIRT3 (118 to 399 aa) expressed in Escherichia coli BL21 cellsMore data for this Ligand-Target Pair
TargetNAD-dependent protein deacetylase sirtuin-3, mitochondrial(Human)
Sirtris A Gsk
Curated by ChEMBL
Sirtris A Gsk
Curated by ChEMBL
Affinity DataIC50: 103nMAssay Description:Inhibition of recombinant His6 tagged human SIRT3 using 0.105 mM H2N-HK-[N(epsilon)-acetyl-lysine]-LM-COOH as substrate measured after 10 mins HPLC a...More data for this Ligand-Target Pair
TargetNAD-dependent protein deacetylase sirtuin-3, mitochondrial(Human)
Sirtris A Gsk
Curated by ChEMBL
Sirtris A Gsk
Curated by ChEMBL
Affinity DataIC50: 110nMAssay Description:Inhibition of human His-tagged SIRT3 (102 to 399) expressed in Escherichia coli BL21(DE3) assessed as inhibition of deacetylation of Ac-RHKKAcW-NH2 s...More data for this Ligand-Target Pair
TargetNAD-dependent protein deacetylase sirtuin-3, mitochondrial(Human)
Sirtris A Gsk
Curated by ChEMBL
Sirtris A Gsk
Curated by ChEMBL
Affinity DataIC50: 110nMAssay Description:Inhibition of recombinant human SIRT3 (118 to 399 residues) defatty-acylase activity expressed in Escherichia coli using SFP3 as substrate measured a...More data for this Ligand-Target Pair
TargetNAD-dependent protein deacetylase sirtuin-3, mitochondrial(Human)
Sirtris A Gsk
Curated by ChEMBL
Sirtris A Gsk
Curated by ChEMBL
Affinity DataIC50: 120nMAssay Description:Inhibition of human SIRT3 (118 to 399 aa) expressed in Escherichia coli BL21 cellsMore data for this Ligand-Target Pair
TargetNAD-dependent protein deacetylase sirtuin-3, mitochondrial(Human)
Sirtris A Gsk
Curated by ChEMBL
Sirtris A Gsk
Curated by ChEMBL
Affinity DataIC50: 130nMAssay Description:Inhibition of recombinant human SIRT3 (118 to 399 residues) demyristoylase activity expressed in Escherichia coli using p53(Myr)-AMC as substrate mea...More data for this Ligand-Target Pair
TargetNAD-dependent protein deacetylase sirtuin-3, mitochondrial(Human)
Sirtris A Gsk
Curated by ChEMBL
Sirtris A Gsk
Curated by ChEMBL
Affinity DataIC50: 150nMAssay Description:Inhibition of human His-tagged SIRT3 (102 to 399) expressed in Escherichia coli BL21(DE3) assessed as inhibition of deacetylation of Ac-RHKKAcW-NH2 s...More data for this Ligand-Target Pair
TargetNAD-dependent protein deacetylase sirtuin-3, mitochondrial(Human)
Sirtris A Gsk
Curated by ChEMBL
Sirtris A Gsk
Curated by ChEMBL
Affinity DataIC50: 170nMAssay Description:Inhibition of human SIRT3 (118 to 399 aa) expressed in Escherichia coli BL21 cellsMore data for this Ligand-Target Pair
TargetNAD-dependent protein deacetylase sirtuin-3, mitochondrial(Human)
Sirtris A Gsk
Curated by ChEMBL
Sirtris A Gsk
Curated by ChEMBL
Affinity DataIC50: 170nMAssay Description:Inhibition of human SIRT3 (118 to 399 aa) expressed in Escherichia coli BL21 cellsMore data for this Ligand-Target Pair
TargetNAD-dependent protein deacetylase sirtuin-3, mitochondrial(Human)
Sirtris A Gsk
Curated by ChEMBL
Sirtris A Gsk
Curated by ChEMBL
Affinity DataIC50: 180nMAssay Description:Inhibition of recombinant human SIRT3 (118 to 399 residues) defatty-acylase activity expressed in Escherichia coli using SFP3 as substrate measured a...More data for this Ligand-Target Pair
TargetNAD-dependent protein deacetylase sirtuin-3, mitochondrial(Human)
Sirtris A Gsk
Curated by ChEMBL
Sirtris A Gsk
Curated by ChEMBL
Affinity DataIC50: 190nMAssay Description:Inhibition of recombinant human SIRT3 (118 to 399 residues) demyristoylase activity expressed in Escherichia coli using p53(Myr)-AMC as substrate mea...More data for this Ligand-Target Pair
TargetNAD-dependent protein deacetylase sirtuin-3, mitochondrial(Human)
Sirtris A Gsk
Curated by ChEMBL
Sirtris A Gsk
Curated by ChEMBL
Affinity DataIC50: 210nMAssay Description:Inhibition of human SIRT3 (118 to 399 aa) expressed in Escherichia coli BL21 cellsMore data for this Ligand-Target Pair
TargetNAD-dependent protein deacetylase sirtuin-3, mitochondrial(Human)
Sirtris A Gsk
Curated by ChEMBL
Sirtris A Gsk
Curated by ChEMBL
Affinity DataIC50: 270nMAssay Description:Inhibition of recombinant His6 tagged human SIRT3 using 0.105 mM H2N-HK-[N(epsilon)-acetyl-lysine]-LM-COOH as substrate measured after 10 mins HPLC a...More data for this Ligand-Target Pair
