Compile Data Set for Download or QSAR
Report error Found 1849 Enz. Inhib. hit(s) with BLAST sequence identity > 85%
TargetCyclin-dependent kinase 5 activator 1 Cyclin-dependent kinase 5 activator 1(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50400564(CHEMBL2206242)
Affinity DataEC50:  3.03E+3nMAssay Description:Inhibition of human Cdk5/p35 activityMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCyclin-dependent kinase 5 activator 1 Cyclin-dependent kinase 5 activator 1(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50505541(CHEMBL4465866)
Affinity DataKd:  87nMAssay Description:Binding affinity to recombinant human full-length N-terminal GST-tagged CDK5 (1 to 292 residues)/N-terminal His6-tagged p25 (99 to 307 residues) expr...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetCyclin-dependent kinase 5 activator 1 Cyclin-dependent kinase 5 activator 1(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM6878(5-amino-N-(2,6-difluorophenyl)-3-[(4-sulfamoylphen...)
Affinity DataIC50: 0.200nMAssay Description:Inhibition of GST-tagged CDK5/p25 (unknown origin) expressed in Baculovirus infected Sf9 cells using histone H1 as substrate as substrate in presence...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCyclin-dependent kinase 5 activator 1 Cyclin-dependent kinase 5 activator 1(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50585763(CHEMBL5075328)
Affinity DataIC50: 0.200nMAssay Description:Inhibition of full length N-terminal GST fused human CDK5(1 to 292 residues)/ p25 (99 to 307 residues) expressed in baculovirus expression system usi...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCyclin-dependent kinase 5 activator 1 Cyclin-dependent kinase 5 activator 1(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50585766(CHEMBL5080866)
Affinity DataIC50: 0.200nMAssay Description:Inhibition of Nano-Luc fused human full length CDK5/P35 transfected in HEK293 cells incubated for 1 hr by NanoBRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetCyclin-dependent kinase 5 activator 1 Cyclin-dependent kinase 5 activator 1(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50585759(CHEMBL5081712)
Affinity DataIC50: 0.600nMAssay Description:Inhibition of full length N-terminal GST fused human CDK5(1 to 292 residues)/ p25 (99 to 307 residues) expressed in baculovirus expression system usi...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCyclin-dependent kinase 5 activator 1 Cyclin-dependent kinase 5 activator 1(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50585762(CHEMBL5077138)
Affinity DataIC50: 0.600nMAssay Description:Inhibition of full length N-terminal GST fused human CDK5(1 to 292 residues)/ p25 (99 to 307 residues) expressed in baculovirus expression system usi...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetCyclin-dependent kinase 5 activator 1 Cyclin-dependent kinase 5 activator 1(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50585768(CHEMBL5074832)
Affinity DataIC50: 0.600nMAssay Description:Inhibition of full length N-terminal GST fused human CDK5(1 to 292 residues)/ p25 (99 to 307 residues) expressed in baculovirus expression system usi...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetCyclin-dependent kinase 5 activator 1 Cyclin-dependent kinase 5 activator 1(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50585770(CHEMBL5080351)
Affinity DataIC50: 0.600nMAssay Description:Inhibition of full length N-terminal GST fused human CDK5(1 to 292 residues)/ p25 (99 to 307 residues) expressed in baculovirus expression system usi...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetCyclin-dependent kinase 5 activator 1 Cyclin-dependent kinase 5 activator 1(Human)
G1 Therapeutics

US Patent
LigandPNGBDBM601933(US11643416, Compound 1 | 4-((6'-hydroxy-8'-oxo-7',...)
Affinity DataIC50: 0.680nMAssay Description:Selected compounds disclosed herein were tested in kinase assays by Nanosyn (Santa Clara, Calif.) to determine their inhibitory effect on these CDKs....More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
US Patent

TargetCyclin-dependent kinase 5 activator 1 Cyclin-dependent kinase 5 activator 1(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM601933(US11643416, Compound 1 | 4-((6'-hydroxy-8'-oxo-7',...)
Affinity DataIC50: 0.680nMAssay Description:Selected compounds disclosed herein were tested in kinase assays by Nanosyn (Santa Clara, CA) to determine their inhibitory effect on these CDKs. The...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
US Patent

