BDBM50204472 CHEMBL3915177

SMILES OCc1ccc(o1)-c1nc(-c2cc(cc(c2)C(F)(F)F)C(F)(F)F)c2ccccn12

InChI Key InChIKey=TYHUMMGPUUALTI-UHFFFAOYSA-N

Data  1 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 50204472   

TargetEndothelial PAS domain-containing protein 1/Hypoxia-inducible factor 1-alpha(Human)
Tokyo Institute of Innovative Research

Curated by ChEMBL
LigandPNGBDBM50204472(CHEMBL3915177)
Affinity DataIC50: 2.50E+4nMAssay Description:Inhibition of hypoxia-induced HIF1 transcriptional activity in human HeLa cells measured after 12 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2018
Entry Details Article
PubMed