BDBM50232139 1-(6,7-dihydro-5H-[1]pyridin-7-yl)-3-(1H-indazol-4-yl)-urea::CHEMBL399978

SMILES O=C(NC1CCc2cccnc12)Nc1cccc2[nH]ncc12

InChI Key InChIKey=MNELSNAYLAVDIE-UHFFFAOYSA-N

Data  1 IC50

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 50232139   

TargetTransient receptor potential cation channel subfamily V member 1(Human)
Abbott Laboratories

Curated by ChEMBL

LigandBDBM50232139(1-(6,7-dihydro-5H-[1]pyridin-7-yl)-3-(1H-indazol-4...)Copy SMILESCopy InChI

Affinity DataIC50: 1.35E+3nMAssay Description:Blockade of human TRPV1 receptor assessed as inhibition of capsaicin-induced calcium fluxMore data for this Ligand-Target Pair

Target InfoPDBKEGG
UniProtKB/SwissProt
GoogleScholar

Ligand InfoCHEMBLPC cidPC sidSimilars

In Depth
Date in BDB:
11/11/2009
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