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TargetHeme-binding protein A(Haemophilus parasuis)
Ghent University

LigandPNGBDBM225232(S-methylglutathione)
Affinity DataKd:  900nMpH: 7.4 T: 2°CAssay Description:Experiments were carried out using a VP-ITC MicroCalorimeter (MicroCal) at 37°C, and data were analyzed using the Origen ITC analysis software packag...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/9/2017
Entry Details Article
PubMed
TargetNuclear receptor ROR-gamma(Human)
Inventiva

Curated by ChEMBL
LigandPNGBDBM50546040(CHEMBL4792595)
Affinity DataEC50:  880nMAssay Description:Inverse agonist activity at pSG5GAL4-DBD/LBD fused human RORgamma receptor expressed in COS7 cells co-expressing 5 copies of GAL4 response element af...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/21/2022
Entry Details Article
PubMed
TargetNuclear receptor ROR-gamma(Human)
Inventiva

Curated by ChEMBL
LigandPNGBDBM50546015(CHEMBL4745812)
Affinity DataEC50:  1.36E+3nMAssay Description:Inverse agonist activity at pSG5GAL4-DBD/LBD fused human RORgamma receptor expressed in COS7 cells co-expressing 5 copies of GAL4 response element af...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/21/2022
Entry Details Article
PubMed
TargetNuclear receptor ROR-gamma(Human)
Inventiva

Curated by ChEMBL
LigandPNGBDBM50546029(CHEMBL4763665)
Affinity DataEC50:  940nMAssay Description:Inverse agonist activity at pSG5GAL4-DBD/LBD fused human RORgamma receptor expressed in COS7 cells co-expressing 5 copies of GAL4 response element af...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/21/2022
Entry Details Article
PubMed
TargetNuclear receptor ROR-gamma(Human)
Inventiva

Curated by ChEMBL
LigandPNGBDBM50546018(CHEMBL4779817)
Affinity DataEC50:  210nMAssay Description:Inverse agonist activity at RORgamma in human CD4+ T cells assessed as inhibition of IL17A secretion after 72 hrs by ELISAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/21/2022
Entry Details Article
PubMed
TargetHeme-binding protein A(Actinobacillus pleuropneumoniae)
Ghent University

LigandPNGBDBM50422268(GLUTATHIONE | GSH)
Affinity DataKd:  1.58E+3nMpH: 7.4 T: 2°CAssay Description:Experiments were carried out using a VP-ITC MicroCalorimeter (MicroCal) at 37°C, and data were analyzed using the Origen ITC analysis software packag...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/9/2017
Entry Details Article
PubMed
TargetNuclear receptor ROR-gamma(Human)
Inventiva

Curated by ChEMBL
LigandPNGBDBM50546029(CHEMBL4763665)
Affinity DataEC50: >5.00E+3nMAssay Description:Inverse agonist activity at RORgamma in human CD4+ T cells assessed as inhibition of IL17A secretion after 72 hrs by ELISAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/21/2022
Entry Details Article
PubMed
TargetNuclear receptor ROR-gamma(Human)
Inventiva

Curated by ChEMBL
LigandPNGBDBM50546032(CHEMBL4786464)
Affinity DataEC50: >1.00E+4nMAssay Description:Inverse agonist activity at pSG5GAL4-DBD/LBD fused human RORgamma receptor expressed in COS7 cells co-expressing 5 copies of GAL4 response element af...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/21/2022
Entry Details Article
PubMed
TargetHeme-binding protein A(Actinobacillus pleuropneumoniae)
Ghent University

LigandPNGBDBM225232(S-methylglutathione)
Affinity DataKd:  1.17E+3nMpH: 7.4 T: 2°CAssay Description:Experiments were carried out using a VP-ITC MicroCalorimeter (MicroCal) at 37°C, and data were analyzed using the Origen ITC analysis software packag...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/9/2017
Entry Details Article
PubMed
TargetNuclear receptor ROR-gamma(Human)
Inventiva

