Compile Data Set for Download or QSAR
Report error Found 119 of affinity data for UniProtKB/TrEMBL: Q61606
TargetGlucagon receptor(Mouse)
Sanofi-Aventis Deutschland

Curated by ChEMBL
LigandPNGBDBM50241203(exenatide | HGEGTFTSDLSKQMEEEAVRLFIEWLKNGGPSSGSPPP...)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at mouse glucagon receptor expressed in HEK293 cells assessed as cAMP accumulation after 30 mins by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/19/2020
Entry Details Article
PubMed
TargetGlucagon receptor(Mouse)
Sanofi-Aventis Deutschland

Curated by ChEMBL
LigandPNGBDBM50152769(GLP-1(7-36)-NH2 | NH2-HAEGTFTSDVSSYLEGQAAKEFIAWLVK...)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at mouse glucagon receptor expressed in HEK293 cells assessed as cAMP accumulation after 30 mins by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/19/2020
Entry Details Article
PubMed
TargetGlucagon receptor(Mouse)
Sanofi-Aventis Deutschland

Curated by ChEMBL
LigandPNGBDBM50266690(CHEMBL439305)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at mouse glucagon receptor expressed in HEK293 cells assessed as cAMP accumulation after 30 mins by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/19/2020
Entry Details Article
PubMed
TargetGlucagon receptor(Mouse)
Sanofi-Aventis Deutschland

Curated by ChEMBL
LigandPNGBDBM50266693(CHEBI:5391 | Glucagen Hypokit | Glucagon | Glucago...)
Affinity DataEC50:  0.00130nMAssay Description:Agonist activity at mouse glucagon receptor expressed in HEK293 cells assessed as cAMP accumulation after 30 mins by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/19/2020
Entry Details Article
PubMed
TargetGlucagon receptor(Mouse)
Sanofi-Aventis Deutschland

Curated by ChEMBL
LigandPNGBDBM50266691(CHEMBL4086979)
Affinity DataEC50:  0.0250nMAssay Description:Agonist activity at mouse glucagon receptor expressed in HEK293 cells assessed as cAMP accumulation after 30 mins by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/19/2020
Entry Details Article
PubMed
TargetGlucagon receptor(Mouse)
Sanofi-Aventis Deutschland

Curated by ChEMBL
LigandPNGBDBM50266693(CHEBI:5391 | Glucagen Hypokit | Glucagon | Glucago...)
Affinity DataEC50:  0.0200nMAssay Description:Agonist activity at mouse GCG receptor expressed in CHO cells assessed as increase in cAMP level by TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
TargetGlucagon receptor(Mouse)
Sanofi-Aventis Deutschland

Curated by ChEMBL
LigandPNGBDBM50459979(CHEMBL4227636)
Affinity DataEC50: >100nMAssay Description:Agonist activity at mouse GCG receptor expressed in CHO cells assessed as increase in cAMP level by TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
TargetGlucagon receptor(Mouse)
Sanofi-Aventis Deutschland

Curated by ChEMBL
LigandPNGBDBM50612019(CHEMBL5219598)
Affinity DataEC50:  6.10nMAssay Description:Agonist activity at mouse GCGR expressed in CHO cells assessed as increase in cAMP accumulationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/21/2024
Entry Details
PubMed
TargetGlucagon receptor(Mouse)
Sanofi-Aventis Deutschland

Curated by ChEMBL
LigandPNGBDBM50612020(CHEMBL5285379)
Affinity DataEC50:  5.90nMAssay Description:Agonist activity at mouse GCGR expressed in CHO cells assessed as increase in cAMP accumulationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/21/2024
Entry Details
PubMed
TargetGlucagon receptor(Mouse)
Sanofi-Aventis Deutschland

Curated by ChEMBL
LigandPNGBDBM50612021(CHEMBL5277323)
Affinity DataEC50:  6.10nMAssay Description:Agonist activity at mouse GCGR expressed in CHO cells assessed as increase in cAMP accumulationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/21/2024
Entry Details
PubMed
TargetGlucagon receptor(Mouse)
Sanofi-Aventis Deutschland