TargetCyclin-dependent kinase 5 activator 1 Cyclin-dependent kinase 5 activator 1(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50585761(CHEMBL5078762)
Affinity DataIC50: 0.800nMAssay Description:Inhibition of full length N-terminal GST fused human CDK5(1 to 292 residues)/ p25 (99 to 307 residues) expressed in baculovirus expression system usi...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetCyclin-dependent kinase 5 activator 1 Cyclin-dependent kinase 5 activator 1(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50585774(CHEMBL5086375)
Affinity DataIC50: 0.800nMAssay Description:Inhibition of full length N-terminal GST fused human CDK5(1 to 292 residues)/ p25 (99 to 307 residues) expressed in baculovirus expression system usi...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetCyclin-dependent kinase 5 activator 1 Cyclin-dependent kinase 5 activator 1(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50585780(CHEMBL5090019)
Affinity DataIC50: 0.800nMAssay Description:Inhibition of full length N-terminal GST fused human CDK5(1 to 292 residues)/ p25 (99 to 307 residues) expressed in baculovirus expression system usi...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetCyclin-dependent kinase 5 activator 1 Cyclin-dependent kinase 5 activator 1(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50585785(CHEMBL5077028)
Affinity DataIC50: 0.800nMAssay Description:Inhibition of full length N-terminal GST fused human CDK5(1 to 292 residues)/ p25 (99 to 307 residues) expressed in baculovirus expression system usi...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetCyclin-dependent kinase 5 activator 1 Cyclin-dependent kinase 5 activator 1(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM601933(US11643416, Compound 1 | 4-((6'-hydroxy-8'-oxo-7',...)
Affinity DataIC50: 0.800nMAssay Description:Selected compounds disclosed herein were tested in kinase assays by Nanosyn (Santa Clara, CA) to determine their inhibitory effect on these CDKs. The...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
US Patent

TargetCyclin-dependent kinase 5 activator 1 Cyclin-dependent kinase 5 activator 1(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50585775(CHEMBL5091792)
Affinity DataIC50: 0.900nMAssay Description:Inhibition of full length N-terminal GST fused human CDK5(1 to 292 residues)/ p25 (99 to 307 residues) expressed in baculovirus expression system usi...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetCyclin-dependent kinase 5 activator 1 Cyclin-dependent kinase 5 activator 1(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50585779(CHEMBL5088595)
Affinity DataIC50: 0.900nMAssay Description:Inhibition of full length N-terminal GST fused human CDK5(1 to 292 residues)/ p25 (99 to 307 residues) expressed in baculovirus expression system usi...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetCyclin-dependent kinase 5 activator 1 Cyclin-dependent kinase 5 activator 1(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50139171(Dinaciclib | MK-7965 | SCH-727965 | US11643396, Ex...)
Affinity DataIC50: 1nMAssay Description:Inhibition of recombinant CDK5/p25 (unknown origin) expressed in baculovirus infected Sf9 insect cells using biotinylated histone H1 as substrate aft...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCyclin-dependent kinase 5 activator 1 Cyclin-dependent kinase 5 activator 1(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50139171(Dinaciclib | MK-7965 | SCH-727965 | US11643396, Ex...)
Affinity DataIC50: 1nMAssay Description:Inhibition of CDK5/p35 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetCyclin-dependent kinase 5 activator 1 Cyclin-dependent kinase 5 activator 1(Human)
G1 Therapeutics

US Patent
LigandPNGBDBM601953(US11643416, Compound 55 | 2'-((4-(piperazine-1- ca...)
Affinity DataIC50: 1nMAssay Description:Selected compounds disclosed herein were tested in kinase assays by Nanosyn (Santa Clara, Calif.) to determine their inhibitory effect on these CDKs....More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
US Patent

TargetCyclin-dependent kinase 5 activator 1 Cyclin-dependent kinase 5 activator 1(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50585756(CHEMBL5092400)
Affinity DataIC50: 1nMAssay Description:Inhibition of full length N-terminal GST fused human CDK5(1 to 292 residues)/ p25 (99 to 307 residues) expressed in baculovirus expression system usi...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetCyclin-dependent kinase 5 activator 1 Cyclin-dependent kinase 5 activator 1(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50585782(CHEMBL5080361)
Affinity DataIC50: 1nMAssay Description:Inhibition of full length N-terminal GST fused human CDK5(1 to 292 residues)/ p25 (99 to 307 residues) expressed in baculovirus expression system usi...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetCyclin-dependent kinase 5 activator 1 Cyclin-dependent kinase 5 activator 1(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50585772(CHEMBL5080566)
Affinity DataIC50: 1nMAssay Description:Inhibition of Nano-Luc fused human full length CDK5/P35 transfected in HEK293 cells incubated for 1 hr by NanoBRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
In DepthDetails Article
PubMedPDB3D3D Structure (crystal)
TargetCyclin-dependent kinase 5 activator 1 Cyclin-dependent kinase 5 activator 1(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM601953(US11643416, Compound 55 | 2'-((4-(piperazine-1- ca...)
Affinity DataIC50: 1nMAssay Description:Selected compounds disclosed herein were tested in kinase assays by Nanosyn (Santa Clara, CA) to determine their inhibitory effect on these CDKs. The...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
US Patent

