Report error Found 1117 Enz. Inhib. hit(s) with Target = 'Protein P'
Displayed 1 to 50 (of 1117 total ) | Next | Last >>
Affinity DataIC50: 0.300nMAssay Description:Inhibitory concentration against protein phosphatase 1 (PP1) using phosphorylase-a assayMore data for this Ligand-Target Pair
Affinity DataKd: <1nMAssay Description:Binding affinity to human partial length PBRM1 bromodomain 5 (S645 to D766 residues) expressed in bacterial expression system by BROMOscan assayMore data for this Ligand-Target Pair
Affinity DataKd: <1nMAssay Description:Binding affinity to human partial length PBRM1 bromodomain 2 (S178 to E291 residues) expressed in bacterial expression system by BROMOscan assayMore data for this Ligand-Target Pair
Affinity DataIC50: 2.5nMAssay Description:Histidine-Flag-PB1-BD5 Bromodomain645-766 (S645-D766; Swiss Prot Q86U86; mhhhhhhasdykddddkgslvprgsSGISPKKSKYMTPMQQKLNEVYEAVKNYTDKRGRRLSAI FLRLPSRSELP...More data for this Ligand-Target Pair
TargetProtein phosphatase 3 catalytic subunit alpha(Human)
Merck Research Laboratories
Curated by ChEMBL
Merck Research Laboratories
Curated by ChEMBL
Affinity DataIC50: 2.80nMAssay Description:Inhibitory activity against Calcineurin (CaN phosphatase)More data for this Ligand-Target Pair
Affinity DataIC50: 3nMAssay Description:Test compounds (252 mM stock in DMSO) were diluted 3 folds in series in DMSO and 1.2 μl per well were added into 384-well polypropylene black pl...More data for this Ligand-Target Pair
Affinity DataIC50: 3nMAssay Description:Test compounds (252 mM stock in DMSO) were diluted 3 folds in series in DMSO and 1.2 μl per well were added into 384-well polypropylene black pl...More data for this Ligand-Target Pair
Affinity DataIC50: 3nMAssay Description:Inhibitory concentration against protein phosphatase 1 (PP1) using pNPP assayMore data for this Ligand-Target Pair
Affinity DataIC50: 3nMAssay Description:Inhibitory concentration required against protein phosphatase 1 using pNPP assayMore data for this Ligand-Target Pair
Affinity DataIC50: 3.70nMAssay Description:Histidine-Flag-PB1-BD5 Bromodomain645-766 (S645-D766; Swiss Prot Q86U86; mhhhhhhasdykddddkgslvprgsSGISPKKSKYMTPMQQKLNEVYEAVKNYTDKRGRRLSAI FLRLPSRSELP...More data for this Ligand-Target Pair
Affinity DataIC50: 4nMAssay Description:Test compounds (252 mM stock in DMSO) were diluted 3 folds in series in DMSO and 1.2 μl per well were added into 384-well polypropylene black pl...More data for this Ligand-Target Pair
Affinity DataIC50: 4nMAssay Description:Test compounds (252 mM stock in DMSO) were diluted 3 folds in series in DMSO and 1.2 μl per well were added into 384-well polypropylene black pl...More data for this Ligand-Target Pair
Affinity DataIC50: 4nMAssay Description:Test compounds (252 mM stock in DMSO) were diluted 3 folds in series in DMSO and 1.2 μl per well were added into 384-well polypropylene black pl...More data for this Ligand-Target Pair
Affinity DataIC50: 4nMAssay Description:Test compounds (252 mM stock in DMSO) were diluted 3 folds in series in DMSO and 1.2 μl per well were added into 384-well polypropylene black pl...More data for this Ligand-Target Pair
Affinity DataIC50: 4nMAssay Description:Test compounds (252 mM stock in DMSO) were diluted 3 folds in series in DMSO and 1.2 μl per well were added into 384-well polypropylene black pl...More data for this Ligand-Target Pair
TargetProtein phosphatase 3 catalytic subunit alpha(Human)
Merck Research Laboratories
Curated by ChEMBL
Merck Research Laboratories
Curated by ChEMBL
Affinity DataKd: 4nMAssay Description:Binding affinity to protein phosphatase, calcineurin (CN) was determinedMore data for this Ligand-Target Pair
Affinity DataIC50: 4nMAssay Description:Test compounds (252 mM stock in DMSO) were diluted 3 folds in series in DMSO and 1.2 μl per well were added into 384-well polypropylene black pl...More data for this Ligand-Target Pair
