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TargetProtein kinase C theta type(Human)
Exscientia AI

US Patent
LigandPNGBDBM685558(US20240239794, Example 95)
Affinity DataIC50: 0.126nMAssay Description:PKC-theta and PKC-delta biochemical activities were measured using the PKC-theta HTRF KinEASEkit kit, according to manufacturer's instructions (C...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/30/2024
Entry Details
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TargetProtein kinase C theta type(Human)
Exscientia AI

US Patent
LigandPNGBDBM685502(US20240239794, Example 39)
Affinity DataIC50: 0.200nMAssay Description:PKC-theta and PKC-delta biochemical activities were measured using the PKC-theta HTRF KinEASEkit kit, according to manufacturer's instructions (C...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/30/2024
Entry Details
Go to US Patent

TargetProtein kinase C theta type(Human)
Exscientia AI

US Patent
LigandPNGBDBM685503(US20240239794, Example 40)
Affinity DataIC50: 0.200nMAssay Description:PKC-theta and PKC-delta biochemical activities were measured using the PKC-theta HTRF KinEASEkit kit, according to manufacturer's instructions (C...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/30/2024
Entry Details
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TargetCoagulation factor X(Human)
Sanofi-Aventis R&D

Curated by ChEMBL
LigandPNGBDBM50443857(CHEMBL3091501)
Affinity DataIC50: 0.200nMAssay Description:Inhibition of human coagulation factor 10a using S-2765 as substrate measured up to 20 mins by chromogenic assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/25/2014
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetProtein kinase C theta type(Human)
Exscientia AI

US Patent
LigandPNGBDBM685531(US20240239794, Example 68)
Affinity DataIC50: 0.251nMAssay Description:PKC-theta and PKC-delta biochemical activities were measured using the PKC-theta HTRF KinEASEkit kit, according to manufacturer's instructions (C...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/30/2024
Entry Details
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TargetProtein kinase C theta type(Human)
Exscientia AI

US Patent
LigandPNGBDBM685525(US20240239794, Example 62)
Affinity DataIC50: 0.316nMAssay Description:PKC-theta and PKC-delta biochemical activities were measured using the PKC-theta HTRF KinEASEkit kit, according to manufacturer's instructions (C...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/30/2024
Entry Details
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TargetProtein kinase C theta type(Human)
Exscientia AI

US Patent
LigandPNGBDBM685492(US20240239794, Example 29)
Affinity DataIC50: 0.398nMAssay Description:PKC-theta and PKC-delta biochemical activities were measured using the PKC-theta HTRF KinEASEkit kit, according to manufacturer's instructions (C...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/30/2024
Entry Details
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TargetProtein kinase C theta type(Human)
Exscientia AI

US Patent
LigandPNGBDBM685504(US20240239794, Example 41)
Affinity DataIC50: 0.398nMAssay Description:PKC-theta and PKC-delta biochemical activities were measured using the PKC-theta HTRF KinEASEkit kit, according to manufacturer's instructions (C...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/30/2024
Entry Details
Go to US Patent

TargetCoagulation factor X(Human)
Sanofi-Aventis R&D

Curated by ChEMBL
LigandPNGBDBM50443858(CHEMBL3091502)
Affinity DataIC50: 0.5nMAssay Description:Inhibition of human coagulation factor 10a using S-2765 as substrate measured up to 20 mins by chromogenic assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/25/2014
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetCoagulation factor X(Human)
Sanofi-Aventis R&D

Curated by ChEMBL
LigandPNGBDBM50443846(CHEMBL3091527)
Affinity DataIC50: 0.5nMAssay Description:Inhibition of human coagulation factor 10a using S-2765 as substrate measured up to 20 mins by chromogenic assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/25/2014
Entry Details Article
PubMed
TargetProtein kinase C theta type(Human)
Exscientia AI

US Patent
LigandPNGBDBM685486(US20240239794, Example 23)
Affinity DataIC50: 0.501nMAssay Description:PKC-theta and PKC-delta biochemical activities were measured using the PKC-theta HTRF KinEASEkit kit, according to manufacturer's instructions (C...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/30/2024
Entry Details
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TargetProtein kinase C theta type(Human)
Exscientia AI

US Patent
LigandPNGBDBM685521(US20240239794, Example 58)
Affinity DataIC50: 0.501nMAssay Description:PKC-theta and PKC-delta biochemical activities were measured using the PKC-theta HTRF KinEASEkit kit, according to manufacturer's instructions (C...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/30/2024
Entry Details
Go to US Patent

TargetProtein kinase C theta type(Human)
Exscientia AI

US Patent
LigandPNGBDBM685488(US20240239794, Example 25)
Affinity DataIC50: 0.501nMAssay Description:PKC-theta and PKC-delta biochemical activities were measured using the PKC-theta HTRF KinEASEkit kit, according to manufacturer's instructions (C...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/30/2024
Entry Details
Go to US Patent

