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Report error Found 9 of ic50 data for complexid = 50000653
TargetCasein kinase I isoform alpha/delta/epsilon/gamma-1/gamma-2(Human)
Sichuan University-Oxford University Huaxi Gastrointestinal Cancer Centre

Curated by ChEMBL
LigandPNGBDBM50335638(5-(3-Chlorophenylamino)benzo[c][2,6]naphthyridine-...)
Affinity DataIC50: 4nMAssay Description:Inhibition of CK1 (unknown origin)More data for this Ligand-Target Pair
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PubMed
TargetCasein kinase I isoform alpha/delta/epsilon/gamma-1/gamma-2(Human)
Sichuan University-Oxford University Huaxi Gastrointestinal Cancer Centre

Curated by ChEMBL
LigandPNGBDBM50587013(CHEMBL5091216)
Affinity DataIC50: 230nMAssay Description:Inhibition of CK1 (unknown origin)More data for this Ligand-Target Pair
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PubMed
TargetCasein kinase I isoform alpha/delta/epsilon/gamma-1/gamma-2(Human)
Sichuan University-Oxford University Huaxi Gastrointestinal Cancer Centre

Curated by ChEMBL
LigandPNGBDBM50229971(4-[4-(2,3-dihydro-benzo[1,4]dioxin-6-yl)-5-pyridin...)
Affinity DataIC50: 300nMAssay Description:Inhibition of human CK1 in presence of [gamma33P]-ATPMore data for this Ligand-Target Pair
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PubMed
TargetCasein kinase I isoform alpha/delta/epsilon/gamma-1/gamma-2(Human)
Sichuan University-Oxford University Huaxi Gastrointestinal Cancer Centre

Curated by ChEMBL
LigandPNGBDBM2579(CHEMBL388978 | Staurosporine, 8 | Staurosporin, 4 ...)
Affinity DataIC50: 1.40E+3nMAssay Description:Inhibition of Casein kinase IMore data for this Ligand-Target Pair
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PubMed
TargetCasein kinase I isoform alpha/delta/epsilon/gamma-1/gamma-2(Human)
Sichuan University-Oxford University Huaxi Gastrointestinal Cancer Centre

Curated by ChEMBL
LigandPNGBDBM50169892(3-{4-[4-(3-Chloro-phenylamino)-[1,3,5]triazin-2-yl...)
Affinity DataIC50: 3.05E+3nMAssay Description:Inhibition of Casein kinase IMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCasein kinase I isoform alpha/delta/epsilon/gamma-1/gamma-2(Human)
Sichuan University-Oxford University Huaxi Gastrointestinal Cancer Centre

Curated by ChEMBL
LigandPNGBDBM50179207(JNJ-10198409 | 3-fluoro-N-(6,7-dimethoxy-2,4-dihyd...)
Affinity DataIC50: 7.20E+3nMAssay Description:Inhibitory activity against Casein Kinase 1More data for this Ligand-Target Pair
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PubMed
TargetCasein kinase I isoform alpha/delta/epsilon/gamma-1/gamma-2(Human)
Sichuan University-Oxford University Huaxi Gastrointestinal Cancer Centre

Curated by ChEMBL
LigandPNGBDBM92674(Isoquinolinesulfonamide, CKI-7)
Affinity DataIC50: 9.50E+3nMAssay Description:Inhibition of CK1 (unknown origin)More data for this Ligand-Target Pair
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PubMed
TargetCasein kinase I isoform alpha/delta/epsilon/gamma-1/gamma-2(Human)
Sichuan University-Oxford University Huaxi Gastrointestinal Cancer Centre

Curated by ChEMBL
LigandPNGBDBM50139822(10-Chloro-6-hydroxy-pyrido[1,2-a]quinolinylium; ch...)
Affinity DataIC50: 3.30E+4nMAssay Description:Inhibition of casein kinase IMore data for this Ligand-Target Pair
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TargetCasein kinase I isoform alpha/delta/epsilon/gamma-1/gamma-2(Human)
Sichuan University-Oxford University Huaxi Gastrointestinal Cancer Centre

Curated by ChEMBL
LigandPNGBDBM50132310(20-ethyl-17,23-dioxa-4,14,20,26-tetraazahexacyclo[...)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of Casein kinase IMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed