Compile Data Set for Download or QSAR
Report error Found 53 of ic50 data for complexid = 50000795,50005878,50005882
TargetSomatostatin receptor type 1/2/3/4/5(Rat)
Diatide Research Laboaratories

Curated by ChEMBL
LigandPNGBDBM50476140(CHEMBL373632)
Affinity DataIC50: 0.100nMAssay Description:Displacement of [125I]SRIF-14 from SSTR of rat AR42J cell membranesMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetSomatostatin receptor type 1/2/3/4/5(Human)
Diatide Research Laboaratories

Curated by ChEMBL
LigandPNGBDBM50476134(CHEMBL437296)
Affinity DataIC50: 0.200nMAssay Description:Displacement of [125I-Tyr-11]-SRIF from SSTR of human NCI-H69 cell membranesMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSomatostatin receptor type 1/2/3/4/5(Rat)
Diatide Research Laboaratories

Curated by ChEMBL
LigandPNGBDBM81767(15-28-Somatostatin-28 | CB6417646 | CAS_38916-34-6...)
Affinity DataIC50: 0.200nMAssay Description:Compound was tested for its potency to displace 3-[125I]- - Tyr11-SRIF-14 from somatostatin receptor on membranes of rat cerebral cortexMore data for this Ligand-Target Pair
In DepthDetails

TargetSomatostatin receptor type 1/2/3/4/5(Mouse)
Phenex Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM392076(US10301272, Example 7/9)
Affinity DataIC50: 0.310nMAssay Description:Displacement of [125I]Tyr11-somatostatin-14 from mouse SST receptor after 60 mins by scintillation counting analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetSomatostatin receptor type 1/2/3/4/5(Human)
Diatide Research Laboaratories

Curated by ChEMBL
LigandPNGBDBM50476138(CHEMBL376485)
Affinity DataIC50: 0.350nMAssay Description:Displacement of [125I-Tyr-11]-SRIF from SSTR of human NCI-H69 cell membranesMore data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails Article
PubMed
TargetSomatostatin receptor type 1/2/3/4/5(Rat)
Diatide Research Laboaratories

Curated by ChEMBL
LigandPNGBDBM50476137(CHEMBL222751)
Affinity DataIC50: 0.400nMAssay Description:Displacement of [125I]SRIF-14 from SSTR of rat AR42J cell membranesMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetSomatostatin receptor type 1/2/3/4/5(Rat)
Diatide Research Laboaratories

Curated by ChEMBL
LigandPNGBDBM50214421(SOMATOSTATIN RECEPTOR LIGAND)
Affinity DataIC50: 0.430nMAssay Description:Compound was tested for its inhibitory effect against somatostatin receptor in rat cortex membrane using [125I]Tyr3-octreotide as the radioligandMore data for this Ligand-Target Pair
In DepthDetails

TargetSomatostatin receptor type 1/2/3/4/5(Rat)
Diatide Research Laboaratories

Curated by ChEMBL
LigandPNGBDBM81767(15-28-Somatostatin-28 | CB6417646 | CAS_38916-34-6...)
Affinity DataIC50: 0.430nMAssay Description:Compound was tested for its inhibitory effect against somatostatin receptor in rat cortex membrane using [125I]Tyr3-octreotide as the radioligandMore data for this Ligand-Target Pair
In DepthDetails

TargetSomatostatin receptor type 1/2/3/4/5(Human)
Diatide Research Laboaratories

Curated by ChEMBL
LigandPNGBDBM50212467(Sandostatinm)
Affinity DataIC50: 0.460nMAssay Description:Compound was tested for free energy of binding against somatostatin receptorMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails

TargetSomatostatin receptor type 1/2/3/4/5(Human)
Diatide Research Laboaratories

Curated by ChEMBL
LigandPNGBDBM50476142(CHEMBL376484)
Affinity DataIC50: 0.5nMAssay Description:Displacement of [125I-Tyr-11]-SRIF from SSTR of human NCI-H69 cell membranesMore data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails Article
PubMed
TargetSomatostatin receptor type 1/2/3/4/5(Human)
Diatide Research Laboaratories

