Compile Data Set for Download or QSAR
Report error Found 203 of ic50 data for complexid = 50000780,50005827
TargetVasopressin V1a/V1b receptor(Human)
Central Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50137948(Biphenyl-2-carboxylic acid [2-[3-(4-methyl-[1,4]di...)
Affinity DataIC50: 1nMAssay Description:Inhibitory activity against arginine vasopressin V1 receptor using [3H]AVP as radioligand in human plateletMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetVasopressin V1a/V1b receptor(Rat)
Central Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50137948(Biphenyl-2-carboxylic acid [2-[3-(4-methyl-[1,4]di...)
Affinity DataIC50: 2nMAssay Description:Inhibitory activity against arginine vasopressin V1 receptor using [3H]AVP as radioligand in rat liverMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetVasopressin V1a/V1b receptor(Rat)
Central Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50137945(Biphenyl-2-carboxylic acid [2-[4-(4-methyl-piperaz...)
Affinity DataIC50: 3nMAssay Description:Inhibitory activity against arginine vasopressin V1 receptor using [3H]AVP as radioligand in rat liverMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetVasopressin V1a/V1b receptor(Human)
Central Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50137940(Biphenyl-2-carboxylic acid [2-[4-(4-dimethylamino-...)
Affinity DataIC50: 3nMAssay Description:Inhibitory activity against arginine vasopressin V1 receptor using [3H]AVP as radioligand in human plateletMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetVasopressin V1a/V1b receptor(Human)
Central Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50137953(Biphenyl-2-carboxylic acid [2-[4-(4-diethylamino-p...)
Affinity DataIC50: 4nMAssay Description:Inhibitory activity against arginine vasopressin V1 receptor using [3H]AVP as radioligand in human plateletMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetVasopressin V1a/V1b receptor(Rat)
Central Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50137953(Biphenyl-2-carboxylic acid [2-[4-(4-diethylamino-p...)
Affinity DataIC50: 4nMAssay Description:Inhibitory activity against arginine vasopressin V1 receptor using [3H]AVP as radioligand in rat liverMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetVasopressin V1a/V1b receptor(Human)
Central Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50137945(Biphenyl-2-carboxylic acid [2-[4-(4-methyl-piperaz...)
Affinity DataIC50: 5nMAssay Description:Inhibitory activity against arginine vasopressin V1 receptor using [3H]AVP as radioligand in human plateletMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetVasopressin V1a/V1b receptor(Human)
Central Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50137951(Biphenyl-2-carboxylic acid [2-{4-[(2-dimethylamino...)
Affinity DataIC50: 5nMAssay Description:Inhibitory activity against arginine vasopressin V1 receptor using [3H]AVP as radioligand in human plateletMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetVasopressin V1a/V1b receptor(Rat)
Central Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50137940(Biphenyl-2-carboxylic acid [2-[4-(4-dimethylamino-...)
Affinity DataIC50: 6nMAssay Description:Inhibitory activity against arginine vasopressin V1 receptor using [3H]AVP as radioligand in rat liverMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetVasopressin V1a/V1b receptor(Rat)
Central Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50291329(8-arginine vasopressin trisulphide | CHEMBL267405)
Affinity DataIC50: 9.5nMAssay Description:Tested for the TYR(Me)2 arginine-vasopressin as radioligand at 0.3 nM in A7r5 cellsMore data for this Ligand-Target Pair
In DepthDetails Article

TargetVasopressin V1a/V1b receptor(Rat)
Central Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM35667([3H]Argipressin tannate | AVP | [3H]Arginine vasop...)
Affinity DataIC50: 10nMAssay Description:Tested for the TYR(Me)2 arginine-vasopressin as radioligand at 0.3 nM in A7r5 cellsMore data for this Ligand-Target Pair
In DepthDetails Article

TargetVasopressin V1a/V1b receptor(Human)
Central Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50137942(Biphenyl-2-carboxylic acid [2-(4-[1,4']bipiperidin...)
Affinity DataIC50: 10nMAssay Description:Inhibitory activity against arginine vasopressin V1 receptor using [3H]AVP as radioligand in human plateletMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetVasopressin V1a/V1b receptor(Human)
Central Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50137956(Biphenyl-2-carboxylic acid [2-[4-(4-methyl-piperaz...)