Curated by ChEMBL
LigandPNGBDBM50612022(CHEMBL5287118)
Affinity DataEC50:  3.40nMAssay Description:Agonist activity at mouse GCGR expressed in CHO cells assessed as increase in cAMP accumulationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/21/2024
Entry Details
PubMed
TargetGlucagon receptor(Mouse)
Sanofi-Aventis Deutschland

Curated by ChEMBL
LigandPNGBDBM50612023(CHEMBL5266722)
Affinity DataEC50:  0.940nMAssay Description:Agonist activity at mouse GCGR expressed in CHO cells assessed as increase in cAMP accumulationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/21/2024
Entry Details
PubMed
TargetGlucagon receptor(Mouse)
Sanofi-Aventis Deutschland

Curated by ChEMBL
LigandPNGBDBM50612024(CHEMBL5275572)
Affinity DataEC50:  1.40nMAssay Description:Agonist activity at mouse GCGR expressed in CHO cells assessed as increase in cAMP accumulationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/21/2024
Entry Details
PubMed
TargetGlucagon receptor(Mouse)
Sanofi-Aventis Deutschland

Curated by ChEMBL
LigandPNGBDBM50612025(CHEMBL5272283)
Affinity DataEC50:  9nMAssay Description:Agonist activity at mouse GCGR expressed in CHO cells assessed as increase in cAMP accumulationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/21/2024
Entry Details
PubMed
TargetGlucagon receptor(Mouse)
Sanofi-Aventis Deutschland

Curated by ChEMBL
LigandPNGBDBM50612026(CHEMBL5288119)
Affinity DataEC50:  0.530nMAssay Description:Agonist activity at mouse GCGR expressed in CHO cells assessed as increase in cAMP accumulationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/21/2024
Entry Details
PubMed
TargetGlucagon receptor(Mouse)
Sanofi-Aventis Deutschland

Curated by ChEMBL
LigandPNGBDBM50612027(CHEMBL5282576)
Affinity DataEC50:  0.680nMAssay Description:Agonist activity at mouse GCGR expressed in CHO cells assessed as increase in cAMP accumulationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/21/2024
Entry Details
PubMed
TargetGlucagon receptor(Mouse)
Sanofi-Aventis Deutschland

Curated by ChEMBL
LigandPNGBDBM50612028(CHEMBL5268054)
Affinity DataEC50:  0.590nMAssay Description:Agonist activity at mouse GCGR expressed in CHO cells assessed as increase in cAMP accumulationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/21/2024
Entry Details
PubMed
TargetGlucagon receptor(Mouse)
Sanofi-Aventis Deutschland

Curated by ChEMBL
LigandPNGBDBM50266693(CHEBI:5391 | Glucagen Hypokit | Glucagon | Glucago...)
Affinity DataEC50:  0.340nMAssay Description:Agonist activity at mouse GCGR expressed in CHO cells assessed as increase in cAMP accumulationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/21/2024
Entry Details
PubMed
TargetGlucagon receptor(Mouse)
Sanofi-Aventis Deutschland

Curated by ChEMBL
LigandPNGBDBM50566470(CHEMBL4857523)
Affinity DataIC50: 0.530nMAssay Description:Antagonist activity at mouse GCGR expressed in CHO-K1 cells assessed as inhibition of glucogon-induced cAMP productionMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2022
Entry Details Article
PubMed
TargetGlucagon receptor(Mouse)
Sanofi-Aventis Deutschland

Curated by ChEMBL
LigandPNGBDBM50566469(CHEMBL4876736)
Affinity DataIC50: 23nMAssay Description:Antagonist activity at mouse GCGR expressed in CHO-K1 cells assessed as inhibition of glucogon-induced cAMP productionMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2022
Entry Details Article
PubMed
TargetGlucagon receptor(Mouse)
Sanofi-Aventis Deutschland