Curated by ChEMBL
LigandPNGBDBM50476141(CHEMBL426548)
Affinity DataIC50: 0.640nMAssay Description:Displacement of [125I-Tyr-11]-SRIF from SSTR of human NCI-H69 cell membranesMore data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails Article
PubMed
TargetSomatostatin receptor type 1/2/3/4/5(Rat)
Diatide Research Laboaratories

Curated by ChEMBL
LigandPNGBDBM50476135(CHEMBL374316)
Affinity DataIC50: 0.700nMAssay Description:Displacement of [125I]SRIF-14 from SSTR of rat AR42J cell membranesMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetSomatostatin receptor type 1/2/3/4/5(Human)
Diatide Research Laboaratories

Curated by ChEMBL
LigandPNGBDBM50192018(CHEMBL3350037)
Affinity DataIC50: 1.10nMAssay Description:Displacement of [125I-Tyr-11]-SRIF from SSTR of human NCI-H69 cell membranesMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSomatostatin receptor type 1/2/3/4/5(Rat)
Diatide Research Laboaratories

Curated by ChEMBL
LigandPNGBDBM50476143(CHEMBL376001)
Affinity DataIC50: 1.5nMAssay Description:Displacement of [125I]SRIF-14 from SSTR of rat AR42J cell membranesMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetSomatostatin receptor type 1/2/3/4/5(Human)
Diatide Research Laboaratories

Curated by ChEMBL
LigandPNGBDBM50476139(CHEMBL268060)
Affinity DataIC50: 1.60nMAssay Description:Displacement of [125I-Tyr-11]-SRIF from SSTR of human NCI-H69 cell membranesMore data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails Article
PubMed
TargetSomatostatin receptor type 1/2/3/4/5(Human)
Diatide Research Laboaratories

Curated by ChEMBL
LigandPNGBDBM50476136(CHEMBL222699)
Affinity DataIC50: 1.60nMAssay Description:Displacement of [125I-Tyr-11]-SRIF from SSTR of human NCI-H69 cell membranesMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetSomatostatin receptor type 1/2/3/4/5(Human)
Diatide Research Laboaratories

Curated by ChEMBL
LigandPNGBDBM50008923(4-Ethyl-4-hydroxy-1,12-dihydro-4H-2-oxa-6,12a-diaz...)
Affinity DataIC50: 2.20nMAssay Description:Cytotoxic activity against human neuroblastoma IMR32 cells which over-express somatostatin receptorsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSomatostatin receptor type 1/2/3/4/5(Human)
Diatide Research Laboaratories

Curated by ChEMBL
LigandPNGBDBM50222716(CHEMBL2371535)
Affinity DataIC50: 2.80nMAssay Description:Cytotoxic activity against human neuroblastoma IMR32 cells which over-express somatostatin receptorsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSomatostatin receptor type 1/2/3/4/5(Rat)
Diatide Research Laboaratories

Curated by ChEMBL
LigandPNGBDBM50476144(CHEMBL434761)
Affinity DataIC50: 24nMAssay Description:Displacement of [125I]SRIF-14 from SSTR of rat AR42J cell membranesMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetSomatostatin receptor type 1/2/3/4/5(Human)
Diatide Research Laboaratories

Curated by ChEMBL
LigandPNGBDBM50222720(CHEMBL2371563)
Affinity DataIC50: 54nMAssay Description:Cytotoxic activity against human neuroblastoma IMR32 cells which over-express somatostatin receptorsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSomatostatin receptor type 1/2/3/4/5(Human)
Diatide Research Laboaratories

Curated by ChEMBL
LigandPNGBDBM50222719(CHEMBL2371564)
Affinity DataIC50: 571nMAssay Description:Cytotoxic activity against human neuroblastoma IMR32 cells which over-express somatostatin receptorsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSomatostatin receptor type 1/2/3/4/5(Rat)
Diatide Research Laboaratories