TargetProtein phosphatase 3 catalytic subunit alpha(Human)
Merck Research Laboratories
Curated by ChEMBL
Merck Research Laboratories
Curated by ChEMBL
Affinity DataIC50: 4nMAssay Description:Inhibitory activity against Calcineurin (CaN phosphatase)More data for this Ligand-Target Pair
Affinity DataIC50: 4nMAssay Description:Test compounds (252 mM stock in DMSO) were diluted 3 folds in series in DMSO and 1.2 μl per well were added into 384-well polypropylene black pl...More data for this Ligand-Target Pair
Affinity DataIC50: 4nMAssay Description:Test compounds (252 mM stock in DMSO) were diluted 3 folds in series in DMSO and 1.2 μl per well were added into 384-well polypropylene black pl...More data for this Ligand-Target Pair
Affinity DataIC50: 4nMAssay Description:Test compounds (252 mM stock in DMSO) were diluted 3 folds in series in DMSO and 1.2 μl per well were added into 384-well polypropylene black pl...More data for this Ligand-Target Pair
Affinity DataIC50: 4nMAssay Description:Test compounds (252 mM stock in DMSO) were diluted 3 folds in series in DMSO and 1.2 μl per well were added into 384-well polypropylene black pl...More data for this Ligand-Target Pair
Affinity DataIC50: 4nMAssay Description:Test compounds (252 mM stock in DMSO) were diluted 3 folds in series in DMSO and 1.2 μl per well were added into 384-well polypropylene black pl...More data for this Ligand-Target Pair
TargetProtein phosphatase 3 catalytic subunit alpha(Human)
Merck Research Laboratories
Curated by ChEMBL
Merck Research Laboratories
Curated by ChEMBL
Affinity DataIC50: 4.20nMAssay Description:Inhibitory activity against Calcineurin (CaN phosphatase)More data for this Ligand-Target Pair
TargetProtein phosphatase 3 catalytic subunit alpha(Human)
Merck Research Laboratories
Curated by ChEMBL
Merck Research Laboratories
Curated by ChEMBL
Affinity DataIC50: 4.90nMAssay Description:Inhibitory activity against Calcineurin (CaN phosphatase)More data for this Ligand-Target Pair
Affinity DataIC50: 5nMAssay Description:Test compounds (252 mM stock in DMSO) were diluted 3 folds in series in DMSO and 1.2 μl per well were added into 384-well polypropylene black pl...More data for this Ligand-Target Pair
Affinity DataIC50: 5nMAssay Description:Test compounds (252 mM stock in DMSO) were diluted 3 folds in series in DMSO and 1.2 μl per well were added into 384-well polypropylene black pl...More data for this Ligand-Target Pair
Affinity DataIC50: 5nMAssay Description:Test compounds (252 mM stock in DMSO) were diluted 3 folds in series in DMSO and 1.2 μl per well were added into 384-well polypropylene black pl...More data for this Ligand-Target Pair
Affinity DataIC50: 5nMAssay Description:Test compounds (252 mM stock in DMSO) were diluted 3 folds in series in DMSO and 1.2 μl per well were added into 384-well polypropylene black pl...More data for this Ligand-Target Pair
Affinity DataIC50: 5nMAssay Description:Test compounds (252 mM stock in DMSO) were diluted 3 folds in series in DMSO and 1.2 μl per well were added into 384-well polypropylene black pl...More data for this Ligand-Target Pair
Affinity DataIC50: 5nMAssay Description:Test compounds (252 mM stock in DMSO) were diluted 3 folds in series in DMSO and 1.2 μl per well were added into 384-well polypropylene black pl...More data for this Ligand-Target Pair
Affinity DataIC50: 5nMAssay Description:Test compounds (252 mM stock in DMSO) were diluted 3 folds in series in DMSO and 1.2 μl per well were added into 384-well polypropylene black pl...More data for this Ligand-Target Pair
Affinity DataIC50: 5nMAssay Description:Test compounds (252 mM stock in DMSO) were diluted 3 folds in series in DMSO and 1.2 μl per well were added into 384-well polypropylene black pl...More data for this Ligand-Target Pair