Curated by ChEMBL
LigandPNGBDBM50075766(4-[5-(4-Chloro-phenyl)-3-(2-propoxy-phenyl)-1H-pyr...)
Affinity DataIC50: 30nMAssay Description:Binding affinity towards glucagon receptor determined by reduction in binding of 125 I-glucagon to the murine glucagon receptor (mGLUR) expressed on ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGlucagon receptor(Mouse)
Sanofi-Aventis Deutschland

Curated by ChEMBL
LigandPNGBDBM50075775(4-[3-(5-Bromo-2-propoxy-phenyl)-5-(4-chloro-phenyl...)
Affinity DataIC50: 37nMAssay Description:Binding affinity towards glucagon receptor determined by reduction in binding of 125 I-glucagon to the murine glucagon receptor (mGLUR) expressed on ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGlucagon receptor(Mouse)
Sanofi-Aventis Deutschland

Curated by ChEMBL
LigandPNGBDBM50075787(4-[3-(4-Bromo-2-propoxy-phenyl)-5-(4-chloro-phenyl...)
Affinity DataIC50: 49nMAssay Description:Binding affinity towards glucagon receptor determined by reduction in binding of [125I]glucagon to the murine glucagon receptor (GGR) expressed on CH...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGlucagon receptor(Mouse)
Sanofi-Aventis Deutschland

Curated by ChEMBL
LigandPNGBDBM50075783(4-[5-(4-Chloro-phenyl)-3-(5-chloro-2-propoxy-pheny...)
Affinity DataIC50: 50nMAssay Description:Binding affinity towards glucagon receptor determined by reduction in binding of 125 I-glucagon to the murine glucagon receptor (mGLUR) expressed on ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGlucagon receptor(Mouse)
Sanofi-Aventis Deutschland

Curated by ChEMBL
LigandPNGBDBM50075748(4-[5-(4-Chloro-phenyl)-3-cyclohexyl-1H-pyrrol-2-yl...)
Affinity DataIC50: 60nMAssay Description:Binding affinity towards glucagon receptor determined by reduction in binding of 125 I-glucagon to the murine glucagon receptor (mGLUR) expressed on ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGlucagon receptor(Mouse)
Sanofi-Aventis Deutschland

Curated by ChEMBL
LigandPNGBDBM50075780(4-[5-(4-Chloro-phenyl)-3-isopropyl-1H-pyrrol-2-yl]...)
Affinity DataIC50: 60nMAssay Description:Binding affinity towards glucagon receptor determined by reduction in binding of 125 I-glucagon to the murine glucagon receptor (mGLUR) expressed on ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGlucagon receptor(Mouse)
Sanofi-Aventis Deutschland

Curated by ChEMBL
LigandPNGBDBM50075772(4-[3-(2-Butoxy-phenyl)-5-(4-chloro-phenyl)-1H-pyrr...)
Affinity DataIC50: 80nMAssay Description:Binding affinity towards glucagon receptor determined by reduction in binding of [125I]glucagon to the murine glucagon receptor (GGR) expressed on CH...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGlucagon receptor(Mouse)
Sanofi-Aventis Deutschland

Curated by ChEMBL
LigandPNGBDBM50007239(CHEMBL3238226)
Affinity DataIC50: 84nMAssay Description:Displacement of [125I]-glucagon from GCGR in mouse liver membranes after 60 mins by scintillation counting analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2015
Entry Details Article
PubMed
TargetGlucagon receptor(Mouse)
Sanofi-Aventis Deutschland

Curated by ChEMBL
LigandPNGBDBM50007231(CHEMBL3238221)
Affinity DataIC50: 90nMAssay Description:Displacement of [125I]-glucagon from GCGR in mouse liver membranes after 60 mins by scintillation counting analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2015
Entry Details Article
PubMed
TargetGlucagon receptor(Mouse)
Sanofi-Aventis Deutschland

Curated by ChEMBL
LigandPNGBDBM50007240(CHEMBL3238228)
Affinity DataIC50: 96nMAssay Description:Displacement of [125I]-glucagon from GCGR in mouse liver membranes after 60 mins by scintillation counting analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2015
Entry Details Article
PubMed
TargetGlucagon receptor(Mouse)
Sanofi-Aventis Deutschland