TargetProtein kinase C theta type(Human)
Exscientia AI

US Patent
LigandPNGBDBM685514(US20240239794, Example 51)
Affinity DataIC50: 0.501nMAssay Description:PKC-theta and PKC-delta biochemical activities were measured using the PKC-theta HTRF KinEASEkit kit, according to manufacturer's instructions (C...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/30/2024
Entry Details
Go to US Patent

TargetCoagulation factor X(Human)
Sanofi-Aventis R&D

Curated by ChEMBL
LigandPNGBDBM50443847(CHEMBL3091526)
Affinity DataIC50: 0.600nMAssay Description:Inhibition of human coagulation factor 10a using S-2765 as substrate measured up to 20 mins by chromogenic assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/25/2014
Entry Details Article
PubMed
TargetProtein kinase C theta type(Human)
Exscientia AI

US Patent
LigandPNGBDBM685510(US20240239794, Example 47)
Affinity DataIC50: 0.631nMAssay Description:PKC-theta and PKC-delta biochemical activities were measured using the PKC-theta HTRF KinEASEkit kit, according to manufacturer's instructions (C...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/30/2024
Entry Details
Go to US Patent

TargetProtein kinase C theta type(Human)
Exscientia AI

US Patent
LigandPNGBDBM685522(US20240239794, Example 59)
Affinity DataIC50: 0.631nMAssay Description:PKC-theta and PKC-delta biochemical activities were measured using the PKC-theta HTRF KinEASEkit kit, according to manufacturer's instructions (C...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/30/2024
Entry Details
Go to US Patent

TargetProtein kinase C theta type(Human)
Exscientia AI

US Patent
LigandPNGBDBM685543(US20240239794, Example 80)
Affinity DataIC50: 0.794nMAssay Description:PKC-theta and PKC-delta biochemical activities were measured using the PKC-theta HTRF KinEASEkit kit, according to manufacturer's instructions (C...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/30/2024
Entry Details
Go to US Patent

TargetProtein kinase C theta type(Human)
Exscientia AI

US Patent
LigandPNGBDBM685545(US20240239794, Example 82)
Affinity DataIC50: 0.794nMAssay Description:PKC-theta and PKC-delta biochemical activities were measured using the PKC-theta HTRF KinEASEkit kit, according to manufacturer's instructions (C...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/30/2024
Entry Details
Go to US Patent

TargetProtein kinase C theta type(Human)
Exscientia AI

US Patent
LigandPNGBDBM685569(US20240239794, Example 106)
Affinity DataIC50: 0.794nMAssay Description:PKC-theta and PKC-delta biochemical activities were measured using the PKC-theta HTRF KinEASEkit kit, according to manufacturer's instructions (C...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/30/2024
Entry Details
Go to US Patent

TargetProtein kinase C theta type(Human)
Exscientia AI

US Patent
LigandPNGBDBM685513(US20240239794, Example 50)
Affinity DataIC50: 0.794nMAssay Description:PKC-theta and PKC-delta biochemical activities were measured using the PKC-theta HTRF KinEASEkit kit, according to manufacturer's instructions (C...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/30/2024
Entry Details
Go to US Patent

TargetProtein kinase C theta type(Human)
Exscientia AI

US Patent
LigandPNGBDBM685567(US20240239794, Example 104)
Affinity DataIC50: 0.794nMAssay Description:PKC-theta and PKC-delta biochemical activities were measured using the PKC-theta HTRF KinEASEkit kit, according to manufacturer's instructions (C...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/30/2024
Entry Details
Go to US Patent

TargetP2Y purinoceptor 12(Human)
Sanofi R & D

Curated by ChEMBL
LigandPNGBDBM50100263(CHEMBL3326907)
Affinity DataIC50: 0.900nMAssay Description:Displacement of [33P]2MeS-ADP from P2Y12 receptor (unknown origin) transfected in CHO cells after 30 mins by scintillation counting analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/30/2016
Entry Details Article
PubMed
TargetProtein kinase C theta type(Human)
Exscientia AI

US Patent
LigandPNGBDBM685541(US20240239794, Example 78)
Affinity DataIC50: 1nMAssay Description:PKC-theta and PKC-delta biochemical activities were measured using the PKC-theta HTRF KinEASEkit kit, according to manufacturer's instructions (C...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/30/2024
Entry Details
Go to US Patent

TargetProtein kinase C theta type(Human)
Exscientia AI

US Patent
LigandPNGBDBM685550(US20240239794, Example 87)
Affinity DataIC50: 1nMAssay Description:PKC-theta and PKC-delta biochemical activities were measured using the PKC-theta HTRF KinEASEkit kit, according to manufacturer's instructions (C...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/30/2024
Entry Details
Go to US Patent