Curated by ChEMBL
LigandPNGBDBM50020202(CHEMBL2369466 | D-Tic-c(Cys-Tyr-D-Trp-Lys-Thr-Pen-...)
Affinity DataIC50: 949nMAssay Description:Binding affinity in competition with [125I]- CGP-23996 in somatostatin receptor binding to rat brain membraneMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSomatostatin receptor type 1/2/3/4/5(Human)
Diatide Research Laboaratories

Curated by ChEMBL
LigandPNGBDBM50222717(CHEMBL2371567)
Affinity DataIC50: 1.00E+3nMAssay Description:Cytotoxic activity against human neuroblastoma IMR32 cells which over-express somatostatin receptorsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSomatostatin receptor type 1/2/3/4/5(Human)
Diatide Research Laboaratories

Curated by ChEMBL
LigandPNGBDBM50222718(CHEMBL2371562)
Affinity DataIC50: 1.00E+3nMAssay Description:Cytotoxic activity against human neuroblastoma IMR32 cells which over-express somatostatin receptorsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSomatostatin receptor type 1/2/3/4/5(Mouse)
Phenex Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM81767(15-28-Somatostatin-28 | CB6417646 | CAS_38916-34-6...)
Affinity DataIC50: 1.30E+3nMAssay Description:Compound was tested for its binding affinity against somatostatin receptors on AtT-20 cellsMore data for this Ligand-Target Pair
In DepthDetails

TargetSomatostatin receptor type 1/2/3/4/5(Rat)
Diatide Research Laboaratories

Curated by ChEMBL
LigandPNGBDBM50020209(CHEMBL410090 | CTP)
Affinity DataIC50: 1.46E+3nMAssay Description:Binding affinity in competition with [125I]- CGP-23996 in somatostatin receptor binding to rat brain membraneMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSomatostatin receptor type 1/2/3/4/5(Rat)
Diatide Research Laboaratories

Curated by ChEMBL
LigandPNGBDBM50020205(CHEMBL216354 | D-Tic-c(Cys-Tyr-D-Trp-Lys-Thr-Pen-)...)
Affinity DataIC50: 1.50E+3nMAssay Description:Binding affinity in competition with [125I]- CGP-23996 in somatostatin receptor binding to rat brain membraneMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSomatostatin receptor type 1/2/3/4/5(Rat)
Diatide Research Laboaratories

Curated by ChEMBL
LigandPNGBDBM50020213(CHEMBL264082 | D-Trpc(-Cys-Tyr-D-Trp-Lys-Thr-Pen-)...)
Affinity DataIC50: 1.60E+3nMAssay Description:Binding affinity in competition with [125I]- CGP-23996 in somatostatin receptor binding to rat brain membraneMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSomatostatin receptor type 1/2/3/4/5(Rat)
Diatide Research Laboaratories

Curated by ChEMBL
LigandPNGBDBM50020211(CHEMBL216353 | D-Phec(-Cys-Tyr-D-Trp-Lys-Thr-Pen-)...)
Affinity DataIC50: 1.80E+3nMAssay Description:Binding affinity in competition with [125I]- CGP-23996 in somatostatin receptor binding to rat brain membraneMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSomatostatin receptor type 1/2/3/4/5(Rat)
Diatide Research Laboaratories

Curated by ChEMBL
LigandPNGBDBM50020216(CHEMBL413831 | D-Phec(-Cys-Tyr-D-Trp-Lys-Thr-Pen)-...)
Affinity DataIC50: 1.89E+3nMAssay Description:Binding affinity in competition with [125I]- CGP-23996 in somatostatin receptor binding to rat brain membraneMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSomatostatin receptor type 1/2/3/4/5(Rat)
Diatide Research Laboaratories

Curated by ChEMBL
LigandPNGBDBM50020198(CHEMBL308471 | D-Phec(-Cys-Tyr-D-Trp-Lys-Thr-Pen-)...)
Affinity DataIC50: 1.94E+3nMAssay Description:Binding affinity in competition with [125I]- CGP-23996 in somatostatin receptor binding to rat brain membraneMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSomatostatin receptor type 1/2/3/4/5(Rat)
Diatide Research Laboaratories