Curated by ChEMBL
LigandPNGBDBM50007228(CHEMBL3238219)
Affinity DataIC50: 100nMAssay Description:Displacement of [125I]-glucagon from GCGR in mouse liver membranes after 60 mins by scintillation counting analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2015
Entry Details Article
PubMed
TargetGlucagon receptor(Mouse)
Sanofi-Aventis Deutschland

Curated by ChEMBL
LigandPNGBDBM50007219(CHEMBL3238214)
Affinity DataIC50: 110nMAssay Description:Displacement of [125I]-glucagon from GCGR in mouse liver membranes after 60 mins by scintillation counting analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2015
Entry Details Article
PubMed
TargetGlucagon receptor(Mouse)
Sanofi-Aventis Deutschland

Curated by ChEMBL
LigandPNGBDBM50007223(CHEMBL3238215)
Affinity DataIC50: 110nMAssay Description:Displacement of [125I]-glucagon from GCGR in mouse liver membranes after 60 mins by scintillation counting analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2015
Entry Details Article
PubMed
TargetGlucagon receptor(Mouse)
Sanofi-Aventis Deutschland

Curated by ChEMBL
LigandPNGBDBM50360601(CHEMBL1933349 | MK-0893)
Affinity DataIC50: 122nMAssay Description:Antagonist activity at mouse GCGR expressed in CHO cells assessed as inhibition of glucagon-induced cAMP accumulation preincubated for 30 mins prior ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetGlucagon receptor(Mouse)
Sanofi-Aventis Deutschland

Curated by ChEMBL
LigandPNGBDBM50007226(CHEMBL3238218)
Affinity DataIC50: 130nMAssay Description:Displacement of [125I]-glucagon from GCGR in mouse liver membranes after 60 mins by scintillation counting analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2015
Entry Details Article
PubMed
TargetGlucagon receptor(Mouse)
Sanofi-Aventis Deutschland

Curated by ChEMBL
LigandPNGBDBM50007296(CHEMBL3238246)
Affinity DataIC50: 130nMAssay Description:Displacement of [125I]-glucagon from GCGR in mouse liver membranes after 60 mins by scintillation counting analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2015
Entry Details Article
PubMed
TargetGlucagon receptor(Mouse)
Sanofi-Aventis Deutschland

Curated by ChEMBL
LigandPNGBDBM50007225(CHEMBL3238217)
Affinity DataIC50: 140nMAssay Description:Displacement of [125I]-glucagon from GCGR in mouse liver membranes after 60 mins by scintillation counting analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2015
Entry Details Article
PubMed
TargetGlucagon receptor(Mouse)
Sanofi-Aventis Deutschland

Curated by ChEMBL
LigandPNGBDBM50007233(CHEMBL3238223)
Affinity DataIC50: 140nMAssay Description:Displacement of [125I]-glucagon from GCGR in mouse liver membranes after 60 mins by scintillation counting analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2015
Entry Details Article
PubMed
TargetGlucagon receptor(Mouse)
Sanofi-Aventis Deutschland

Curated by ChEMBL
LigandPNGBDBM50075752(4-[5-(4-Chloro-phenyl)-3-(2-isobutoxy-phenyl)-1H-p...)
Affinity DataIC50: 150nMAssay Description:Binding affinity towards glucagon receptor determined by reduction in binding of 125 I-glucagon to the murine glucagon receptor (mGLUR) expressed on ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGlucagon receptor(Mouse)
Sanofi-Aventis Deutschland

Curated by ChEMBL
LigandPNGBDBM50007224(CHEMBL3238216)
Affinity DataIC50: 160nMAssay Description:Displacement of [125I]-glucagon from GCGR in mouse liver membranes after 60 mins by scintillation counting analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2015
Entry Details Article
PubMed
TargetGlucagon receptor(Mouse)
Sanofi-Aventis Deutschland