Affinity DataIC50: 5nMAssay Description:Protein phosphatase inhibitory activity of calyculin derivatives.More data for this Ligand-Target Pair
Affinity DataIC50: 5nMAssay Description:Test compounds (252 mM stock in DMSO) were diluted 3 folds in series in DMSO and 1.2 μl per well were added into 384-well polypropylene black pl...More data for this Ligand-Target Pair
Affinity DataKd: 5nMAssay Description:Binding affinity to PBRM1 bromodomain 2 (unknown origin) assessed as dissociation constant by BROMOscan LeadHunter assayMore data for this Ligand-Target Pair
Affinity DataIC50: 5nMAssay Description:Test compounds (252 mM stock in DMSO) were diluted 3 folds in series in DMSO and 1.2 μl per well were added into 384-well polypropylene black pl...More data for this Ligand-Target Pair
Affinity DataIC50: 5nMAssay Description:Test compounds (252 mM stock in DMSO) were diluted 3 folds in series in DMSO and 1.2 μl per well were added into 384-well polypropylene black pl...More data for this Ligand-Target Pair
Affinity DataIC50: 5nMAssay Description:Test compounds (252 mM stock in DMSO) were diluted 3 folds in series in DMSO and 1.2 μl per well were added into 384-well polypropylene black pl...More data for this Ligand-Target Pair
Affinity DataIC50: 5nMAssay Description:Test compounds (252 mM stock in DMSO) were diluted 3 folds in series in DMSO and 1.2 μl per well were added into 384-well polypropylene black pl...More data for this Ligand-Target Pair
Affinity DataIC50: 5nMAssay Description:Test compounds (252 mM stock in DMSO) were diluted 3 folds in series in DMSO and 1.2 μl per well were added into 384-well polypropylene black pl...More data for this Ligand-Target Pair
Affinity DataIC50: 5nMAssay Description:Test compounds (252 mM stock in DMSO) were diluted 3 folds in series in DMSO and 1.2 μl per well were added into 384-well polypropylene black pl...More data for this Ligand-Target Pair
Affinity DataIC50: 5nMAssay Description:Test compounds (252 mM stock in DMSO) were diluted 3 folds in series in DMSO and 1.2 μl per well were added into 384-well polypropylene black pl...More data for this Ligand-Target Pair
Affinity DataIC50: 5nMAssay Description:Test compounds (252 mM stock in DMSO) were diluted 3 folds in series in DMSO and 1.2 μl per well were added into 384-well polypropylene black pl...More data for this Ligand-Target Pair
Affinity DataIC50: 5nMAssay Description:Test compounds (252 mM stock in DMSO) were diluted 3 folds in series in DMSO and 1.2 μl per well were added into 384-well polypropylene black pl...More data for this Ligand-Target Pair
Affinity DataIC50: 5nMAssay Description:Test compounds (252 mM stock in DMSO) were diluted 3 folds in series in DMSO and 1.2 μl per well were added into 384-well polypropylene black pl...More data for this Ligand-Target Pair
Affinity DataIC50: 5nMAssay Description:Test compounds (252 mM stock in DMSO) were diluted 3 folds in series in DMSO and 1.2 μl per well were added into 384-well polypropylene black pl...More data for this Ligand-Target Pair
Affinity DataIC50: 5.20nMAssay Description:Histidine-Flag-PB1-BD5 Bromodomain645-766 (S645-D766; Swiss Prot Q86U86; mhhhhhhasdykddddkgslvprgsSGISPKKSKYMTPMQQKLNEVYEAVKNYTDKRGRRLSAI FLRLPSRSELP...More data for this Ligand-Target Pair
Affinity DataIC50: 5.30nMAssay Description:Histidine-Flag-PB1-BD5 Bromodomain645-766 (S645-D766; Swiss Prot Q86U86; mhhhhhhasdykddddkgslvprgsSGISPKKSKYMTPMQQKLNEVYEAVKNYTDKRGRRLSAI FLRLPSRSELP...More data for this Ligand-Target Pair
TargetProtein phosphatase 3 catalytic subunit alpha(Human)
Merck Research Laboratories
Curated by ChEMBL
Merck Research Laboratories
Curated by ChEMBL
Affinity DataIC50: 5.90nMAssay Description:Inhibitory activity against Calcineurin (CaN phosphatase)More data for this Ligand-Target Pair















