Affinity DataIC50: 10nMAssay Description:Inhibitory activity against arginine vasopressin V1 receptor using [3H]AVP as radioligand in human plateletMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetVasopressin V1a/V1b receptor(Rat)
Central Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50137949(Biphenyl-2-carboxylic acid [2-[4-(4-methyl-[1,4]di...)
Affinity DataIC50: 20nMAssay Description:Inhibitory activity against arginine vasopressin V1 receptor using [3H]AVP as radioligand in rat liverMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetVasopressin V1a/V1b receptor(Rat)
Central Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50137951(Biphenyl-2-carboxylic acid [2-{4-[(2-dimethylamino...)
Affinity DataIC50: 20nMAssay Description:Inhibitory activity against arginine vasopressin V1 receptor using [3H]AVP as radioligand in rat liverMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetVasopressin V1a/V1b receptor(Rat)
Central Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50137946(Biphenyl-2-carboxylic acid [2-[2-(4-dimethylamino-...)
Affinity DataIC50: 20nMAssay Description:Inhibitory activity against arginine vasopressin V1 receptor using [3H]AVP as radioligand in rat liverMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetVasopressin V1a/V1b receptor(Rat)
Central Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50137942(Biphenyl-2-carboxylic acid [2-(4-[1,4']bipiperidin...)
Affinity DataIC50: 20nMAssay Description:Inhibitory activity against arginine vasopressin V1 receptor using [3H]AVP as radioligand in rat liverMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetVasopressin V1a/V1b receptor(Rat)
Central Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50137956(Biphenyl-2-carboxylic acid [2-[4-(4-methyl-piperaz...)
Affinity DataIC50: 20nMAssay Description:Inhibitory activity against arginine vasopressin V1 receptor using [3H]AVP as radioligand in rat liverMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetVasopressin V1a/V1b receptor(Human)
Central Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50137949(Biphenyl-2-carboxylic acid [2-[4-(4-methyl-[1,4]di...)
Affinity DataIC50: 50nMAssay Description:Inhibitory activity against arginine vasopressin V1 receptor using [3H]AVP as radioligand in human plateletMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetVasopressin V1a/V1b receptor(Human)
Central Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50137946(Biphenyl-2-carboxylic acid [2-[2-(4-dimethylamino-...)
Affinity DataIC50: 50nMAssay Description:Inhibitory activity against arginine vasopressin V1 receptor using [3H]AVP as radioligand in human plateletMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetVasopressin V1a/V1b receptor(Human)
Central Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50204026(CHEMBL369150)
Affinity DataIC50: 60nMAssay Description:Inhibitory activity against arginine vasopressin V1 receptor using [3H]AVP as radioligand in human plateletMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetVasopressin V1a/V1b receptor(Rat)
Central Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50043204(1N-[2-hydroxy-7,7-dimethyl-1-spiro[1H-indene-1,4'-...)
Affinity DataIC50: 67nMAssay Description:Inhibition of radioligand [3H]AVP binding to the vasopressin V1 receptor in rat liver tissueMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetVasopressin V1a/V1b receptor(Rat)
Central Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50043080(3-[7,7-dimethyl-1-spiro[2,3-dihydro-1H-indene-1,4'...)
Affinity DataIC50: 110nMAssay Description:Inhibition of radioligand [3H]AVP binding to the vasopressin V1 receptor in rat liver tissueMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetVasopressin V1a/V1b receptor(Rat)
Central Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50043141(5-(3-amino-1H-1,2,4-triazol-5-ylaminomethyl)-3-[7,...)
Affinity DataIC50: 120nMAssay Description:Inhibition of radioligand [3H]AVP binding to the vasopressin V1 receptor in rat liver tissueMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetVasopressin V1a/V1b receptor(Rat)
Central Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50043114(3-{1-[7,7-dimethyl-1-spiro[2,3-dihydro-1H-indene-1...)