Curated by ChEMBL
LigandPNGBDBM50007232(CHEMBL3238222)
Affinity DataIC50: 170nMAssay Description:Displacement of [125I]-glucagon from GCGR in mouse liver membranes after 60 mins by scintillation counting analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2015
Entry Details Article
PubMed
TargetGlucagon receptor(Mouse)
Sanofi-Aventis Deutschland

Curated by ChEMBL
LigandPNGBDBM50007230(CHEMBL3238220)
Affinity DataIC50: 190nMAssay Description:Displacement of [125I]-glucagon from GCGR in mouse liver membranes after 60 mins by scintillation counting analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2015
Entry Details Article
PubMed
TargetGlucagon receptor(Mouse)
Sanofi-Aventis Deutschland

Curated by ChEMBL
LigandPNGBDBM50071899(4-[5-(4-Chloro-phenyl)-3-(4-fluoro-phenyl)-1H-pyrr...)
Affinity DataIC50: 200nMAssay Description:Binding affinity towards glucagon receptor determined by reduction in binding of 125 I-glucagon to the murine glucagon receptor (mGLUR) expressed on ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGlucagon receptor(Mouse)
Sanofi-Aventis Deutschland

Curated by ChEMBL
LigandPNGBDBM50007241(CHEMBL3238229)
Affinity DataIC50: 200nMAssay Description:Displacement of [125I]-glucagon from GCGR in mouse liver membranes after 60 mins by scintillation counting analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2015
Entry Details Article
PubMed
TargetGlucagon receptor(Mouse)
Sanofi-Aventis Deutschland

Curated by ChEMBL
LigandPNGBDBM50075764(4-[3,5-Bis-(4-chloro-phenyl)-1H-pyrrol-2-yl]-pyrid...)
Affinity DataIC50: 220nMAssay Description:Binding affinity towards glucagon receptor determined by reduction in binding of 125 I-glucagon to the murine glucagon receptor (mGLUR) expressed on ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGlucagon receptor(Mouse)
Sanofi-Aventis Deutschland

Curated by ChEMBL
LigandPNGBDBM50075767(4-[3-(3-Bromo-phenyl)-5-(4-chloro-phenyl)-1H-pyrro...)
Affinity DataIC50: 230nMAssay Description:Binding affinity towards glucagon receptor determined by reduction in binding of 125 I-glucagon to the murine glucagon receptor (mGLUR) expressed on ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGlucagon receptor(Mouse)
Sanofi-Aventis Deutschland

Curated by ChEMBL
LigandPNGBDBM50075751(4-[4-(4-Fluoro-phenyl)-5-pyridin-4-yl-1H-pyrrol-2-...)
Affinity DataIC50: 230nMAssay Description:Binding affinity towards glucagon receptor determined by reduction in binding of 125 I-glucagon to the murine glucagon receptor (mGLUR) expressed on ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGlucagon receptor(Mouse)
Sanofi-Aventis Deutschland

Curated by ChEMBL
LigandPNGBDBM50075758(4-[5-(4-Chloro-phenyl)-3-(4-methoxy-phenyl)-1H-pyr...)
Affinity DataIC50: 240nMAssay Description:Binding affinity towards glucagon receptor determined by reduction in binding of 125 I-glucagon to the murine glucagon receptor (mGLUR) expressed on ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGlucagon receptor(Mouse)
Sanofi-Aventis Deutschland

Curated by ChEMBL
LigandPNGBDBM50075775(4-[3-(5-Bromo-2-propoxy-phenyl)-5-(4-chloro-phenyl...)
Affinity DataIC50: 250nMAssay Description:Binding affinity towards glucagon receptor determined by reduction in binding of 125 I-glucagon to the murine glucagon receptor (mGLUR) expressed on ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGlucagon receptor(Mouse)
Sanofi-Aventis Deutschland

Curated by ChEMBL
LigandPNGBDBM50075749(4-[3-(2-Allyloxy-phenyl)-5-(4-chloro-phenyl)-1H-py...)
Affinity DataIC50: 270nMAssay Description:Binding affinity towards glucagon receptor determined by reduction in binding of 125 I-glucagon to the murine glucagon receptor (mGLUR) expressed on ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
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