Compile Data Set for Download or QSAR
Report error Found 2 Enz. Inhib. hit(s) with Target = 'P2Y purinoceptor 12' and Ligand = 'BDBM50100245'
TargetP2Y purinoceptor 12(Human)
Sanofi R & D

Curated by ChEMBL
LigandPNGBDBM50100245(CHEMBL3325894)
Affinity DataIC50: 7nMAssay Description:Displacement of [33P]2MeS-ADP from P2Y12 receptor (unknown origin) transfected in CHO cells after 30 mins by scintillation counting analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/30/2016
Entry Details Article
PubMed
TargetP2Y purinoceptor 12(Rat)
Sanofi R & D

Curated by ChEMBL
LigandPNGBDBM50100245(CHEMBL3325894)
Affinity DataIC50: 20nMAssay Description:Antagonist activity at P2Y12 receptor in Sprague-Dawley rat platelet rich plasma assessed as inhibition of ADP-induced aggregationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/30/2016
Entry Details Article
PubMed