Curated by ChEMBL
LigandPNGBDBM50546041(CHEMBL4800301)
Affinity DataEC50:  630nMAssay Description:Inverse agonist activity at pSG5GAL4-DBD/LBD fused human RORgamma receptor expressed in COS7 cells co-expressing 5 copies of GAL4 response element af...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/21/2022
Entry Details Article
PubMed
TargetNuclear receptor ROR-gamma(Human)
Inventiva

Curated by ChEMBL
LigandPNGBDBM50546026(CHEMBL4782026)
Affinity DataEC50:  1.66E+3nMAssay Description:Inverse agonist activity at pSG5GAL4-DBD/LBD fused human RORgamma receptor expressed in COS7 cells co-expressing 5 copies of GAL4 response element af...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/21/2022
Entry Details Article
PubMed
TargetNuclear receptor ROR-gamma(Human)
Inventiva

Curated by ChEMBL
LigandPNGBDBM50546021(CHEMBL4759286)
Affinity DataEC50:  960nMAssay Description:Inverse agonist activity at pSG5GAL4-DBD/LBD fused human RORgamma receptor expressed in COS7 cells co-expressing 5 copies of GAL4 response element af...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/21/2022
Entry Details Article
PubMed
TargetNuclear receptor ROR-gamma(Human)
Inventiva

Curated by ChEMBL
LigandPNGBDBM50546037(CHEMBL4786942)
Affinity DataEC50:  220nMAssay Description:Inverse agonist activity at pSG5GAL4-DBD/LBD fused human RORgamma receptor expressed in COS7 cells co-expressing 5 copies of GAL4 response element af...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/21/2022
Entry Details Article
PubMed
LigandPNGBDBM126826(US8785467, 1-29)
Affinity DataEC50:  2.00E+3nMAssay Description:Activation of PXR (unknown origin) assessed as CYP3A4 inductionMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/13/2024
Entry Details
PubMed
TargetNuclear receptor ROR-gamma(Human)
Inventiva

Curated by ChEMBL
LigandPNGBDBM50546034(CHEMBL4747263)
Affinity DataEC50:  910nMAssay Description:Inverse agonist activity at pSG5GAL4-DBD/LBD fused human RORgamma receptor expressed in COS7 cells co-expressing 5 copies of GAL4 response element af...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/21/2022
Entry Details Article
PubMed
TargetNuclear receptor ROR-gamma(Human)
Inventiva

Curated by ChEMBL
LigandPNGBDBM50546024(CHEMBL4739928)
Affinity DataEC50:  1.51E+3nMAssay Description:Inverse agonist activity at pSG5GAL4-DBD/LBD fused human RORgamma receptor expressed in COS7 cells co-expressing 5 copies of GAL4 response element af...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/21/2022
Entry Details Article
PubMed
LigandPNGBDBM163722(US9062059, 1-2)
Affinity DataEC50: >3.00E+4nMAssay Description:Activation of PXR (unknown origin) assessed as CYP3A4 inductionMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/13/2024
Entry Details
PubMed
LigandPNGBDBM50616544(MK-8189 | Mk-8189)
Affinity DataEC50: >3.00E+4nMAssay Description:Activation of PXR (unknown origin) assessed as CYP3A4 inductionMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/13/2024
Entry Details
PubMed
TargetHeme-binding protein A(Actinobacillus pleuropneumoniae)
Ghent University

LigandPNGBDBM225231(OXIGLUTATIONE | Disulfide, Glutathione | Oxidized ...)
Affinity DataKd:  330nMpH: 7.4 T: 2°CAssay Description:Experiments were carried out using a VP-ITC MicroCalorimeter (MicroCal) at 37°C, and data were analyzed using the Origen ITC analysis software packag...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/9/2017
Entry Details Article
PubMed
TargetNuclear receptor ROR-gamma(Human)
Inventiva

Curated by ChEMBL
LigandPNGBDBM50546033(CHEMBL4752056)
Affinity DataEC50:  1.39E+3nMAssay Description:Inverse agonist activity at pSG5GAL4-DBD/LBD fused human RORgamma receptor expressed in COS7 cells co-expressing 5 copies of GAL4 response element af...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/21/2022
Entry Details Article
PubMed
TargetNuclear receptor ROR-gamma(Human)
Inventiva