Affinity DataIC50: 160nMAssay Description:Inhibition of radioligand [3H]AVP binding to the vasopressin V1 receptor in rat liver tissueMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetVasopressin V1a/V1b receptor(Rat)
Central Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50137943(Biphenyl-2-carboxylic acid (4-{8-[2-(4-methyl-pipe...)
Affinity DataIC50: 200nMAssay Description:Inhibitory activity against arginine vasopressin V1 receptor using [3H]AVP as radioligand in rat liverMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetVasopressin V1a/V1b receptor(Rat)
Central Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50137941(Biphenyl-2-carboxylic acid {4-[8-(2-pyrrolidin-1-y...)
Affinity DataIC50: 200nMAssay Description:Inhibitory activity against arginine vasopressin V1 receptor using [3H]AVP as radioligand in rat liverMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetVasopressin V1a/V1b receptor(Rat)
Central Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50204026(CHEMBL369150)
Affinity DataIC50: 200nMAssay Description:Inhibitory activity against arginine vasopressin V1 receptor using [3H]AVP as radioligand in rat liverMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetVasopressin V1a/V1b receptor(Rat)
Central Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50043180(1N-[2-hydroxy-7,7-dimethyl-1-spiro[1H-indene-1,4'-...)
Affinity DataIC50: 290nMAssay Description:Inhibition of radioligand [3H]AVP binding to the vasopressin V1 receptor in rat liver tissueMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetVasopressin V1a/V1b receptor(Rat)
Central Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50137954(Biphenyl-2-carboxylic acid {4-[8-(2-dimethylamino-...)
Affinity DataIC50: 300nMAssay Description:Inhibitory activity against arginine vasopressin V1 receptor using [3H]AVP as radioligand in rat liverMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetVasopressin V1a/V1b receptor(Rat)
Central Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50043088(3-[7,7-dimethyl-1-spiro[2,3-dihydro-1H-indene-1,4'...)
Affinity DataIC50: 300nMAssay Description:Inhibition of radioligand [3H]AVP binding to the vasopressin V1 receptor in rat liver tissueMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetVasopressin V1a/V1b receptor(Rat)
Central Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50043117(1-[7,7-dimethyl-1-spiro[2,3-dihydro-1H-indene-1,4'...)
Affinity DataIC50: 300nMAssay Description:Inhibition of radioligand [3H]AVP binding to the vasopressin V1 receptor in rat liver tissueMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetVasopressin V1a/V1b receptor(Rat)
Central Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50043075(1N-[7,7-dimethyl-1-spiro[2,3-dihydro-1H-indene-1,4...)
Affinity DataIC50: 300nMAssay Description:Inhibition of radioligand [3H]AVP binding to the vasopressin V1 receptor in rat liver tissueMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetVasopressin V1a/V1b receptor(Rat)
Central Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50043106(methyl 3-[2-hydroxy-7,7-dimethyl-1-spiro[1H-indene...)
Affinity DataIC50: 300nMAssay Description:Inhibition of radioligand [3H]AVP binding to the vasopressin V1 receptor in rat liver tissueMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetVasopressin V1a/V1b receptor(Rat)
Central Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50043155(1N-[7,7-dimethyl-1-spiro[2,3-dihydro-1H-indene-1,4...)
Affinity DataIC50: 300nMAssay Description:Inhibition of radioligand [3H]AVP binding to the vasopressin V1 receptor in rat liver tissueMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetVasopressin V1a/V1b receptor(Rat)
Central Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50043055(2-{3-[7,7-dimethyl-1-spiro[2,3-dihydro-1H-indene-1...)
Affinity DataIC50: 300nMAssay Description:Inhibition of radioligand [3H]AVP binding to the vasopressin V1 receptor in rat liver tissueMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetVasopressin V1a/V1b receptor(Rat)
Central Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50043090(1N-[2-hydroxy-7,7-dimethyl-1-spiro[1H-indene-1,4'-...)
Affinity DataIC50: 300nMAssay Description:Inhibition of radioligand [3H]AVP binding to the vasopressin V1 receptor in rat liver tissueMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetVasopressin V1a/V1b receptor(Rat)
Central Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50043145(3N-[2-hydroxy-7,7-dimethyl-1-spiro[1H-indene-1,4'-...)
