BDBM50232143 CHEMBL398339::N-[(1S)-5-tert-butyl-2,3-dihydro-1H-inden-1-yl]-N'-1H-indazol-4-ylurea

SMILES CC(C)(C)c1ccc2[C@H](CCc2c1)NC(=O)Nc1cccc2[nH]ncc12

InChI Key InChIKey=TYOYXJNGINZFET-UHFFFAOYSA-N

Data  1 IC50

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 50232143   

TargetTransient receptor potential cation channel subfamily V member 1(Human)
Abbott Laboratories

Curated by ChEMBL

LigandBDBM50232143(N-[(1S)-5-tert-butyl-2,3-dihydro-1H-inden-1-yl]-N'...)Copy SMILESCopy InChI

Affinity DataIC50: 123nMAssay Description:Blockade of human TRPV1 receptor assessed as inhibition of capsaicin-induced calcium fluxMore data for this Ligand-Target Pair

Target InfoPDBKEGG
UniProtKB/SwissProt
GoogleScholar

Ligand InfoPurchaseCHEMBLPC cidPC sidSimilars

In Depth
Date in BDB:
11/11/2009
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