Curated by ChEMBL
LigandPNGBDBM50020200(CHEMBL405672 | D-Ticc(-Cys-Tyr-D-Typ-Lys-Thr-Pen-)...)
Affinity DataIC50: 1.99E+3nMAssay Description:Binding affinity in competition with [125I]- CGP-23996 in somatostatin receptor binding to rat brain membraneMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSomatostatin receptor type 1/2/3/4/5(Rat)
Diatide Research Laboaratories

Curated by ChEMBL
LigandPNGBDBM50020214(CHEMBL302596 | D-Phec(-Cys-Tyr-D-Trp-Lys-D-Pen-)Th...)
Affinity DataIC50: 6.10E+3nMAssay Description:Binding affinity in competition with [125I]- CGP-23996 in somatostatin receptor binding to rat brain membraneMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSomatostatin receptor type 1/2/3/4/5(Rat)
Diatide Research Laboaratories

Curated by ChEMBL
LigandPNGBDBM50214420(CHEMBL330352)
Affinity DataIC50: 6.50E+3nMAssay Description:Compound was tested for its inhibitory effect against somatostatin receptor in rat cortex membrane using [125I]Tyr3-octreotide as the radioligandMore data for this Ligand-Target Pair
In DepthDetails

TargetSomatostatin receptor type 1/2/3/4/5(Rat)
Diatide Research Laboaratories

Curated by ChEMBL
LigandPNGBDBM50214420(CHEMBL330352)
Affinity DataIC50: 7.00E+3nMAssay Description:Compound was tested for its inhibitory effect against somatostatin receptor in rat cortex membrane using [125I]Tyr3-octreotide as the radioligandMore data for this Ligand-Target Pair
In DepthDetails

TargetSomatostatin receptor type 1/2/3/4/5(Rat)
Diatide Research Laboaratories

Curated by ChEMBL
LigandPNGBDBM50214420(CHEMBL330352)
Affinity DataIC50: 7.00E+3nMAssay Description:Compound was tested for its inhibitory effect against somatostatin receptor in rat cortex membrane using [125I]Tyr3-octreotide as the radioligandMore data for this Ligand-Target Pair
In DepthDetails

TargetSomatostatin receptor type 1/2/3/4/5(Rat)
Diatide Research Laboaratories

Curated by ChEMBL
LigandPNGBDBM50020199(CHEMBL441164 | D-N-Me-Phec(-Cys-Tyr-D-Trp-Orn-Thr-...)
Affinity DataIC50: 8.05E+3nMAssay Description:Binding affinity in competition with [125I]- CGP-23996 in somatostatin receptor binding to rat brain membraneMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSomatostatin receptor type 1/2/3/4/5(Rat)
Diatide Research Laboaratories

Curated by ChEMBL
LigandPNGBDBM50020212(CHEMBL405244 | D-Phec(-Cys-Tyr-D-Trp-Lys-Thr-Pen-)...)
Affinity DataIC50: 8.30E+3nMAssay Description:Binding affinity in competition with [125I]- CGP-23996 in somatostatin receptor binding to rat brain membraneMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSomatostatin receptor type 1/2/3/4/5(Rat)
Diatide Research Laboaratories

Curated by ChEMBL
LigandPNGBDBM50020208(CHEMBL1795717 | TCTAP)
Affinity DataIC50: 8.45E+3nMAssay Description:Binding affinity in competition with [125I]- CGP-23996 in somatostatin receptor binding to rat brain membraneMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSomatostatin receptor type 1/2/3/4/5(Rat)
Diatide Research Laboaratories

Curated by ChEMBL
LigandPNGBDBM50020204(CHEMBL66403 | D-Phec(-Cys-Tyr-Asn-Pen-)Thr-NH2)
Affinity DataIC50: 1.00E+4nMAssay Description:Binding affinity in competition with [125I]- CGP-23996 in somatostatin receptor binding to rat brain membraneMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSomatostatin receptor type 1/2/3/4/5(Rat)
Diatide Research Laboaratories

Curated by ChEMBL
LigandPNGBDBM50213874(CHEMBL432503)
Affinity DataIC50: 1.00E+4nMAssay Description:Compound was tested for its potency to displace 3-[125I]- - Tyr11-SRIF-14 from somatostatin receptor on membranes of rat cerebral cortexMore data for this Ligand-Target Pair
In DepthDetails