Curated by ChEMBL
LigandPNGBDBM50546030(CHEMBL4745208)
Affinity DataEC50:  220nMAssay Description:Inverse agonist activity at pSG5GAL4-DBD/LBD fused human RORgamma receptor expressed in COS7 cells co-expressing 5 copies of GAL4 response element af...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/21/2022
Entry Details Article
PubMed
TargetNuclear receptor ROR-gamma(Human)
Inventiva

Curated by ChEMBL
LigandPNGBDBM50546017(CHEMBL4779432)
Affinity DataEC50:  250nMAssay Description:Inverse agonist activity at pSG5GAL4-DBD/LBD fused human RORgamma receptor expressed in COS7 cells co-expressing 5 copies of GAL4 response element af...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/21/2022
Entry Details Article
PubMed
TargetHbpA(Pasteurella multocida)
Ghent University

LigandPNGBDBM50422268(GLUTATHIONE | GSH)
Affinity DataKd:  260nMpH: 7.4 T: 2°CAssay Description:Experiments were carried out using a VP-ITC MicroCalorimeter (MicroCal) at 37°C, and data were analyzed using the Origen ITC analysis software packag...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/9/2017
Entry Details Article
PubMed
TargetNuclear receptor ROR-gamma(Human)
Inventiva

Curated by ChEMBL
LigandPNGBDBM50546023(CHEMBL4749883)
Affinity DataEC50:  810nMAssay Description:Inverse agonist activity at pSG5GAL4-DBD/LBD fused human RORgamma receptor expressed in COS7 cells co-expressing 5 copies of GAL4 response element af...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/21/2022
Entry Details Article
PubMed
TargetNuclear receptor ROR-gamma(Human)
Inventiva

Curated by ChEMBL
LigandPNGBDBM50546038(CHEMBL4788490)
Affinity DataEC50:  760nMAssay Description:Inverse agonist activity at pSG5GAL4-DBD/LBD fused human RORgamma receptor expressed in COS7 cells co-expressing 5 copies of GAL4 response element af...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/21/2022
Entry Details Article
PubMed
TargetNuclear receptor ROR-gamma(Human)
Inventiva

Curated by ChEMBL
LigandPNGBDBM50546027(CHEMBL4779716)
Affinity DataEC50:  100nMAssay Description:Inverse agonist activity at pSG5GAL4-DBD/LBD fused human RORgamma receptor expressed in COS7 cells co-expressing 5 copies of GAL4 response element af...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/21/2022
Entry Details Article
PubMed
TargetNuclear receptor ROR-gamma(Human)
Inventiva

Curated by ChEMBL
LigandPNGBDBM50546016(CHEMBL4787298)
Affinity DataEC50:  170nMAssay Description:Inverse agonist activity at pSG5GAL4-DBD/LBD fused human RORgamma receptor expressed in COS7 cells co-expressing 5 copies of GAL4 response element af...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/21/2022
Entry Details Article
PubMed
TargetNuclear receptor ROR-gamma(Human)
Inventiva

Curated by ChEMBL
LigandPNGBDBM50546018(CHEMBL4779817)
Affinity DataEC50:  350nMAssay Description:Inverse agonist activity at pSG5GAL4-DBD/LBD fused human RORgamma receptor expressed in COS7 cells co-expressing 5 copies of GAL4 response element af...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/21/2022
Entry Details Article
PubMed
TargetNuclear receptor ROR-gamma(Human)
Inventiva

Curated by ChEMBL
LigandPNGBDBM50546024(CHEMBL4739928)
Affinity DataEC50:  1.39E+3nMAssay Description:Inverse agonist activity at RORgamma in human CD4+ T cells assessed as inhibition of IL17A secretion after 72 hrs by ELISAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/21/2022
Entry Details Article
PubMed
TargetNuclear receptor ROR-gamma(Human)
Inventiva

