Compile Data Set for Download or QSAR
Report error Found 249 of ic50 data for complexid = 50000024
LigandPNGBDBM50191913(N-(2-methyl-4-(2-(pyrrolidin-1-yl)ethyl)phenyl)-4-...)
Affinity DataIC50: 0.600nMAssay Description:Inhibition of CDK1/cyclinB by Flashplate assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50191929(2-(4-(4-(1H-pyrrolo[2,3-b]pyridin-3-yl)pyrimidin-2...)
Affinity DataIC50: 0.600nMAssay Description:Inhibition of CDK1/cyclinB by Flashplate assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50191918(N-(2-methyl-4-(2-(piperidin-1-yl)ethyl)phenyl)-4-(...)
Affinity DataIC50: 1nMAssay Description:Inhibition of CDK1/cyclinB by Flashplate assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50191924(N-(2-methyl-4-(2-morpholinoethyl)phenyl)-4-(1H-pyr...)
Affinity DataIC50: 1.90nMAssay Description:Inhibition of CDK1/cyclinB by Flashplate assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50191922(trans-N1-(4-(1H-pyrrolo[2,3-b]pyridin-3-yl)pyrimid...)
Affinity DataIC50: 2nMAssay Description:Inhibition of CDK1/cyclinB by Flashplate assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM2579(CHEMBL388978 | Staurosporine, 8 | Staurosporin, 4 ...)
Affinity DataIC50: 2.5nMAssay Description:Inhibition of CDK1/cyclin B (unknown origin) after 40 mins by scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50191925(4-(1H-pyrrolo[2,3-b]pyridin-3-yl)-N-o-tolylpyrimid...)
Affinity DataIC50: 3nMAssay Description:Inhibition of CDK1/cyclinB by Flashplate assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM2579(CHEMBL388978 | Staurosporine, 8 | Staurosporin, 4 ...)
Affinity DataIC50: 3.20nMAssay Description:Inhibition of CDK1/cyclin BMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50338873(N-(5-Amino-1-(4-methoxybenzyl)-1H-pyrazol-4-yl)-5-...)
Affinity DataIC50: 3.20nMAssay Description:Inhibition of CDK1/cyclin BMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM27216((2R)-2-({6-[(3-chlorophenyl)amino]-9-(propan-2-yl)...)
Affinity DataIC50: 4nMAssay Description:Inhibition of Cyclin B-cyclin-dependent kinase 1More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM2579(CHEMBL388978 | Staurosporine, 8 | Staurosporin, 4 ...)
Affinity DataIC50: 6nMAssay Description:Inhibition of CDK1/cyclinBMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM7478(CHEMBL23254 | 2-chloro-4-[(2-{[(2R)-1-hydroxy-3-me...)
Affinity DataIC50: 6nMAssay Description:Inhibition of cyclin dependent kinase 1-cyclinBMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50191914(N-(2-chlorophenyl)-4-(1H-pyrrolo[2,3-b]pyridin-3-y...)
Affinity DataIC50: 9nMAssay Description:Inhibition of CDK1/cyclinB by Flashplate assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM2579(CHEMBL388978 | Staurosporine, 8 | Staurosporin, 4 ...)
Affinity DataIC50: 12nMAssay Description:Inhibition of Cyclin B-cyclin-dependent kinase 1More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50191919(N-(2-bromophenyl)-4-(1H-pyrrolo[2,3-b]pyridin-3-yl...)
Affinity DataIC50: 13nMAssay Description:Inhibition of CDK1/cyclinB by Flashplate assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50191912(N-cyclohexyl-4-(1H-pyrrolo[2,3-b]pyridin-3-yl)pyri...)
Affinity DataIC50: 14nMAssay Description:Inhibition of CDK1/cyclinB by Flashplate assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50132003((Z)-1H,1''H-[2,3'']Biindolylidene-3,2''-dione 3-ox...)
Affinity DataIC50: 18nMAssay Description:Inhibition of CDK1/cyclinBMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50366800(OLOMOUCINE II)
Affinity DataIC50: 20nMAssay Description:Inhibition of recombinant Cyclin-dependent kinase 1-cyclin BMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50169892(3-{4-[4-(3-Chloro-phenylamino)-[1,3,5]triazin-2-yl...)
Affinity DataIC50: 21nMAssay Description:Inhibition of CDK1/cyclin BMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM7491(4-[2-Amino-5-oxo-1,5-dihydro-imidazol-(4Z)-ylidene...)
Affinity DataIC50: 22nMAssay Description:Inhibition of CDK1/cyclinBMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM7238(cid_5289419 | 3-(3H-Imidazol-4-ylmethylene)-5-meth...)
Affinity DataIC50: 22nMAssay Description:Inhibition of CDK1/cyclinBMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM7263(CHEMBL299756 | 9-oxo-8,18-diazatetracyclo[9.7.0.0^...)
Affinity DataIC50: 24nMAssay Description:Inhibition of CDK1/cyclin B expressed in M phase starfish oocyteMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50191928(1-(3-(2-(cyclohexylamino)pyrimidin-4-yl)-1H-pyrrol...)
Affinity DataIC50: 31nMAssay Description:Inhibition of CDK1/cyclinB by Flashplate assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM7262(NSC 705701 | BDBM84528 | alsterpaullone | 9-Nitrop...)
Affinity DataIC50: 35nMAssay Description:Inhibition of CDK1/cyclin B expressed in M phase starfish oocyteMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM7262(NSC 705701 | BDBM84528 | alsterpaullone | 9-Nitrop...)
Affinity DataIC50: 35nMAssay Description:Inhibition of CDK1/cyclinBMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50191916(4-(1H-pyrrolo[2,3-b]pyridin-3-yl)-N-p-tolylpyrimid...)