TargetCyclin-dependent kinase 5 activator 1 Cyclin-dependent kinase 5 activator 1(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50585760(CHEMBL5077125)
Affinity DataIC50: 1.10nMAssay Description:Inhibition of full length N-terminal GST fused human CDK5(1 to 292 residues)/ p25 (99 to 307 residues) expressed in baculovirus expression system usi...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetCyclin-dependent kinase 5 activator 1 Cyclin-dependent kinase 5 activator 1(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50059889(3-methoxy-2-methyl-4-methylamino-(2S,3S,4S,6R)-29-...)
Affinity DataIC50: 1.20nMAssay Description:Inhibition of CDK5/P25 (unknown origin)-mediated phosphorylation of peptide substrate incubated for 15 mins prior to substrate addition measured afte...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCyclin-dependent kinase 5 activator 1 Cyclin-dependent kinase 5 activator 1(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50585769(CHEMBL5094270)
Affinity DataIC50: 1.20nMAssay Description:Inhibition of full length N-terminal GST fused human CDK5(1 to 292 residues)/ p25 (99 to 307 residues) expressed in baculovirus expression system usi...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetCyclin-dependent kinase 5 activator 1 Cyclin-dependent kinase 5 activator 1(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50585777(CHEMBL5083778)
Affinity DataIC50: 1.20nMAssay Description:Inhibition of full length N-terminal GST fused human CDK5(1 to 292 residues)/ p25 (99 to 307 residues) expressed in baculovirus expression system usi...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetCyclin-dependent kinase 5 activator 1 Cyclin-dependent kinase 5 activator 1(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50585764(CHEMBL5088315)
Affinity DataIC50: 1.20nMAssay Description:Inhibition of Nano-Luc fused human full length CDK5/P35 transfected in HEK293 cells incubated for 1 hr by NanoBRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetCyclin-dependent kinase 5 activator 1 Cyclin-dependent kinase 5 activator 1(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50585771(CHEMBL5078192)
Affinity DataIC50: 1.20nMAssay Description:Inhibition of Nano-Luc fused human full length CDK5/P35 transfected in HEK293 cells incubated for 1 hr by NanoBRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetCyclin-dependent kinase 5 activator 1 Cyclin-dependent kinase 5 activator 1(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM2579(CHEMBL388978 | Staurosporine, 8 | Staurosporin, 4 ...)
Affinity DataIC50: 1.30nMAssay Description:Inhibition of human CDK5/p35 using histone H1 as substrate by [gamma-33P]-ATP assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCyclin-dependent kinase 5 activator 1 Cyclin-dependent kinase 5 activator 1(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM601934(US11643416, Compound 2 | 4-((7'-oxo-7',8'-dihydro-...)
Affinity DataIC50: 1.30nMAssay Description:Selected compounds disclosed herein were tested in kinase assays by Nanosyn (Santa Clara, CA) to determine their inhibitory effect on these CDKs. The...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
US Patent

TargetCyclin-dependent kinase 5 activator 1 Cyclin-dependent kinase 5 activator 1(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50414916(CHEMBL567005)
Affinity DataIC50: 1.40nMAssay Description:Inhibition of human CDK5/p25 assessed as histone h1 phosphorylation in presence of ATPMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCyclin-dependent kinase 5 activator 1 Cyclin-dependent kinase 5 activator 1(Human)
G1 Therapeutics

US Patent
LigandPNGBDBM601934(US11643416, Compound 2 | 4-((7'-oxo-7',8'-dihydro-...)
Affinity DataIC50: 1.40nMAssay Description:Selected compounds disclosed herein were tested in kinase assays by Nanosyn (Santa Clara, Calif.) to determine their inhibitory effect on these CDKs....More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
US Patent

TargetCyclin-dependent kinase 5 activator 1 Cyclin-dependent kinase 5 activator 1(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50585765(CHEMBL5078596)
Affinity DataIC50: 1.40nMAssay Description:Inhibition of full length N-terminal GST fused human CDK5(1 to 292 residues)/ p25 (99 to 307 residues) expressed in baculovirus expression system usi...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetCyclin-dependent kinase 5 activator 1 Cyclin-dependent kinase 5 activator 1(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM601934(US11643416, Compound 2 | 4-((7'-oxo-7',8'-dihydro-...)
Affinity DataIC50: 1.40nMAssay Description:Selected compounds disclosed herein were tested in kinase assays by Nanosyn (Santa Clara, CA) to determine their inhibitory effect on these CDKs. The...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
US Patent