TargetSomatostatin receptor type 1/2/3/4/5(Rat)
Diatide Research Laboaratories

Curated by ChEMBL
LigandPNGBDBM50213872(CHEMBL47019)
Affinity DataIC50: 1.10E+4nMAssay Description:Compound was tested for its potency to displace 3-[125I]- - Tyr11-SRIF-14 from somatostatin receptor on membranes of rat cerebral cortexMore data for this Ligand-Target Pair
In DepthDetails

TargetSomatostatin receptor type 1/2/3/4/5(Rat)
Diatide Research Laboaratories

Curated by ChEMBL
LigandPNGBDBM50213871(CHEMBL47648)
Affinity DataIC50: 1.20E+4nMAssay Description:Compound was tested for its potency to displace 3-[125I]- - Tyr11-SRIF-14 from somatostatin receptor on membranes of rat cerebral cortexMore data for this Ligand-Target Pair
In DepthDetails

TargetSomatostatin receptor type 1/2/3/4/5(Rat)
Diatide Research Laboaratories

Curated by ChEMBL
LigandPNGBDBM50213869(CHEMBL3037859)
Affinity DataIC50: 1.20E+4nMAssay Description:Compound was tested for its potency to displace 3-[125I]- - Tyr11-SRIF-14 from somatostatin receptor on membranes of rat cerebral cortexMore data for this Ligand-Target Pair
In DepthDetails

TargetSomatostatin receptor type 1/2/3/4/5(Rat)
Diatide Research Laboaratories

Curated by ChEMBL
LigandPNGBDBM50452485(CHEMBL2369462)
Affinity DataIC50: 1.36E+4nMAssay Description:Binding affinity in competition with [125I]- CGP-23996 in somatostatin receptor binding to rat brain membraneMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSomatostatin receptor type 1/2/3/4/5(Rat)
Diatide Research Laboaratories

Curated by ChEMBL
LigandPNGBDBM50213870(CHEMBL294905)
Affinity DataIC50: 1.40E+4nMAssay Description:Compound was tested for its potency to displace 3-[125I]- - Tyr11-SRIF-14 from somatostatin receptor on membranes of rat cerebral cortexMore data for this Ligand-Target Pair
In DepthDetails

TargetSomatostatin receptor type 1/2/3/4/5(Rat)
Diatide Research Laboaratories

Curated by ChEMBL
LigandPNGBDBM50213873(CHEMBL45323)
Affinity DataIC50: 1.50E+4nMAssay Description:Compound was tested for its potency to displace 3-[125I]- - Tyr11-SRIF-14 from somatostatin receptor on membranes of rat cerebral cortexMore data for this Ligand-Target Pair
In DepthDetails

TargetSomatostatin receptor type 1/2/3/4/5(Rat)
Diatide Research Laboaratories

Curated by ChEMBL
LigandPNGBDBM50020207(CHEMBL2369473 | Gly-D-Ticc(-Cys-Tyr-D-Trp-Orn-Thr-...)
Affinity DataIC50: 1.94E+4nMAssay Description:Binding affinity in competition with [125I]- CGP-23996 in somatostatin receptor binding to rat brain membraneMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSomatostatin receptor type 1/2/3/4/5(Rat)
Diatide Research Laboaratories

Curated by ChEMBL
LigandPNGBDBM50020197(CHEMBL2369475 | TCTOP)
Affinity DataIC50: 2.04E+4nMAssay Description:Binding affinity in competition with [125I]- CGP-23996 in somatostatin receptor binding to rat brain membraneMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSomatostatin receptor type 1/2/3/4/5(Rat)
Diatide Research Laboaratories

Curated by ChEMBL
LigandPNGBDBM50212468(CHEMBL28415)
Affinity DataIC50: 2.30E+4nMAssay Description:Radioligand binding studies on rat cortex membranes using 125 I-Tyrs-octreotide as ligand was determinedMore data for this Ligand-Target Pair
In DepthDetails

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