TargetCoagulation factor X(Human)
Sanofi-Aventis R&D

Curated by ChEMBL
LigandPNGBDBM50443861(CHEMBL3091515)
Affinity DataIC50: 1nMAssay Description:Inhibition of human coagulation factor 10a using S-2765 as substrate measured up to 20 mins by chromogenic assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/25/2014
Entry Details Article
PubMed
TargetCoagulation factor X(Human)
Sanofi-Aventis R&D

Curated by ChEMBL
LigandPNGBDBM50443844(CHEMBL3091506)
Affinity DataIC50: 1nMAssay Description:Inhibition of human coagulation factor 10a using S-2765 as substrate measured up to 20 mins by chromogenic assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/25/2014
Entry Details Article
PubMed
TargetCoagulation factor X(Human)
Sanofi-Aventis R&D

Curated by ChEMBL
LigandPNGBDBM50443853(CHEMBL3091519 | US20230391761, Reference 1)
Affinity DataIC50: 1nMAssay Description:Inhibition of human coagulation factor 10a using S-2765 as substrate measured up to 20 mins by chromogenic assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/25/2014
Entry Details Article
PubMed
TargetProtein kinase C theta type(Human)
Exscientia AI

US Patent
LigandPNGBDBM685540(US20240239794, Example 77 | One More Step Will be ...)
Affinity DataIC50: 1nMAssay Description:PKC-theta and PKC-delta biochemical activities were measured using the PKC-theta HTRF KinEASEkit kit, according to manufacturer's instructions (C...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/30/2024
Entry Details
Go to US Patent

TargetProtein kinase C theta type(Human)
Exscientia AI

US Patent
LigandPNGBDBM685553(US20240239794, Example 90)
Affinity DataIC50: 1nMAssay Description:PKC-theta and PKC-delta biochemical activities were measured using the PKC-theta HTRF KinEASEkit kit, according to manufacturer's instructions (C...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/30/2024
Entry Details
Go to US Patent

TargetCoagulation factor X(Human)
Sanofi-Aventis R&D

Curated by ChEMBL
LigandPNGBDBM50443848(CHEMBL3091525)
Affinity DataIC50: 1.10nMAssay Description:Inhibition of human coagulation factor 10a using S-2765 as substrate measured up to 20 mins by chromogenic assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/25/2014
Entry Details Article
PubMed
TargetCoagulation factor X(Human)
Sanofi-Aventis R&D

Curated by ChEMBL
LigandPNGBDBM50443862(CHEMBL3091514)
Affinity DataIC50: 1.10nMAssay Description:Inhibition of human coagulation factor 10a using S-2765 as substrate measured up to 20 mins by chromogenic assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/25/2014
Entry Details Article
PubMed
TargetCoagulation factor X(Human)
Sanofi-Aventis R&D

Curated by ChEMBL
LigandPNGBDBM50443869(CHEMBL3091507)
Affinity DataIC50: 1.10nMAssay Description:Inhibition of human coagulation factor 10a using S-2765 as substrate measured up to 20 mins by chromogenic assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/25/2014
Entry Details Article
PubMed
TargetCoagulation factor X(Human)
Sanofi-Aventis R&D

Curated by ChEMBL
LigandPNGBDBM50443867(CHEMBL3091509)
Affinity DataIC50: 1.20nMAssay Description:Inhibition of human coagulation factor 10a using S-2765 as substrate measured up to 20 mins by chromogenic assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/25/2014
Entry Details Article
PubMed
TargetProtein kinase C theta type(Human)
Exscientia AI

US Patent
LigandPNGBDBM685494(US20240239794, Example 31)
Affinity DataIC50: 1.26nMAssay Description:PKC-theta and PKC-delta biochemical activities were measured using the PKC-theta HTRF KinEASEkit kit, according to manufacturer's instructions (C...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/30/2024
Entry Details
Go to US Patent

TargetProtein kinase C theta type(Human)
Exscientia AI

US Patent
LigandPNGBDBM685520(US20240239794, Example 57)
Affinity DataIC50: 1.26nMAssay Description:PKC-theta and PKC-delta biochemical activities were measured using the PKC-theta HTRF KinEASEkit kit, according to manufacturer's instructions (C...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/30/2024
Entry Details
Go to US Patent

TargetProtein kinase C theta type(Human)
Exscientia AI

US Patent
LigandPNGBDBM685493(US20240239794, Example 30)
Affinity DataIC50: 1.26nMAssay Description:PKC-theta and PKC-delta biochemical activities were measured using the PKC-theta HTRF KinEASEkit kit, according to manufacturer's instructions (C...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/30/2024
Entry Details
Go to US Patent

TargetProtein kinase C theta type(Human)
Exscientia AI

US Patent
LigandPNGBDBM685501(US20240239794, Example 38)
Affinity DataIC50: 1.26nMAssay Description:PKC-theta and PKC-delta biochemical activities were measured using the PKC-theta HTRF KinEASEkit kit, according to manufacturer's instructions (C...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/30/2024
Entry Details
Go to US Patent