TargetCyclin-dependent kinase 5 activator 1 Cyclin-dependent kinase 5 activator 1(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50433369(CHEMBL2377825)
Affinity DataIC50: 1.5nMAssay Description:Inhibition of CDK5/P25 (unknown origin)-mediated phosphorylation of peptide substrate incubated for 15 mins prior to substrate addition measured afte...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCyclin-dependent kinase 5 activator 1 Cyclin-dependent kinase 5 activator 1(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50139171(Dinaciclib | MK-7965 | SCH-727965 | US11643396, Ex...)
Affinity DataIC50: 1.60nMAssay Description:Inhibition of full length N-terminal GST fused human CDK5(1 to 292 residues)/ p25 (99 to 307 residues) expressed in baculovirus expression system usi...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCyclin-dependent kinase 5 activator 1 Cyclin-dependent kinase 5 activator 1(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50585766(CHEMBL5080866)
Affinity DataIC50: 1.80nMAssay Description:Inhibition of full length N-terminal GST fused human CDK5(1 to 292 residues)/ p25 (99 to 307 residues) expressed in baculovirus expression system usi...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetCyclin-dependent kinase 5 activator 1 Cyclin-dependent kinase 5 activator 1(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM2579(CHEMBL388978 | Staurosporine, 8 | Staurosporin, 4 ...)
Affinity DataIC50: 1.90nMAssay Description:Inhibition of human CDK5/p35 using histone H1 as substrate by [gamma-33P]-ATP assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCyclin-dependent kinase 5 activator 1 Cyclin-dependent kinase 5 activator 1(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50193093(RGB-286638)
Affinity DataIC50: 2nMAssay Description:Inhibition of CDK5/p35 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCyclin-dependent kinase 5 activator 1 Cyclin-dependent kinase 5 activator 1(Human)
G1 Therapeutics

US Patent
LigandPNGBDBM601942(US11643416, Compound 42 | 4-((8'-methyl-7'-oxo-7',...)
Affinity DataIC50: 2nMAssay Description:Selected compounds disclosed herein were tested in kinase assays by Nanosyn (Santa Clara, Calif.) to determine their inhibitory effect on these CDKs....More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
US Patent

TargetCyclin-dependent kinase 5 activator 1 Cyclin-dependent kinase 5 activator 1(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50585772(CHEMBL5080566)
Affinity DataIC50: 2nMAssay Description:Inhibition of full length N-terminal GST fused human CDK5(1 to 292 residues)/ p25 (99 to 307 residues) expressed in baculovirus expression system usi...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
In DepthDetails Article
PubMedPDB3D3D Structure (crystal)
TargetCyclin-dependent kinase 5 activator 1 Cyclin-dependent kinase 5 activator 1(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM601942(US11643416, Compound 42 | 4-((8'-methyl-7'-oxo-7',...)
Affinity DataIC50: 2nMAssay Description:Selected compounds disclosed herein were tested in kinase assays by Nanosyn (Santa Clara, CA) to determine their inhibitory effect on these CDKs. The...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
US Patent

TargetCyclin-dependent kinase 5 activator 1 Cyclin-dependent kinase 5 activator 1(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM2579(CHEMBL388978 | Staurosporine, 8 | Staurosporin, 4 ...)
Affinity DataIC50: 2.10nMAssay Description:Inhibition of human CDK5/p25 using histone H1 as substrate by [gamma-33P]-ATP assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCyclin-dependent kinase 5 activator 1 Cyclin-dependent kinase 5 activator 1(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50585783(CHEMBL5070707)
Affinity DataIC50: 2.20nMAssay Description:Inhibition of full length N-terminal GST fused human CDK5(1 to 292 residues)/ p25 (99 to 307 residues) expressed in baculovirus expression system usi...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetCyclin-dependent kinase 5 activator 1 Cyclin-dependent kinase 5 activator 1(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50585784(CHEMBL5087911)
Affinity DataIC50: 2.20nMAssay Description:Inhibition of full length N-terminal GST fused human CDK5(1 to 292 residues)/ p25 (99 to 307 residues) expressed in baculovirus expression system usi...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetCyclin-dependent kinase 5 activator 1 Cyclin-dependent kinase 5 activator 1(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50261164(CHEMBL4103221)
Affinity DataIC50: 2.30nMAssay Description:Inhibition of CDK5/p35 (unknown origin) using ULingt-4E-BP as substrate after 1 hr in presence of ATP by fluorescence assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetCyclin-dependent kinase 5 activator 1 Cyclin-dependent kinase 5 activator 1(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50585781(CHEMBL5084200)
Affinity DataIC50: 2.30nMAssay Description:Inhibition of full length N-terminal GST fused human CDK5(1 to 292 residues)/ p25 (99 to 307 residues) expressed in baculovirus expression system usi...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
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