Affinity DataIC50: 40nMAssay Description:Inhibition of CDK1/cyclinB by Flashplate assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50191923(N-(2-methoxyphenyl)-4-(1H-pyrrolo[2,3-b]pyridin-3-...)
Affinity DataIC50: 44nMAssay Description:Inhibition of CDK1/cyclinB by Flashplate assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM7265(NSC 708244 | 4,5-dimethoxy-9-oxo-8,18-diazatetracy...)
Affinity DataIC50: 44nMAssay Description:Inhibition of CDK1/cyclin B expressed in M phase starfish oocyteMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
LigandPNGBDBM50191932(N-(2-fluorophenyl)-4-(1H-pyrrolo[2,3-b]pyridin-3-y...)
Affinity DataIC50: 46nMAssay Description:Inhibition of CDK1/cyclinB by Flashplate assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM7269(CHEMBL121492 | 3-[9-oxo-14-(trifluoromethyl)-8,18-...)
Affinity DataIC50: 47nMAssay Description:Inhibition of Cyclin-dependent kinase 1-cyclin B from Starfish oocytesMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM27216((2R)-2-({6-[(3-chlorophenyl)amino]-9-(propan-2-yl)...)
Affinity DataIC50: 50nMAssay Description:Inhibition of recombinant Cyclin-dependent kinase 1-cyclin BMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50191917(N-phenyl-4-(1H-pyrrolo[2,3-b]pyridin-3-yl)pyrimidi...)
Affinity DataIC50: 54nMAssay Description:Inhibition of CDK1/cyclinB by Flashplate assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50191926(4-(1H-pyrrolo[2,3-b]pyridin-3-yl)-N-(2-(trifluorom...)
Affinity DataIC50: 56nMAssay Description:Inhibition of CDK1/cyclinB by Flashplate assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50335638(5-(3-Chlorophenylamino)benzo[c][2,6]naphthyridine-...)
Affinity DataIC50: 56nMAssay Description:Inhibition of human recombinant CDK1/Cyclin B by radiometric assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50191920(4-(1H-pyrrolo[2,3-b]pyridin-3-yl)-N-m-tolylpyrimid...)
Affinity DataIC50: 57nMAssay Description:Inhibition of CDK1/cyclinB by Flashplate assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50191915(N-(2-ethylphenyl)-4-(1H-pyrrolo[2,3-b]pyridin-3-yl...)
Affinity DataIC50: 68nMAssay Description:Inhibition of CDK1/cyclinB by Flashplate assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM10642(CHEMBL83320 | 2-[({2-[(1-hydroxy-3-methylbutan-2-y...)
Affinity DataIC50: 80nMAssay Description:Inhibition of recombinant Cyclin-dependent kinase 1-cyclin BMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50120508(2-(3-hydroxypropylamino)-6-(o -hydroxybenzylamino)...)
Affinity DataIC50: 100nMAssay Description:Inhibition of recombinant Cyclin-dependent kinase 1-cyclin BMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM10635(3-{[(2-{[1-(hydroxymethyl)-2-methylpropyl]amino}-9...)
Affinity DataIC50: 120nMAssay Description:Inhibition of recombinant Cyclin-dependent kinase 1-cyclin BMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50191921(N-cyclohexyl-4-(1-(methylsulfonyl)-1H-pyrrolo[2,3-...)
Affinity DataIC50: 128nMAssay Description:Inhibition of CDK1/cyclinB by Flashplate assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50191931(2-(4-(1H-pyrrolo[2,3-b]pyridin-3-yl)pyrimidin-2-yl...)
Affinity DataIC50: 139nMAssay Description:Inhibition of CDK1/cyclinB by Flashplate assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50120510(4-{[2-(1-Hydroxymethyl-2-methyl-propylamino)-9-iso...)
Affinity DataIC50: 150nMAssay Description:Inhibition of recombinant Cyclin-dependent kinase 1-cyclin BMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM7377(CHEMBL75680 | aloisine A | 7-n-Butyl-6-(4-hydroxyp...)
Affinity DataIC50: 150nMAssay Description:Inhibition of CDK1/cyclinBMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50191930(N-(cyclohexylmethyl)-4-(1H-pyrrolo[2,3-b]pyridin-3...)
Affinity DataIC50: 151nMAssay Description:Inhibition of CDK1/cyclinB by Flashplate assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50147458((3-{3-[4-(2-Methoxy-phenyl)-2,5-dioxo-2,5-dihydro-...)
Affinity DataIC50: 170nMAssay Description:Inhibition of Cyclin-dependent kinase 1-cyclin BMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50113281(AT-7519 | US20240293557, Compound AMC-3-098)
Affinity DataIC50: 200nMAssay Description:Inhibition of CDK1/cyclin B (unknown origin) by radiometric filter binding assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM5655(2-(2-chlorophenyl)-5,7-dihydroxy-8-[(3S,4R)-3-hydr...)
Affinity DataIC50: 200nMAssay Description:Inhibition of Cyclin-dependent kinase 1-cyclin B from M phase starfish (Marthasterias glacialis) oocytesMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50120512(3-{[2-(1-Hydroxymethyl-propylamino)-9-isopropyl-9H...)
Affinity DataIC50: 200nMAssay Description:Inhibition of recombinant Cyclin-dependent kinase 1-cyclin BMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM7273(CHEMBL319373 | 14-bromo-4,5-dimethoxy-8,18-diazate...)
Affinity DataIC50: 200nMAssay Description:Inhibition of CDK1/cyclin B expressed in M phase starfish oocyteMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50132310(20-ethyl-17,23-dioxa-4,14,20,26-tetraazahexacyclo[...)
Affinity DataIC50: 240nMAssay Description:Inhibition of CDK1/cyclinBMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
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