TargetProtein kinase C theta type(Human)
Exscientia AI

US Patent
LigandPNGBDBM685542(US20240239794, Example 79)
Affinity DataIC50: 1.26nMAssay Description:PKC-theta and PKC-delta biochemical activities were measured using the PKC-theta HTRF KinEASEkit kit, according to manufacturer's instructions (C...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/30/2024
Entry Details
Go to US Patent

TargetCoagulation factor X(Human)
Sanofi-Aventis R&D

Curated by ChEMBL
LigandPNGBDBM50443864(CHEMBL3091512)
Affinity DataIC50: 1.40nMAssay Description:Inhibition of human coagulation factor 10a using S-2765 as substrate measured up to 20 mins by chromogenic assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/25/2014
Entry Details Article
PubMed
TargetCoagulation factor X(Human)
Sanofi-Aventis R&D

Curated by ChEMBL
LigandPNGBDBM50443865(CHEMBL3091511)
Affinity DataIC50: 1.40nMAssay Description:Inhibition of human coagulation factor 10a using S-2765 as substrate measured up to 20 mins by chromogenic assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/25/2014
Entry Details Article
PubMed
TargetProtein kinase C theta type(Human)
Exscientia AI

US Patent
LigandPNGBDBM685497(US20240239794, Example 34)
Affinity DataIC50: 1.58nMAssay Description:PKC-theta and PKC-delta biochemical activities were measured using the PKC-theta HTRF KinEASEkit kit, according to manufacturer's instructions (C...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/30/2024
Entry Details
Go to US Patent

TargetProtein kinase C theta type(Human)
Exscientia AI

US Patent
LigandPNGBDBM685546(US20240239794, Example 83)
Affinity DataIC50: 1.58nMAssay Description:PKC-theta and PKC-delta biochemical activities were measured using the PKC-theta HTRF KinEASEkit kit, according to manufacturer's instructions (C...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/30/2024
Entry Details
Go to US Patent

TargetCoagulation factor X(Human)
Sanofi-Aventis R&D

Curated by ChEMBL
LigandPNGBDBM50443856(CHEMBL3091503)
Affinity DataIC50: 1.80nMAssay Description:Inhibition of human coagulation factor 10a using S-2765 as substrate measured up to 20 mins by chromogenic assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/25/2014
Entry Details Article
PubMed
TargetCoagulation factor X(Human)
Sanofi-Aventis R&D

Curated by ChEMBL
LigandPNGBDBM50443845(CHEMBL3091528)
Affinity DataIC50: 1.80nMAssay Description:Inhibition of human coagulation factor 10a using S-2765 as substrate measured up to 20 mins by chromogenic assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/25/2014
Entry Details Article
PubMed
TargetCoagulation factor X(Human)
Sanofi-Aventis R&D

Curated by ChEMBL
LigandPNGBDBM50443866(CHEMBL3091510)
Affinity DataIC50: 1.90nMAssay Description:Inhibition of human coagulation factor 10a using S-2765 as substrate measured up to 20 mins by chromogenic assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/25/2014
Entry Details Article
PubMed
TargetProtein kinase C theta type(Human)
Exscientia AI

US Patent
LigandPNGBDBM685491(US20240239794, Example 28)
Affinity DataIC50: 2nMAssay Description:PKC-theta and PKC-delta biochemical activities were measured using the PKC-theta HTRF KinEASEkit kit, according to manufacturer's instructions (C...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/30/2024
Entry Details
Go to US Patent

TargetProtein kinase C theta type(Human)
Exscientia AI

US Patent
LigandPNGBDBM685538(US20240239794, Example 75)
Affinity DataIC50: 2nMAssay Description:PKC-theta and PKC-delta biochemical activities were measured using the PKC-theta HTRF KinEASEkit kit, according to manufacturer's instructions (C...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/30/2024
Entry Details
Go to US Patent

TargetProtein kinase C theta type(Human)
Exscientia AI

US Patent
LigandPNGBDBM685519(US20240239794, Example 56)
Affinity DataIC50: 2nMAssay Description:PKC-theta and PKC-delta biochemical activities were measured using the PKC-theta HTRF KinEASEkit kit, according to manufacturer's instructions (C...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/30/2024
Entry Details
Go to US Patent

TargetProtein kinase C theta type(Human)
Exscientia AI

US Patent
LigandPNGBDBM685524(US20240239794, Example 61)
Affinity DataIC50: 2nMAssay Description:PKC-theta and PKC-delta biochemical activities were measured using the PKC-theta HTRF KinEASEkit kit, according to manufacturer's instructions (C...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/30/2024
Entry Details
Go to US Patent

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