BDBM50019977 CHEMBL3287828

SMILES Clc1ccc(NC(=N)c2cccs2)cc1CSC1CCCC1

InChI Key InChIKey=DSJGZGZLLJYVLQ-UHFFFAOYSA-N

Data  2 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 2 hits for monomerid = 50019977   

TargetPyroglutamylated RF-amide peptide receptor(Human)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50019977(CHEMBL3287828)
Affinity DataIC50: 3.98E+3nMAssay Description:Displacement of [125I]-QRFP43 from human GPR103 receptor overexpressed in HEK membranes after 90 mins by liquid scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/11/2015
Entry Details Article
PubMed
TargetPyroglutamylated RF-amide peptide receptor(Human)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50019977(CHEMBL3287828)
Affinity DataIC50: 1.00E+3nMAssay Description:Antagonist activity at human GPR103 receptor assessed as inhibition of inositol-1-phosphate production by cell-based assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/11/2015
Entry Details Article
PubMed