Affinity DataIC50: 300nMAssay Description:Inhibition of radioligand [3H]AVP binding to the vasopressin V1 receptor in rat liver tissueMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetVasopressin V1a/V1b receptor(Rat)
Central Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50043059(1N-[2-hydroxy-7,7-dimethyl-1-spiro[1H-indene-1,4'-...)
Affinity DataIC50: 300nMAssay Description:Inhibition of radioligand [3H]AVP binding to the vasopressin V1 receptor in rat liver tissueMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetVasopressin V1a/V1b receptor(Rat)
Central Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50043116(1N-{2-[2-hydroxy-7,7-dimethyl-1-spiro[1H-indene-1,...)
Affinity DataIC50: 300nMAssay Description:Inhibition of radioligand [3H]AVP binding to the vasopressin V1 receptor in rat liver tissueMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetVasopressin V1a/V1b receptor(Rat)
Central Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50043189(1N-[7,7-dimethyl-1-spiro[2,3-dihydro-1H-indene-1,4...)
Affinity DataIC50: 300nMAssay Description:Inhibition of radioligand [3H]AVP binding to the vasopressin V1 receptor in rat liver tissueMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetVasopressin V1a/V1b receptor(Rat)
Central Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50043143(1N-[2-hydroxy-7,7-dimethyl-1-spiro[1H-indene-1,4'-...)
Affinity DataIC50: 310nMAssay Description:Inhibition of radioligand [3H]AVP binding to the vasopressin V1 receptor in rat liver tissueMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetVasopressin V1a/V1b receptor(Rat)
Central Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50043120(1N-[7,7-dimethyl-1-spiro[2,3-dihydro-1H-indene-1,4...)
Affinity DataIC50: 320nMAssay Description:Inhibition of radioligand [3H]AVP binding to the vasopressin V1 receptor in rat liver tissueMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetVasopressin V1a/V1b receptor(Rat)
Central Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50043093(3-[7,7-dimethyl-1-spiro[2,3-dihydro-1H-indene-1,4'...)
Affinity DataIC50: 370nMAssay Description:Inhibition of radioligand [3H]AVP binding to the vasopressin V1 receptor in rat liver tissueMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetVasopressin V1a/V1b receptor(Human)
Central Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50137954(Biphenyl-2-carboxylic acid {4-[8-(2-dimethylamino-...)
Affinity DataIC50: 400nMAssay Description:Inhibitory activity against arginine vasopressin V1 receptor using [3H]AVP as radioligand in human plateletMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetVasopressin V1a/V1b receptor(Human)
Central Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50137947(Biphenyl-2-carboxylic acid [4-(8-benzyl-5,6,7,8-te...)
Affinity DataIC50: 400nMAssay Description:Inhibitory activity against arginine vasopressin V1 receptor using [3H]AVP as radioligand in human plateletMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetVasopressin V1a/V1b receptor(Rat)
Central Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50043077(2-{1-[7,7-dimethyl-1-spiro[2,3-dihydro-1H-indene-1...)
Affinity DataIC50: 410nMAssay Description:Inhibition of radioligand [3H]AVP binding to the vasopressin V1 receptor in rat liver tissueMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetVasopressin V1a/V1b receptor(Rat)
Central Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50043118(3-[7,7-dimethyl-1-spiro[2,3-dihydro-1H-indene-1,4'...)
Affinity DataIC50: 420nMAssay Description:Inhibition of radioligand [3H]AVP binding to the vasopressin V1 receptor in rat liver tissueMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetVasopressin V1a/V1b receptor(Rat)
Central Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50043118(3-[7,7-dimethyl-1-spiro[2,3-dihydro-1H-indene-1,4'...)
Affinity DataIC50: 420nMAssay Description:Inhibition of radioligand [3H]AVP binding to the vasopressin V1 receptor in rat liver tissueMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetVasopressin V1a/V1b receptor(Rat)
Central Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50043118(3-[7,7-dimethyl-1-spiro[2,3-dihydro-1H-indene-1,4'...)
Affinity DataIC50: 420nMAssay Description:Inhibition of radioligand [3H]AVP binding to the vasopressin V1 receptor in rat liver tissueMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
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