TargetNAD-dependent protein deacetylase sirtuin-3, mitochondrial(Human)
Sirtris A Gsk
Curated by ChEMBL
Sirtris A Gsk
Curated by ChEMBL
Affinity DataIC50: 280nMAssay Description:Inhibition of human His-tagged SIRT3 (102 to 399) expressed in Escherichia coli BL21(DE3) assessed as inhibition of deacetylation of Ac-RHKKAcW-NH2 s...More data for this Ligand-Target Pair
TargetNAD-dependent protein deacetylase sirtuin-3, mitochondrial(Human)
Sirtris A Gsk
Curated by ChEMBL
Sirtris A Gsk
Curated by ChEMBL
Affinity DataIC50: 300nMAssay Description:Inhibition of human His-tagged SIRT3 (102 to 399) expressed in Escherichia coli BL21(DE3) assessed as inhibition of deacetylation of Ac-RHKKAcW-NH2 s...More data for this Ligand-Target Pair
TargetNAD-dependent protein deacetylase sirtuin-3, mitochondrial(Human)
Sirtris A Gsk
Curated by ChEMBL
Sirtris A Gsk
Curated by ChEMBL
Affinity DataIC50: 320nMAssay Description:Inhibition of human His6-tagged SIRT3 after 10 mins by HPLC analysis in presence of beta-NADMore data for this Ligand-Target Pair
TargetNAD-dependent protein deacetylase sirtuin-3, mitochondrial(Human)
Sirtris A Gsk
Curated by ChEMBL
Sirtris A Gsk
Curated by ChEMBL
Affinity DataIC50: 330nMAssay Description:Inhibition of recombinant human SIRT3 (118 to 399 residues) demyristoylase activity expressed in Escherichia coli using p53(Myr)-AMC as substrate mea...More data for this Ligand-Target Pair
TargetNAD-dependent protein deacetylase sirtuin-3, mitochondrial(Human)
Sirtris A Gsk
Curated by ChEMBL
Sirtris A Gsk
Curated by ChEMBL
Affinity DataIC50: 340nMAssay Description:Inhibition of recombinant human SIRT3 (118 to 399 residues) demyristoylase activity expressed in Escherichia coli using p53(Myr)-AMC as substrate mea...More data for this Ligand-Target Pair
TargetNAD-dependent protein deacetylase sirtuin-3, mitochondrial(Human)
Sirtris A Gsk
Curated by ChEMBL
Sirtris A Gsk
Curated by ChEMBL
Affinity DataIC50: 360nMAssay Description:Inhibition of human His6-tagged SIRT3 after 10 mins by HPLC analysis in presence of beta-NADMore data for this Ligand-Target Pair
TargetNAD-dependent protein deacetylase sirtuin-3, mitochondrial(Human)
Sirtris A Gsk
Curated by ChEMBL
Sirtris A Gsk
Curated by ChEMBL
Affinity DataIC50: 370nMAssay Description:Inhibition of human His-tagged SIRT3 (102 to 399) expressed in Escherichia coli BL21(DE3) assessed as inhibition of deacetylation of Ac-RHKKAcW-NH2 s...More data for this Ligand-Target Pair
TargetNAD-dependent protein deacetylase sirtuin-3, mitochondrial(Human)
Sirtris A Gsk
Curated by ChEMBL
Sirtris A Gsk
Curated by ChEMBL
Affinity DataIC50: 430nMAssay Description:Inhibition of human SIRT3 (118 to 399 aa) expressed in Escherichia coli BL21 cellsMore data for this Ligand-Target Pair
TargetNAD-dependent protein deacetylase sirtuin-3, mitochondrial(Human)
Sirtris A Gsk
Curated by ChEMBL
Sirtris A Gsk
Curated by ChEMBL
Affinity DataIC50: 450nMAssay Description:Inhibition of human His6-tagged SIRT3 after 10 mins by HPLC analysis in presence of beta-NADMore data for this Ligand-Target Pair
TargetNAD-dependent protein deacetylase sirtuin-3, mitochondrial(Human)
Sirtris A Gsk
Curated by ChEMBL
Sirtris A Gsk
Curated by ChEMBL
Affinity DataIC50: 470nMAssay Description:Inhibition of recombinant human His6-tagged SIRT3 using H2N-HK-[Nepsilon-acetyl-lysine]-LM-COOH as substrate incubated for 10 mins in presence of bet...More data for this Ligand-Target Pair
TargetNAD-dependent protein deacetylase sirtuin-3, mitochondrial(Human)
Sirtris A Gsk
Curated by ChEMBL
Sirtris A Gsk
Curated by ChEMBL
Affinity DataIC50: 480nMAssay Description:Inhibition of SIRT3 (unknown origin)More data for this Ligand-Target Pair
TargetNAD-dependent protein deacetylase sirtuin-3, mitochondrial(Human)
Sirtris A Gsk
Curated by ChEMBL
Sirtris A Gsk
Curated by ChEMBL
Affinity DataIC50: 480nMAssay Description:Inhibition of recombinant human SIRT3 (118 to 399 residues) demyristoylase activity expressed in Escherichia coli using p53(Myr)-AMC as substrate mea...More data for this Ligand-Target Pair