Curated by ChEMBL
LigandPNGBDBM50546019(CHEMBL4752983)
Affinity DataEC50:  770nMAssay Description:Inverse agonist activity at RORgamma in human CD4+ T cells assessed as inhibition of IL17A secretion after 72 hrs by ELISAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/21/2022
Entry Details Article
PubMed
TargetNuclear receptor ROR-gamma(Human)
Inventiva

Curated by ChEMBL
LigandPNGBDBM50546028(CHEMBL4763038)
Affinity DataEC50:  1.83E+3nMAssay Description:Inverse agonist activity at RORgamma in human CD4+ T cells assessed as inhibition of IL17A secretion after 72 hrs by ELISAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/21/2022
Entry Details Article
PubMed
TargetNuclear receptor ROR-gamma(Human)
Inventiva

Curated by ChEMBL
LigandPNGBDBM50546025(CHEMBL4763421)
Affinity DataEC50:  890nMAssay Description:Inverse agonist activity at RORgamma in human CD4+ T cells assessed as inhibition of IL17A secretion after 72 hrs by ELISAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/21/2022
Entry Details Article
PubMed
TargetNuclear receptor ROR-gamma(Human)
Inventiva

Curated by ChEMBL
LigandPNGBDBM50546021(CHEMBL4759286)
Affinity DataEC50:  830nMAssay Description:Inverse agonist activity at RORgamma in human CD4+ T cells assessed as inhibition of IL17A secretion after 72 hrs by ELISAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/21/2022
Entry Details Article
PubMed
LigandPNGBDBM50616532(CHEMBL5424297)
Affinity DataEC50:  2.70E+4nMAssay Description:Activation of PXR (unknown origin) assessed as CYP3A4 inductionMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/13/2024
Entry Details
PubMed
TargetNuclear receptor ROR-gamma(Human)
Inventiva

Curated by ChEMBL
LigandPNGBDBM50426729(CHEMBL2326845)
Affinity DataEC50:  930nMAssay Description:Inverse agonist activity at RORgamma in human CD4+ T cells assessed as inhibition of IL17A secretion after 72 hrs by ELISAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/21/2022
Entry Details Article
PubMed
TargetNuclear receptor ROR-gamma(Human)
Inventiva

Curated by ChEMBL
LigandPNGBDBM50546026(CHEMBL4782026)
Affinity DataEC50:  2.07E+3nMAssay Description:Inverse agonist activity at RORgamma in human CD4+ T cells assessed as inhibition of IL17A secretion after 72 hrs by ELISAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/21/2022
Entry Details Article
PubMed
TargetNuclear receptor ROR-gamma(Human)
Inventiva

Curated by ChEMBL
LigandPNGBDBM50546017(CHEMBL4779432)
Affinity DataEC50:  210nMAssay Description:Inverse agonist activity at RORgamma in human CD4+ T cells assessed as inhibition of IL17A secretion after 72 hrs by ELISAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/21/2022
Entry Details Article
PubMed
TargetNuclear receptor ROR-gamma(Human)
Inventiva

Curated by ChEMBL
LigandPNGBDBM50546019(CHEMBL4752983)
Affinity DataEC50:  170nMAssay Description:Inverse agonist activity at pSG5GAL4-DBD/LBD fused human RORgamma receptor expressed in COS7 cells co-expressing 5 copies of GAL4 response element af...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/21/2022
Entry Details Article
PubMed
TargetHbpA(Pasteurella multocida)
Ghent University

LigandPNGBDBM225231(OXIGLUTATIONE | Disulfide, Glutathione | Oxidized ...)
Affinity DataKd:  150nMpH: 7.4 T: 2°CAssay Description:Experiments were carried out using a VP-ITC MicroCalorimeter (MicroCal) at 37°C, and data were analyzed using the Origen ITC analysis software packag...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/9/2017
Entry Details Article
PubMed
LigandPNGBDBM126830(US8785467, 1-39)
Affinity DataEC50:  6.00E+3nMAssay Description:Activation of PXR (unknown origin) assessed as CYP3A4 inductionMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/13/2024
Entry Details
PubMed
TargetNuclear receptor ROR-gamma(Human)
Inventiva

Curated by ChEMBL
LigandPNGBDBM50546030(CHEMBL4745208)
Affinity DataEC50:  150nMAssay Description:Inverse agonist activity at RORgamma in human CD4+ T cells assessed as inhibition of IL17A secretion after 72 hrs by ELISAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/21/2022
Entry Details Article
PubMed
LigandPNGBDBM147134(US8957077, J-5)
Affinity DataEC50:  2.30E+4nMAssay Description:Activation of PXR (unknown origin) assessed as CYP3A4 inductionMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/13/2024
Entry Details
PubMed
TargetNuclear receptor ROR-gamma(Human)
Inventiva

Curated by ChEMBL
LigandPNGBDBM50546027(CHEMBL4779716)
Affinity DataEC50:  1.01E+3nMAssay Description:Inverse agonist activity at RORgamma in human CD4+ T cells assessed as inhibition of IL17A secretion after 72 hrs by ELISAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/21/2022
Entry Details Article
PubMed
TargetNuclear receptor ROR-gamma(Human)
Inventiva

Curated by ChEMBL
LigandPNGBDBM50426729(CHEMBL2326845)
Affinity DataEC50:  1.08E+3nMAssay Description:Inverse agonist activity at pSG5GAL4-DBD/LBD fused human RORgamma receptor expressed in COS7 cells co-expressing 5 copies of GAL4 response element af...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/21/2022
Entry Details Article
PubMed
TargetHbpA(Pasteurella multocida)
Ghent University

LigandPNGBDBM225232(S-methylglutathione)
Affinity DataKd:  550nMpH: 7.4 T: 2°CAssay Description:Experiments were carried out using a VP-ITC MicroCalorimeter (MicroCal) at 37°C, and data were analyzed using the Origen ITC analysis software packag...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/9/2017
Entry Details Article
PubMed
TargetNuclear receptor ROR-gamma(Human)
Inventiva

Curated by ChEMBL
LigandPNGBDBM50546020(CHEMBL4740086)
Affinity DataEC50:  440nMAssay Description:Inverse agonist activity at pSG5GAL4-DBD/LBD fused human RORgamma receptor expressed in COS7 cells co-expressing 5 copies of GAL4 response element af...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/21/2022
Entry Details Article
PubMed
TargetNuclear receptor ROR-gamma(Human)
Inventiva

Curated by ChEMBL
LigandPNGBDBM50546035(CHEMBL4760072)
Affinity DataEC50:  900nMAssay Description:Inverse agonist activity at pSG5GAL4-DBD/LBD fused human RORgamma receptor expressed in COS7 cells co-expressing 5 copies of GAL4 response element af...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/21/2022
Entry Details Article
PubMed
TargetNuclear receptor ROR-gamma(Human)
Inventiva

Curated by ChEMBL
LigandPNGBDBM50546025(CHEMBL4763421)
Affinity DataEC50:  320nMAssay Description:Inverse agonist activity at pSG5GAL4-DBD/LBD fused human RORgamma receptor expressed in COS7 cells co-expressing 5 copies of GAL4 response element af...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/21/2022
Entry Details Article
PubMed
TargetNuclear receptor ROR-gamma(Human)
Inventiva

Curated by ChEMBL
LigandPNGBDBM50546020(CHEMBL4740086)
Affinity DataEC50:  470nMAssay Description:Inverse agonist activity at RORgamma in human CD4+ T cells assessed as inhibition of IL17A secretion after 72 hrs by ELISAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/21/2022
Entry Details Article
PubMed
TargetHeme-binding protein A(Haemophilus parasuis)
Ghent University

LigandPNGBDBM50422268(GLUTATHIONE | GSH)
Affinity DataKd:  1.90E+3nMpH: 7.4 T: 2°CAssay Description:Experiments were carried out using a VP-ITC MicroCalorimeter (MicroCal) at 37°C, and data were analyzed using the Origen ITC analysis software packag...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/9/2017
Entry Details Article
PubMed
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